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09/2009 - Državni zavod za intelektualno vlasništvo

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HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601 3463<br />

(31) 856079 P (32) 02.11.2006. (33) US<br />

(54) NICOTINIC ACETYLCHOLINE RECEPTORSUB-TYPE<br />

SELECTIVE AMIDES OF DIAZABICYCLOALKANES<br />

(71) Targacept, Inc., 200 East First Street, Suite 300, Winston-Salem,<br />

NC 27101-4165, US<br />

(72) MAZUROV, Anatoly, 3704 Timberoak Drive, Greensboro, North<br />

Carolina 27410, US<br />

MIAO, Lan, 226 March Ferry Road, Advance, North Carolina 27006,<br />

US<br />

XIAO, Yun-de, 2079 Waterford Village Drive, Clemmons, North<br />

Carolina 27012, US<br />

HAMMOND, Philip S., 1162 Bradley Road, Pinnacle, North Carolina<br />

27043, US<br />

MILLER, Craig H., 1564 Sharon Road, Winston-salem, North<br />

Carolina 27103, US<br />

AKIREDDY, Srinivisa Rao, 5829 Fox Point Circle, Winston-salem,<br />

North Carolina 27104, US<br />

MURTHY, V. Srinivasa, 595 Stonebridge Drive, Winston-salem,<br />

North Carolina 27104, US<br />

WHITAKER, Regina C., 3257 U.S. Hwy. 158, Mocksville, North<br />

Carolina 27028, US<br />

BREINING, Scott R., 2363 Rosewood Avenue, Winston-salem,<br />

North Carolina 27103, US<br />

MELVIN, Matt S., 2074 Craig Street, Winston-salem, North Carolina<br />

27103, US<br />

(51) MKP<br />

C07D 473/06 (2006.01) (97) EP 2<strong>09</strong>7415 *<br />

C07D 473/04 (2006.01)<br />

A61K 31/495 (2006.01)<br />

A61P 25/00 (2006.01)<br />

(86) PCT/EP2007011172 19.12.2007.<br />

(96) EP 07856895.3 19.12.2007.<br />

(87) WO2008077557, 03.07.2008. 200827<br />

(97) EP 2<strong>09</strong>7415, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

(31) 06026739 (32) 22.12.2006. (33) EP<br />

945248 P 20.06.2007. US<br />

(54) 8-ETHINYLXANTHINE DERIVATIVES AS SELECTIVE A2A<br />

RECEPTOR ANTAGONISTS<br />

(71) Schwarz Pharma AG, Alfred-Nobel-Strasse 10, 40789 Monheim,<br />

DE<br />

(72) MUELLER, Christa, Buschstrasse 52, 53113 Bonn, DE<br />

HOCKEMEYER, Joerg, Bonner Talweg 30, 53113 Bonn, DE<br />

TZVETKOV, Nikolay, Steinweg 44, 53121 Bonn, DE<br />

BURBIEL, Joachim, Ahrweg 95, 53347 Alfter, DE<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>9802 *<br />

(86) PCT/GB2007050697 19.11.2007.<br />

(96) EP 078249<strong>09</strong>.1 19.11.2007.<br />

(87) WO2008065444, 05.06.2008. 200823<br />

(97) EP 2<strong>09</strong>9802, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 0623750 (32) 28.11.2006. (33) GB<br />

(54) SUBSTITUTED QUINAZOLINES<br />

(71) Shire LLC, 9200 Brookfield Court, Florence, KY 41042, US<br />

(72) FRANKLIN, Richard, Shire LLC 9200 Brookfiled Court, Florence,<br />

Kentucky 41042, US<br />

GOLDING, Bernard, Shire LLC 9200 Brookfield Court, Florence,<br />

Kentucky 41042, US<br />

YU, Kin T., 55 Corporate Drive, Bridgewater, New Jersey 08807,<br />

US<br />

ZILBERSTEIN, Asher, c/o sanofi-aventis 1041 Route 202-206 Mail<br />

Code: BRW-303A, Bridgewater, New Jersey 08807, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>47<strong>09</strong> *<br />

A61K 31/505 (2006.01)<br />

A61P 29/00 (2006.01)<br />

A61P 25/22 (2006.01)<br />

A61P 25/24 (2006.01)<br />

A61P 25/30 (2006.01)<br />

(86) PCT/US2007078605 17.<strong>09</strong>.2007.<br />

(96) EP 07842582.4 17.<strong>09</strong>.2007.<br />

(87) WO2008036579, 27.03.2008. 200813<br />

(97) EP 2<strong>09</strong>47<strong>09</strong>, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 826264 P (32) 20.<strong>09</strong>.2006. (33) US<br />

(54) THIAZOLE PYRAZOLOPYRIMIDINES AS CRF1 RECEPTOR<br />

ANTAGONISTS<br />

(71) ELI LILLY AND COMPANY, Lilly Corporate Center, Indianapolis,<br />

Indiana 46285, US<br />

(72) CHEN, Zhaogen, 10532 Titan Run, Carmel, Indiana 46032, US<br />

HAMDOUCHI, Chafiq, Hamdouchi, 14469 Twin Oaks Drive,<br />

Carmel, Indiana 46032, US<br />

HEMBRE, Erik, James, 1332 North New Jersey Street,<br />

Indianapolis, Indiana 46202, US<br />

HIPSKIND, Philip, Arthur, 4255 Cabin Court, New Palestine,<br />

Indiana 46163, US<br />

MYERS, Jason, Kenneth, 8021 Springwater Circle, Indianapolis,<br />

Indiana 46256, US<br />

TAKAKUWA, Takako, 7653 Germander Lane, Indianapolis, Indiana<br />

46237, US<br />

TOTH, James, Lee, 4642 South 625 West, Knightstown, Indiana<br />

46148, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>9803 *<br />

C07D 495/04 (2006.01)<br />

A61K 31/495 (2006.01)<br />

A61K 31/53 (2006.01)<br />

A61P 35/00 (2006.01)<br />

A61P 29/00 (2006.01)<br />

(86) PCT/US2007024364 20.11.2007.<br />

(96) EP 07853151.4 20.11.2007.<br />

(87) WO2008063669, 29.05.2008. 200822<br />

(97) EP 2<strong>09</strong>9803, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 860155 P (32) 20.11.2006. (33) US<br />

(54) HETEROBICYCLIC MATRIX METALLOPROTEASE INHIBITORS<br />

(71) Alantos Pharmaceuticals Holding, Inc., M/s 28-2-C One Amgen<br />

Center Drive, Thousand Oaks, CA 91320-1799, US<br />

(72) BLUHM, Harald, Dreihausener Weg 2, 59757 Arnsberg-Neheim, DE<br />

HOCHGÜRTEL, Matthias, Lavendelweg 22, 69198 Schriesheim,<br />

DE<br />

KROTH, Heiko, Marie-Curie-Weg 3, 69181 Leimen, DE<br />

ESSERS, Michael, Kalmuentener Strasse 81b, 51467 Bergisch<br />

Gladbach, DE<br />

GEGE, Christian, Elsenzstr. 7, 69256 Mauer, DE<br />

RICHTER, Frank, Muehlingstrasse 15, 69121 Handschuhsheim, DE<br />

TAVERAS, Arthur, 6 Joslin Lane, Southborough, Massachusetts<br />

01772, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>4708 *<br />

A61K 31/4985 (2006.01)<br />

A61P 19/02 (2006.01)<br />

(86) PCT/US2007078103 11.<strong>09</strong>.2007.<br />

(96) EP 07842207.8 11.<strong>09</strong>.2007.<br />

(87) WO2008033798, 20.03.2008. 200812<br />

(97) EP 2<strong>09</strong>4708, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 825168 P (32) 11.<strong>09</strong>.2006. (33) US<br />

(54) A PYRROLOPYRAZIN AS SYK-KINASE INHIBITOR<br />

(71) Sanofi-Aventis, 174 Avenue de France, 75013 Paris, FR<br />

(72) GILLESPY, Timothy A., 55 Corporate Drive, Bridgewater, New<br />

Jersey 08807, US<br />

EYNOTT, Paul, 55 Corporate Drive, Bridgewater, New Jersey<br />

08807, US<br />

ALLEN, Eli<strong>za</strong>beth M., 55 Corporate Drive, Bridgewater, New Jersey<br />

08807, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>4707 *<br />

C07D 495/04 (2006.01)<br />

A61K 31/495 (2006.01)<br />

A61K 31/53 (2006.01)<br />

A61P 35/00 (2006.01)<br />

A61P 29/00 (2006.01)<br />

(86) PCT/US2007024365 20.11.2007.<br />

(96) EP 07853152.2 20.11.2007.<br />

(87) WO2008063670, 29.05.2008. 200822<br />

(97) EP 2<strong>09</strong>4707, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 860155 P (32) 20.11.2006. (33) US<br />

(54) HETEROBICYCLIC MATRIX METALLOPROTEASE INHIBITORS<br />

(71) Alantos Pharmaceuticals Holding, Inc., M/s 28-2-C One Amgen<br />

Center Drive, Thousand Oaks, CA 91320-1799, US<br />

(72) HOCHGÜRTEL, Matthias, Lavendelweg 22, 69198 Schriesheim,<br />

DE<br />

ISSN 1331-2030

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