09/2009 - Državni zavod za intelektualno vlasništvo

3462 HR - Patenti - Hrvatski glasnik intelektualnog vlasništva 16, 2009, 9, 3373 – 3601
(54) PYRROLO [2, 3-B]PYRIDINE DERIVATIVES AS KINASE
MODULATORS
(71) PLEXXIKON, INC., 91 Bolivar Drive, Suite A, Berkeley, CA 94710,
US
(72) SPEVAK, Wayne, 1585 Campus Drive, Berkeley, CA 94708, US
CHO, Hanna, 425 Orange Street, 314, Oakland, CA 94610, US
IBRAHIM, Prabha N., 3380 Lubich Drive, Mountain View, CA
94040, US
SHI, Shenghua, 3979 Via Cangrejo, San Diego, CA 92130, US
MAMO, Shumeye, 3000 Courtland Avenue, Oakland, CA 94619,
US
GILLETTE, Sam, 1042 Underhills Road, Oakland, CA 94610, US
ZHU, Hongyao, 91 Bolivar Drive, Suite A, Berkeley, CA 94710, US
(51) MKP
C07D 471/04 (2006.01) (97) EP 2094699 *
A61K 31/437 (2006.01)
A61P 35/00 (2006.01)
(86) PCT/FR2007001651 10.10.2007.
(96) EP 07858418.2 10.10.2007.
(87) WO2008046982, 24.04.2008. 200817
(97) EP 2094699, 02.09.2009. 200936, Fr
(31) 0608924 (32) 12.10.2006. (33) FR
(54) NEW IMIDAZOLONE DERIVATIVES, PREPARATION THEREOF
AS DRUGS, PHARMACEUTICAL COMPOSITIONS, AND USE
THEREOF AS PROTEIN KINASE INHIBITORS, IN PARTICULAR
CDC7
(71) Sanofi-Aventis, 174 Avenue de France, 75013 Paris, FR
(72) LEROY, Vincent, Sanofi-Aventis Département des Brevets 174
Avenue de France, 75013 Paris, FR
BACQUE, Eric, Sanofi-Aventis Département des Brevets 174
Avenue de France, 75013 Paris, FR
CONSEILLER, Emmanuel, Sanofi-Aventis Département des
Brevets 174 Avenue de France, 75013 Paris, FR
STEINMETZ, Anke, Sanofi-Aventis Département des Brevets 174
Avenue de France, 75013 Paris, FR
RONAN, Baptiste, Sanofi-Aventis Département des Brevets 174
Avenue de France, 75013 Paris, FR
LETALLEC, Jean-Philippe, Sanofi-Aventis Département des
Brevets 174 Avenue de France, 75013 Paris, FR
(51) MKP
C07D 471/04 (2006.01) (97) EP 2094700 *
A61K 31/4745 (2006.01)
A61P 35/00 (2006.01)
(86) PCT/US2007084893 16.11.2007.
(96) EP 07864492.9 16.11.2007.
(87) WO2008064093, 29.05.2008. 200822
(97) EP 2094700, 02.09.2009. 200936, En
(31) 866483 P (32) 20.11.2006. (33) US
(54) SALTS AND CRYSTALL FORMS OF 2-METHYL-2-[4-(3-
METHYL-2-OXO-8-QUINOLIN-3-YL-2,3-DIHYDRO-IMIDAZO[4,5-
C]QUINOLIN-1-YL)-PHENYL]-PROPIONITRILE
(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
(72) STOWASSER, Frank, Wieladinger Strasse 3, 79730 Murg, DE
BÄNZIGER, Markus, Dahlienstrasse 27, 4416 Bubendorf, CH
GARAD, Sudhakar Devidasrao, 36 Jonathan Lane, Malden,
Massachusetts 02148, US
(51) MKP
C07D 471/04 (2006.01) (97) EP 2086975 *
A61K 31/4375 (2006.01)
A61P 3/06 (2006.01)
(86) PCT/US2007084927 16.11.2007.
(96) EP 07864519.9 16.11.2007.
(87) WO2008064107, 29.05.2008. 200822
(97) EP 2086975, 12.08.2009. 200933, En
(31) 860202 P (32) 20.11.2006. (33) US
(54) 7,8-DIHYDRO-1,6-NAPHTHYRIDIN-5(6H)-ONES AND RELATED
BICYCLIC COMPOUNDS AS INHIBITORS OF DIPEPTIDYL
PEPTIDASE IV AND METHODS
(71) Bristol-Myers Squibb Company, Route 206 and Province Line
Road, Princeton, NJ 08543-4000, US
(72) FEVIG, John M., Bristol-Myers Squibb Company 311 Pennington-
Rocky Hill Road, Pennington, NJ 08534, US
FENG, Jianxin, Bristol-Myers Squibb Company 311 Pennington-
Rocky Hill Road, Hopewell, NJ 08534, US
(51) MKP
C07D 471/04 (2006.01) (97) EP 2086972 *
A61K 31/437 (2006.01)
(86) PCT/US2007085289 20.11.2007.
(96) EP 07864681.7 20.11.2007.
(87) WO2008064255, 29.05.2008. 200822
(97) EP 2086972, 12.08.2009. 200933, En
(31) 860749 P (32) 22.11.2006. (33) US
(54) COMPOUNDS MODULATING C-FMS AND/OR C-KIT ACTIVITY
AND USES THEREFOR
(71) PLEXXIKON, INC., 91 Bolivar Drive, Suite A, Berkeley, CA 94710,
US
(72) ZHANG, Chao, 397 Springfield Plaza, Moraga, CA 94556, US
ZHANG, Jiazhong, 1469 Bellevue Avenue, Apt. 211, Burlingame,
CA 94010, US
IBRAHIM, Prabha N., 3380 Lubich Drive, Mountain View, CA
94040, US
ARTIS, Dean R., 50 Arlmont Drive, Kensington, CA 94707, US
BREMER, Ryan, 476 Weldon Avenue Apt. 3, Oakland, CA 94610,
US
WU, Guoxian, 240 Ventura Avenue, Palo Alto, CA 94306, US
ZHU, Hongyao, 91 Bolivar Drive Suite A, Berkeley, CA 94710, US
NESPI, Marika, 564 San Luis Road, Berkeley, CA 94707, US
(51) MKP
C07D 471/04 (2006.01) (97) EP 2094701 *
A61K 31/437 (2006.01)
A61P 25/00 (2006.01)
A61P 29/00 (2006.01)
A61P 35/00 (2006.01)
(86) PCT/US2007088412 20.12.2007.
(96) EP 07871726.1 20.12.2007.
(87) WO2008080001, 03.07.2008. 200827
(97) EP 2094701, 02.09.2009. 200936, En
(31) 877052 P (32) 21.12.2006. (33) US
(54) COMPOUNDS AND METHODS FOR KINASE MODULATION,
AND INDICATIONS THEREFOR
(71) PLEXXIKON, INC., 91 Bolivar Drive, Suite A, Berkeley, CA 94710,
US
(72) IBRAHIM, Prabha N., 3380 Lubich Drive, Mountain View, CA
94040, US
BREMER, Ryan, 476 Weldon Avenue, Apt. 3, Oakland, CA 94610,
US
ZHANG, Chao, 397 Springfield Plaza, Moraga, CA 94556, US
ZHANG, Jiazhong, 888 Foster City Blvd., Apt. Q4, Foster City, CA
94404, US
HIRTH, Klaus-Peter, 334 Collingwood Street, San Francisco, CA
94114, US
WU, Guoxian, 240 Ventura Avenue, Palo Alto, CA 94306, US
ZHU, Hongyao, 91 Bolivar Drive, Suite A, Berkeley, CA 94710, US
(51) MKP
C07D 471/04 (2006.01) (97) EP 2020410
A61K 31/519 (2006.01)
A61P 35/00 (2006.01)
(96) EP 08017944.3 29.06.2006.
(97) EP 2020410, 04.02.2009. 200906, Fr
(31) 0507032 (32) 01.07.2005. (33) FR
(54) Pyrido[2,3d]pyrimidine derivatives, process for their
preparation and their therapeutical use
(71) sanofi-aventis, 174, Avenue de France, 75013 Paris, FR
(72) Bourrie, Bernard, 678 Rue Colline, 34980 Saint Gely du Fesc, FR
Casellas, Pierre, 10 Rue Carl von Linné, 34090 Montpellier, FR
Jegham, Samir, 206 Rue des Asphodeles, 34980 Montpellier, FR
Muneaux, Claude, Chemin Perayrols, 34270 Les Matelles, FR
Perreaut, Pierre, 110 Allée des Peupliers, 34980 Saint Clément de
Riviere, FR
(51) MKP
C07D 471/08 (2006.01) (97) EP 2094703 *
A61P 25/00 (2006.01)
A61K 31/407 (2006.01)
C07D 487/04 (2006.01)
(86) PCT/US2007083330 01.11.2007.
(96) EP 07863786.5 01.11.2007.
(87) WO2008057938, 15.05.2008. 200820
(97) EP 2094703, 02.09.2009. 200936, En
ISSN 1331-2030