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09/2009 - Državni zavod za intelektualno vlasništvo

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3460 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />

(97) EP 2<strong>09</strong>1949, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) 0625647 (32) 21.12.2006. (33) GB<br />

0707615 19.04.2007. GB<br />

(54) INDOLE DERIVATIVES AS S1P1 RECEPTOR AGONISTS<br />

(71) Glaxo Group Limited, Glaxo Wellcome House Berkeley Avenue,<br />

Greenford Middlesex UB6 0NN, GB<br />

(72) AHMED, Mahmood, GlaxoSmithKline Biopolis at One-North The<br />

Helios Block 03-01/02 11 Biopolis Way, Singapore 138667, SG<br />

MYATT, James, GlaxoSmithKline New Frontiers Science Park<br />

South Third Avenue, Harlow Essex CM19 5AW, GB<br />

NORTON, David, GlaxoSmithKline New Frontiers Science Park<br />

South Third Avenue, Harlow Essex CM19 5AW, GB<br />

RIVERS, Dean Andrew, GlaxoSmithKline Biopolis at One-North The<br />

Helios Block 03-01/02 11 Biopolis Way, Singapore 138667, SG<br />

(51) MKP<br />

C07D 413/10 (2006.01) (97) EP 2<strong>09</strong>1950 *<br />

C07D 413/14 (2006.01)<br />

A61K 31/4245 (2006.01)<br />

A61P 37/00 (2006.01)<br />

(86) PCT/EP2007064181 19.12.2007.<br />

(96) EP 07857804.4 19.12.2007.<br />

(87) WO2008074820, 26.06.2008. 200826<br />

(97) EP 2<strong>09</strong>1950, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) 0625648 (32) 21.12.2006. (33) GB<br />

(54) OXADIAZOLE DERIVATIVES AS S1P1 RECEPTOR AGONISTS<br />

(71) Glaxo Group Limited, Glaxo Wellcome House Berkeley Avenue,<br />

Greenford Middlesex UB6 0NN, GB<br />

(72) AHMED, Mahmood, GlaxoSmithKline Biopolis at One-North The<br />

Helios Block 03-01/02 11 Biopolis Way, Singapore 138667, SG<br />

MYATT, James, GlaxoSmithKline New Frontiers Science Park<br />

South Third Avenue, Harlow Essex CM19 5AW, GB<br />

NORTON, David, GlaxoSmithKline New Frontiers Science Park<br />

South Third Avenue, Harlow Essex CM19 5AW, GB<br />

RIVERS, Dean Andrew, GlaxoSmithKline Biopolis at One-North The<br />

Helios Block 03-01/02 11 Biopolis Way, Singapore 138667, SG<br />

(51) MKP<br />

C07D 413/12 (2006.01) (97) EP 2<strong>09</strong>9792 *<br />

C07D 491/04 (2006.01)<br />

C07D 495/04 (2006.01)<br />

C07D 495/14 (2006.01)<br />

C07D 495/22 (2006.01)<br />

A61K 31/519 (2006.01)<br />

A61P 29/00 (2006.01)<br />

(86) PCT/US2007024362 20.11.2007.<br />

(96) EP 07853149.8 20.11.2007.<br />

(87) WO2008063667, 29.05.2008. 200822<br />

(97) EP 2<strong>09</strong>9792, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 860195 P (32) 20.11.2006. (33) US<br />

(54) HETEROTRICYCLIC METALLOPROTEASE INHIBITORS<br />

(71) Alantos Pharmaceuticals Holding, Inc., M/s 28-2-C One Amgen<br />

Center Drive, Thousand Oaks, CA 91320-1799, US<br />

(72) GEGE, Christian, Elsenzstrasse 7, 69256 Mauer, DE<br />

CHEVRIER, Carine, Rüdigerstrasse 8, 80639 München, FR<br />

SCHNEIDER, Matthias, Adalbert-Stifter-Strasse 8, 69221<br />

Dossenheim, DE<br />

BLUHM, Harald, Bergstrasse 30c, 69221 Dossenheim, DE<br />

HOCHGÜRTEL, Matthias, Lavendelweg 22, 69198 Schriesheim,<br />

DE<br />

DENG, Hongbo, 178 Woodland Road, Southborough,<br />

Massachusetts 01772, US<br />

GALLAGHER, Brian M., 28 Orchard Street, Merrimac,<br />

Massachusetts 01860, US<br />

SUCHOLEIKI, Irving, 225 Mystic Valley Parkway, Winchester,<br />

Massachusetts 01890, US<br />

TAVERAS, Arthur, 6 Joslin Lane, Southborough, Massachusetts<br />

01772, US<br />

(51) MKP<br />

C07D 413/14 (2006.01) (97) EP 2086968 *<br />

C07D 471/04 (2006.01)<br />

A61K 31/4375 (2006.01)<br />

A61K 31/47<strong>09</strong> (2006.01)<br />

A61P 31/00 (2006.01)<br />

(86) PCT/IB2007054557 <strong>09</strong>.11.2007.<br />

(96) EP 07827038.6 <strong>09</strong>.11.2007.<br />

(87) WO2008056335, 15.05.2008. 200820<br />

(97) EP 2086968, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) PCT/IB2006/054189 (32) 10.11.2006. (33) WO<br />

(54) 5-HYDROXYMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES<br />

(71) Actelion Pharmaceuticals Ltd., Gewerbestrasse 16, 4123 Allschwil,<br />

CH<br />

(72) HUBSCHWERLEN, Christian, 15, rue de la gendarmerie, 68480<br />

Durmenach, FR<br />

PANCHAUD, Philippe, Spitzwaldstrasse 143d, 4123 Allschwil, CH<br />

SPECKLIN, Jean-Luc, 2, rue des Faisans, 68680 Kembs, FR<br />

(51) MKP<br />

C07D 413/14 (2006.01) (97) EP 2<strong>09</strong>9793 *<br />

A61K 31/454 (2006.01)<br />

A61P 3/00 (2006.01)<br />

C07D 417/14 (2006.01)<br />

(86) PCT/CA2007002139 28.11.2007.<br />

(96) EP 07845603.5 28.11.2007.<br />

(87) WO2008064474, 05.06.2008. 200823<br />

(97) EP 2<strong>09</strong>9793, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 872216 P (32) 01.12.2006. (33) US<br />

898900 P 01.02.2007. US<br />

(54) AZACYCLOALKANE DERIVATIVES AS INHIBITORS OF<br />

STEAROYL-COENZYME A DELTA-9 DESATURASE<br />

(71) Merck Frosst Canada Ltd., 16711 Trans-Canada Highway, Kirkland,<br />

Québec H9H 3L1, CA<br />

(72) LACHANCE, Nicolas, 16711 Trans-Canada Highway, Kirkland, QC<br />

H9H 3L1, CA<br />

LI, Chun Sing, 16711 Trans-Canada Highway, Kirkland, QC H9H<br />

3L1, CA<br />

LECLERC, Jean-Philippe, 16711 Trans-Canada Highway, Kirkland,<br />

QC H9H 3L1, CA<br />

RAMTOHUL, Yeeman K., 16711 Trans-Canada Highway, Kirkland,<br />

QC H9H 3L1, CA<br />

(51) MKP<br />

C07D 413/14 (2006.01) (97) EP 2<strong>09</strong>74<strong>09</strong> *<br />

A61K 31/513 (2006.01)<br />

A61P 25/00 (2006.01)<br />

A61P 19/00 (2006.01)<br />

A61P 33/00 (2006.01)<br />

A61P 35/00 (2006.01)<br />

A61P 3/00 (2006.01)<br />

(86) PCT/JP2007075380 26.12.2007.<br />

(96) EP 07860575.5 26.12.2007.<br />

(87) WO2008078837, 03.07.2008. 200827<br />

(97) EP 2<strong>09</strong>74<strong>09</strong>, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

(31) 2006357476 (32) 26.12.2006. (33) JP<br />

(54) 2-SUBSTITUTED-6-HETEROCYCLIC PYRIMIDONE<br />

DERIVATIVES AS TAU PROTEIN KINASE 1 INHBITORS<br />

(71) Mitsubishi Tanabe Pharma Corporation, 2-10, Dosho-machi 3-<br />

chome, Chuo-ku Osaka-shi Osaka 541-8505, JP<br />

Sanofi-Aventis, 174 Avenue de France, 75013 Paris, FR<br />

(72) WATANABE, Kazutoshi, c/o MITSUBISHI TANABE PHARMA<br />

CORPORATION 2-10, Dosho-machi 3-chome Chuo-ku, Osaka-shi<br />

Osaka 541-8505, JP<br />

KOHARA, Toshiyuki, c/o MITSUBISHI TANABE PHARMA<br />

CORPORATION 2-10, Dosho-machi 3-chome Chuo-ku, Osaka-shi<br />

Osaka 541-8505, JP<br />

FUKUNAGA, Kenji, c/o MITSUBISHI TANABE PHARMA<br />

CORPORATION 2-10, Dosho-machi 3-chome Chuo-ku, Osaka-shi<br />

Osaka 541-8505, JP<br />

UEHARA, Fumiaki, c/o MITSUBISHI TANABE PHARMA<br />

CORPORATION 2-10, Dosho-machi 3-chome Chuo-ku, Osaka-shi<br />

Osaka 541-8505, JP<br />

(51) MKP<br />

C07D 417/14 (2006.01) (97) EP 2<strong>09</strong>9794 *<br />

(86) PCT/US2007088124 19.12.2007.<br />

(96) EP 07869520.2 19.12.2007.<br />

(87) WO2008079873, 03.07.2008. 200827<br />

(97) EP 2<strong>09</strong>9794, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 870872 P (32) 20.12.2006. (33) US<br />

(54) THIAZOLYL COMPOUNDS USEFUL AS KINASE INHIBITORS<br />

(71) Bristol-Myers Squibb Company, P.O. Box 4000,<br />

Route 206 and Provinceline Road, Princeton, NJ 08543-4000, US<br />

(72) MARINIER, Anne, One Place Baron, Kirkland, Québec H9J 3E9,<br />

CA<br />

QUESNELLE, Claude, c/o Bristol-Myers Squibb Company Route<br />

206 & Province Line Road, Princeton, New Jersey 08543, US<br />

ISSN 1331-2030

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