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09/2009 - Državni zavod za intelektualno vlasništvo

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HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601 3459<br />

MADDUX, Todd Michael, Pfizer Global Research and Development<br />

700 Chesterfield Parkway West, Chesterfield, MO 63017, US<br />

MASFERRER, Jaime L., Pfizer Global Research and Development<br />

700 Chesterfield Parkway West, Chesterfield, MO 63017, US<br />

(51) MKP<br />

C07D 407/12 (2006.01) (97) EP 2<strong>09</strong>9790 *<br />

C07D 317/22 (2006.01)<br />

C07D 317/20 (2006.01)<br />

C07D 407/04 (2006.01)<br />

C07F 5/02 (2006.01)<br />

(86) PCT/EP2007010185 23.11.2007.<br />

(96) EP 07846785.9 23.11.2007.<br />

(87) WO2008064827, 05.06.2008. 200823<br />

(97) EP 2<strong>09</strong>9790, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 06124837 (32) 27.11.2006. (33) EP<br />

(54) PROCESS FOR PREPARING NEBIVOLOL<br />

(71) ZaCh System S.p.A., Via Lillo del Duca, 10, 20<strong>09</strong>1 Bresso (Milano),<br />

IT<br />

(72) VOLPICELLI, Raffaella, Via Nino Bixio, 31, 36100 Vicen<strong>za</strong>, IT<br />

MARAGNI, Paolo, Via Grioli 32, 46030 Virgilio (Mantova), IT<br />

COTARCA, Livius, Via Mercato, 18, 33052 Cervignano del Friuli<br />

(Udine), IT<br />

FOLETTO, Johnny, Via Molinazzo, 34/A, 37040 Arcole (Verona), IT<br />

MASSACCESI, Franco, Via Trento 1, 36045 Lonigo, IT<br />

(51) MKP<br />

C07D 407/12 (2006.01) (97) EP 2<strong>09</strong>4690 *<br />

C07D 407/14 (2006.01)<br />

C07D 417/14 (2006.01)<br />

C07D 513/04 (2006.01)<br />

A61K 31/427 (2006.01)<br />

A61P 25/00 (2006.01)<br />

(86) PCT/IB2007055326 28.12.2007.<br />

(96) EP 07859531.1 28.12.2007.<br />

(87) WO2008081399, 10.07.2008. 200828<br />

(97) EP 2<strong>09</strong>4690, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) PCT/IB2006/055042 (32) 28.12.2006. (33) WO<br />

(54) 2-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES AS OREXIN<br />

RECEPTOR ANTAGONISTS<br />

(71) Actelion Pharmaceuticals Ltd., Gewerbestrasse 16, 4123 Allschwil,<br />

CH<br />

(72) AISSAOUI, Hamed, 4, Allée des Griottes, F-68840 Pulversheim, FR<br />

BOSS, Christoph, Muesmattweg 89, CH-4123 Allschwil, CH<br />

GUDE, Markus, Grabenring 9, CH-4123 Allschwil, CH<br />

KOBERSTEIN, Ralf, Jahnstrasse 7e, 79539 Lörrach, DE<br />

SIFFERLEN, Thierry, 22, rue de l'Eglise, F-68220 Wentzwiller, FR<br />

TRACHSEL, Daniel, Wildensteinerstrasse 17, CH-4416 Bubendorf,<br />

CH<br />

(51) MKP<br />

C07D 4<strong>09</strong>/04 (2006.01) (97) EP 2086966 *<br />

C07D 4<strong>09</strong>/10 (2006.01)<br />

C07D 4<strong>09</strong>/12 (2006.01)<br />

(86) PCT/EP2007062431 15.11.2007.<br />

(96) EP 07857221.1 15.11.2007.<br />

(87) WO2008059042, 22.05.2008. 200821<br />

(97) EP 2086966, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) 0622992 (32) 17.11.2006. (33) GB<br />

0718031 14.<strong>09</strong>.2007. GB<br />

(54) 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI VIRAL<br />

AGENTS<br />

(71) SmithKline Beecham Corporation, One Franklin Pla<strong>za</strong> P.O. Box<br />

7929, Philadelphia, PA 19101, US<br />

(72) GRIMES, Richard Martin, GlaxoSmithKline Gunnels Wood Road,<br />

Stevenage Hertfordshire SG1 2NY, GB<br />

HARTLEY, Charles David, GlaxoSmithKline Gunnels Wood Road,<br />

Stevenage Hertfordshire SG1 2NY, GB<br />

MORDAUNT, Jacqueline Eli<strong>za</strong>beth, GlaxoSmithKline Gunnels<br />

Wood Road, Stevenage Hertfordshire SG1 2NY, GB<br />

SHAH, Pritom, GlaxoSmithKline Gunnels Wood Road, Stevenage<br />

Hertfordshire SG1 2NY, GB<br />

SLATER, Martin John, GlaxoSmithKline Gunnels Wood Road,<br />

Stevenage Hertfordshire SG1 2NY, GB<br />

WHITE, Gemma Victoria, GlaxoSmithKline Gunnels Wood Road,<br />

Stevenage Hertfordshire SG1 2NY, GB<br />

(51) MKP<br />

C07D 4<strong>09</strong>/04 (2006.01) (97) EP 2089385 *<br />

C07D 231/56 (2006.01)<br />

C07D 237/32 (2006.01)<br />

C07D 239/88 (2006.01)<br />

C07D 487/04 (2006.01)<br />

C07D 495/04 (2006.01)<br />

C07D 498/04 (2006.01)<br />

(86) PCT/US2007083120 31.10.2007.<br />

(96) EP 07863696.6 31.10.2007.<br />

(87) WO2008057871, 15.05.2008. 200820<br />

(97) EP 2089385, 19.08.20<strong>09</strong>. 20<strong>09</strong>34, En<br />

(31) 863837 P (32) 01.11.2006. (33) US<br />

(54) INHIBITORS OF HEPATITIS C VIRUS<br />

(71) Bristol-Myers Squibb Company, Route 206 and Province Line<br />

Road, Princeton, NJ 08543-4000, US<br />

(72) D'ANDREA, Stanley, Bristol-Myers Squibb Company 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

ZHENG, Zhizhen Barbara, Bristol-Myers Squibb Company 5<br />

Research Parkway, Wallingford, Connecticut 06492, US<br />

SCOLA, Paul Michael, Bristol-Myers Squibb Company 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

(51) MKP<br />

C07D 4<strong>09</strong>/04 (2006.01) (97) EP 2086967 *<br />

C07D 231/56 (2006.01)<br />

C07D 237/32 (2006.01)<br />

C07D 239/88 (2006.01)<br />

C07D 487/04 (2006.01)<br />

C07D 495/04 (2006.01)<br />

C07D 498/04 (2006.01)<br />

C07K 5/08 (2006.01)<br />

(86) PCT/US2007083126 31.10.2007.<br />

(96) EP 07863701.4 31.10.2007.<br />

(87) WO2008057873, 15.05.2008. 200820<br />

(97) EP 2086967, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) 863845 P (32) 01.11.2006. (33) US<br />

(54) INHIBITORS OF HEPATITIS C VIRUS<br />

(71) Bristol-Myers Squibb Company, Route 206 and Province Line<br />

Road, Princeton, NJ 08543-4000, US<br />

(72) D'ANDREA, Stanley, Bristol-Myers Squibb Company 5 Research<br />

Parkway, Wallingford, CT 06492, US<br />

SCOLA, Paul Michael, Bristol-Myers Squibb Company 5 Research<br />

Parkway, Wallingford, CT 06492, US<br />

(51) MKP<br />

C07D 4<strong>09</strong>/06 (2006.01) (97) EP 2<strong>09</strong>9791 *<br />

A61K 31/381 (2006.01)<br />

A61P 3/00 (2006.01)<br />

(86) PCT/US2007086247 03.12.2007.<br />

(96) EP 07854902.9 03.12.2007.<br />

(87) WO20080706<strong>09</strong>, 12.06.2008. 200824<br />

(97) EP 2<strong>09</strong>9791, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 868368 P (32) 04.12.2006. (33) US<br />

(54) THIENYL-CONTAINING GLYCOPYRANOSYL DERIVATIVES AS<br />

ANTIDIABETICS<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg 30, 2340 Beerse, BE<br />

Mitsubishi Tanabe Pharma Corporation, 2-10, Dosho-machi 3-<br />

chome, Chuo-ku Osaka-shi Osaka 541-8505, JP<br />

(72) COOK, Kevin L., 69 Wentworth Road, Bedminster, NJ 07921, US<br />

LIM, Heng-keang, 9 Dustin Drive, Lawrenceville, NJ 08648, US<br />

VILLANI, Frank J., 2 Pinewood Lane, Perkasie, Pennsylvania<br />

18944, US<br />

SCOTT, Lorraine, 135 Red Haven Drive, North Wales,<br />

Pennsylvania 19454, US<br />

BAUMANN, Christian Andrew, 231 Biddle Drive, Exton,<br />

Pennsylvania 19341, US<br />

(51) MKP<br />

C07D 413/04 (2006.01) (97) EP 2<strong>09</strong>1949 *<br />

C07D 413/14 (2006.01)<br />

A61K 31/405 (2006.01)<br />

A61P 37/00 (2006.01)<br />

(86) PCT/EP2007064185 19.12.2007.<br />

(96) EP 07857808.5 19.12.2007.<br />

(87) WO2008074821, 26.06.2008. 200826<br />

ISSN 1331-2030

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