09/2009 - Državni zavod za intelektualno vlasništvo
09/2009 - Državni zavod za intelektualno vlasništvo
09/2009 - Državni zavod za intelektualno vlasništvo
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3458 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />
(86) PCT/US2007024690 30.11.2007.<br />
(96) EP 07862400.4 30.11.2007.<br />
(87) WO2008069997, 12.06.2008. 200824<br />
(97) EP 2089382, 19.08.20<strong>09</strong>. 20<strong>09</strong>34, En<br />
(31) 872393 P (32) 01.12.2006. (33) US<br />
959742 P 16.07.2007. US<br />
(54) SUBSTITUTED DIAZEPAN COMPOUNDS AS OREXIN<br />
RECEPTOR ANTAGONISTS<br />
(71) Merck & Co., Inc., 126 East Lincoln Avenue, Rahway, NJ 07065-<br />
<strong>09</strong>07, US<br />
(72) BERGMAN, Jeffrey M., 126 East Lincoln Avenue, Rahway, NJ<br />
07065-<strong>09</strong>07, US<br />
BRESLIN, Michael J., 126 East Lincoln Avenue, Rahway, NJ<br />
07065-<strong>09</strong>07, US<br />
COLEMAN, Paul J., 126 East Lincoln Avenue, Rahway, NJ 07065-<br />
<strong>09</strong>07, US<br />
COX, Christopher D., 126 East Lincoln Avenue, Rahway, NJ 07065-<br />
<strong>09</strong>07, US<br />
MERCER, Swati P., 126 East Lincoln Avenue, Rahway, NJ 07065-<br />
<strong>09</strong>07, US<br />
ROECKER, Anthony J., 126 East Lincoln Avenue, Rahway, NJ<br />
07065-<strong>09</strong>07, US<br />
(51) MKP<br />
C07D 401/14 (2006.01) (97) EP 2<strong>09</strong>4688 *<br />
A61K 31/495 (2006.01)<br />
A61P 29/00 (2006.01)<br />
(86) PCT/US2007026039 20.12.2007.<br />
(96) EP 07863159.5 20.12.2007.<br />
(87) WO2008079279, 03.07.2008. 200827<br />
(97) EP 2<strong>09</strong>4688, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />
(31) 871475 P (32) 22.12.2006. (33) US<br />
(54) HETEROCYCLIC COMPOUNDS WITH CXCR3 ANTAGONIST<br />
ACTIVITY<br />
(71) SCHERING CORPORATION, 2000 Galloping Hill Road, Kenilworth,<br />
NJ 07033, US<br />
Pharmacopeia Inc., 3000 Eastpark Boulevard, Cranbury, NJ 08512,<br />
US<br />
(72) ZENG, Qingbei, 5<strong>09</strong> Cinder Road, Edison, New Jersey 08820, US<br />
ROSENBLUM, Stuart B., 16 Steven Terrace, West Orange, New<br />
Jersey 07052, US<br />
KOZLOWSKI, Joseph A., 1066 Stuart Road, Princeton, New Jersey<br />
08540, US<br />
SHIH, Neng-Yang, 2 Tyler Road, Lexington, Massachusetts 02420,<br />
US<br />
MCGUINNESS, Brian F., 16 Adams Court, Plainsboro, New Jersey<br />
08536, US<br />
HOBBS, Douglas W., 16330 Wilson Farm Drive, Chesterfield,<br />
Missouri 63005, US<br />
(51) MKP<br />
C07D 403/04 (2006.01) (97) EP 2<strong>09</strong>7405 *<br />
C07D 207/<strong>09</strong> (2006.01)<br />
C07D 417/14 (2006.01)<br />
C07D 401/14 (2006.01)<br />
C07D 403/14 (2006.01)<br />
C07D 405/14 (2006.01)<br />
C07D 4<strong>09</strong>/14 (2006.01)<br />
C07D 413/04 (2006.01)<br />
(86) PCT/US2007085218 20.11.2007.<br />
(96) EP 07871535.6 20.11.2007.<br />
(87) WO2008070447, 12.06.2008. 200824<br />
(97) EP 2<strong>09</strong>7405, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />
(31) 860614 P (32) 21.11.2006. (33) US<br />
(54) ANTI-VIRAL COMPOUNDS<br />
(71) Smithkline Beecham Corporation, One Franklin Pla<strong>za</strong> PO Box<br />
7929, Philadelphia, PA 19101, US<br />
(72) LEIVERS, Martin Robert, 91 Central Ave. 103, San Francisco, CA<br />
94117, US<br />
SCHMITZ, Franz Ulrich, 544 Marin Avenue, Mill Valley, CA 94941,<br />
US<br />
ROBERTS, Christopher Don, 1160 Granada St., Belmont, CA<br />
94002, US<br />
DEHGHANI MOHAMMAD ABADI, Ali, 4971 Ponderosa Terrace,<br />
Campbell, CA 95008, US<br />
(51) MKP<br />
C07D 403/12 (2006.01) (97) EP 2<strong>09</strong>7406 *<br />
C07D 239/34 (2006.01)<br />
A61K 31/506 (2006.01)<br />
A61P 11/00 (2006.01)<br />
A61P 11/06 (2006.01)<br />
A61P 19/00 (2006.01)<br />
A61P 19/02 (2006.01)<br />
(86) PCT/GB2007004556 28.11.2007.<br />
(96) EP 07824738.4 28.11.2007.<br />
(87) WO2008065393, 05.06.2008. 200823<br />
(97) EP 2<strong>09</strong>7406, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />
(31) 867606 P (32) 29.11.2006. (33) US<br />
(54) HYDANTOIN DERIVATIVES USED AS MMP INHIBITORS<br />
(71) Astra Zeneca AB, , S-151 85 Södertalje, SE<br />
(72) CHAPMAN, David, AstraZeneca R & D Lund, S-SE-221 87 Lund,<br />
SE<br />
GABOS, Balint, AstraZeneca R & D Lund, S-SE-221 87 Lund, SE<br />
MUNCK AF ROSENSCHOLD, Magnus, AstraZeneca R & D Lund,<br />
S-SE-221 87 Lund, SE<br />
(51) MKP<br />
C07D 403/12 (2006.01) (97) EP 2086965 *<br />
C07D 417/12 (2006.01)<br />
C07D 417/14 (2006.01)<br />
C07D 471/04 (2006.01)<br />
A61K 31/506 (2006.01)<br />
(86) PCT/US2007083334 01.11.2007.<br />
(96) EP 07844798.4 01.11.2007.<br />
(87) WO2008057940, 15.05.2008. 200820<br />
(97) EP 2086965, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />
(31) 856135 P (32) 02.11.2006. (33) US<br />
953025 P 31.07.2007. US<br />
(54) AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS<br />
INHIBITORS OF PROTEIN KINASES<br />
(71) Vertex Pharmaceuticals, Inc., 130 Waverly Street, Cambridge, MA<br />
02139, US<br />
(72) JIMENEZ, Juan-miguel, Unit 88, Milton Park, Abingdon, Oxfordshire<br />
OX14 4RY, GB<br />
COLLIER, Philip, Unit 88, Milton Park, Abingdon, Oxfordshire OX14<br />
4RY, GB<br />
MILLER, Andrew, Unit 88 Milton Park, Abingdon, Oxfordshire OX14<br />
4RY, GB<br />
(51) MKP<br />
C07D 403/14 (2006.01) (97) EP 2<strong>09</strong>9787 *<br />
C07D 471/04 (2006.01)<br />
A61K 31/506 (2006.01)<br />
(86) PCT/US2007088058 19.12.2007.<br />
(96) EP 07855256.9 19.12.2007.<br />
(87) WO2008077086, 26.06.2008. 200826<br />
(97) EP 2<strong>09</strong>9787, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />
(31) 875729 P (32) 19.12.2006. (33) US<br />
953027 P 31.07.2007. US<br />
(54) AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN<br />
KINASES<br />
(71) Vertex Pharmaceuticals, Inc., 130 Waverly Street, Cambridge, MA<br />
02139, US<br />
(72) JIMENEZ, Juan-Miguel, Unit 88 Milton Park, Abingdon Oxfordshire<br />
OX14 4RY, GB<br />
COLLIER, Philip, Unit 88, Milton Park, Abingdon Oxfordshire OX14<br />
4RY, GB<br />
MILLER, Andrew, Unit 88, Milton Park, Abingdon Oxfordshire OX14<br />
4RY, GB<br />
(51) MKP<br />
C07D 405/12 (2006.01) (97) EP 2<strong>09</strong>7407 *<br />
C07D 3<strong>09</strong>/08 (2006.01)<br />
A61K 31/4155 (2006.01)<br />
A61P 11/00 (2006.01)<br />
(86) PCT/IB2007003518 14.11.2007.<br />
(96) EP 07848899.6 14.11.2007.<br />
(87) WO2008065493, 05.06.2008. 200823<br />
(97) EP 2<strong>09</strong>7407, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />
(31) 867337 P (32) 27.11.2006. (33) US<br />
(54) PYRAZOLE ANALOGS<br />
(71) Pfizer Products Inc., Eastern Point Road, Groton,<br />
Connecticut 06340, US<br />
(72) GRANETO, Matthew J., Pfizer Global Research and Development<br />
700 Chesterfield Parkway West, Chesterfield, MO 63017, US<br />
ISSN 1331-2030