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09/2009 - Državni zavod za intelektualno vlasništvo

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3456 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />

(51) MKP<br />

C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>1942 *<br />

C07D 241/20 (2006.01)<br />

A61K 31/501 (2006.01)<br />

A61P 25/00 (2006.01)<br />

(86) PCT/EP2007060748 10.10.2007.<br />

(96) EP 07821116.6 10.10.2007.<br />

(87) WO2008043775, 17.04.2008. 200816<br />

(97) EP 2<strong>09</strong>1942, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) 06122173 (32) 12.10.2006. (33) EP<br />

(54) SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A<br />

MEDICINE<br />

(71) JANSSEN PHARMACEUTICA N.V., Turnhoutsebaan 30, 2340<br />

Beerse, BE<br />

(72) ANDRÉS-GIL, José Ignacio, Johnson & Johnson Pharmaceutical<br />

Research & Development Division of Janssen-Cilag S.A. Calle<br />

Jarama, 75 Poligono Industrial, E-45007 Toledo, ES<br />

ALCÁZAR-VACA, Manuel Jesús, Johnson & Johnson<br />

Pharmaceutical Research & Development Division of Janssen-Cilag<br />

S.A. Calle Jarama, 75 Poligono Industrial, E-45007 Toledo, ES<br />

LINARES DE LA MORENA, Maria Lourdes, Johnson & Johnson<br />

Pharmaceutical Research & Development Division of Janssen-Cilag<br />

S.A. Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />

MARTINEZ GONZALEZ, Sonia, Johnson & Johnson<br />

Pharmaceutical Research & Development Division of Janssen-Cilag<br />

S.A. Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />

OYARZABAL SANTAMARINA, Julen, C/Góngora, 12, 45280 Olias<br />

del Rey (Toledo), ES<br />

PASTOR-FERNÁNDEZ, Joaquin, Johnson & Johnson<br />

Pharmaceutical Research & Development Division of Janssen-Cilag<br />

S.A. Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />

VEGA-RAMIRO, Juan Antonio, Johnson & Johnson Pharmaceutical<br />

Research & Development Division of Janssen-Cilag S.A. Calle<br />

Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />

DELGADO-JIMÉNEZ, Francisca, Johnson & Johnson<br />

Pharmaceutical Research & Development Division of Janssen-Cilag<br />

S.A Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />

DRINKENBURG, Wilhelmus Helena Ignatius Maria, Janssen<br />

Pharmaceutica N.V. Turnhoutseweg 30, 2340 Beerse, BE<br />

(51) MKP<br />

C07D 401/12 (2006.01) (97) EP 2086961 *<br />

C07D 401/14 (2006.01)<br />

A61K 31/4427 (2006.01)<br />

(86) PCT/EP2007062274 13.11.2007.<br />

(96) EP 07822546.3 13.11.2007.<br />

(87) WO2008058961, 22.05.2008. 200821<br />

(97) EP 2086961, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) 06124131 (32) 15.11.2006. (33) EP<br />

(54) HETEROCYCLIC DERIVATIVES AS CETP INHIBITORS<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) IMASE, Hidetomo, Tsukuba Research Institute Okubo 8, Tsukuba<br />

Ibaraki 300-2611, JP<br />

KISHIDA, Masashi, Tsukuba Research Institute Okubo 8, Tsukuba<br />

Ibaraki 300-2611, JP<br />

TAHRI, Abdellah, Rue Maurice Albert Raskin 30, 1070 Anderlecht,<br />

BE<br />

VENDEVILLE, Sandrine Marie Helene, Rue du Bemel 142, 1150<br />

Woluwe-Saint-Pierre, BE<br />

(51) MKP<br />

C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>1938 *<br />

A61K 31/501 (2006.01)<br />

A61P 25/18 (2006.01)<br />

(86) PCT/EP2007063338 05.12.2007.<br />

(96) EP 07847833.6 05.12.2007.<br />

(87) WO2008068277, 12.06.2008. 200824<br />

(97) EP 2<strong>09</strong>1938, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) 06125685 (32) 08.12.2006. (33) EP<br />

(54) PIPERIDINYLAMINO-PYRIDAZINES AND THEIR USE AS FAST<br />

DISSOCIATING DOPAMINE 2 RECEPTOR ANTAGONISTS<br />

(71) JANSSEN PHARMACEUTICA N.V., Turnhoutsebaan 30, 2340<br />

Beerse, BE<br />

(72) MACDONALD, Gregor James, Janssen Pharmaceutica N.V.<br />

Turnhoutseweg 30, 2340 Beerse, BE<br />

ANDRÉS-GIL, José Ignacio, c/o Johnson & Johnson<br />

Pharmaceutical Research and Development Division of Janssen-<br />

Cilag, S.A. Calle Jarama, 75 / Poligono Industrial, 45007 Toledo,<br />

ES<br />

VAN DEN KEYBUS, Frans Alfons Maria, Janssen Pharmaceutica<br />

N.V. Turnhoutseweg 30, 2340 Beerse, BE<br />

BARTOLOMÉ-NEBREDA, José Manuel, c/o Johnson & Johnson<br />

Pharmaceutical Research and Development Division of Janssen-<br />

Cilag, S.A. Calle Jarama, 75 / Poligono Industrial, 45007 Toledo,<br />

ES<br />

VAN GOOL, Michiel Luc Maria, c/o Johnson & Johnson<br />

Pharmaceutical Research and Development Division of Janssen-<br />

Cilag, S.A. Calle Jarama, 75 / Poligono Industrial, 45007 Toledo,<br />

ES<br />

(51) MKP<br />

C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>1939 *<br />

A61K 31/473 (2006.01)<br />

A61P 25/28 (2006.01)<br />

A61P 25/30 (2006.01)<br />

A61P 25/24 (2006.01)<br />

(86) PCT/EP2007064169 19.12.2007.<br />

(96) EP 07857792.1 19.12.2007.<br />

(87) WO2008074816, 26.06.2008. 200826<br />

(97) EP 2<strong>09</strong>1939, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) 06126584 (32) 20.12.2006. (33) EP<br />

875808 P 20.12.2006. US<br />

(54) COMPOUNDS WITH A COMBINATION OF CANNABINOID-CB1<br />

ANTAGONISM AND ACETYLCHOLINESTERASE INHIBITION<br />

(71) Solvay Pharmaceuticals B.V., C.J. van Houtenlaan 36, 1381 CP<br />

Weesp, NL<br />

(72) LANGE, Josephus H.M., Solvay Pharmaceuticals B.V. IPSI<br />

Department C.J. Van Houtenlaan 36, 1381 CP Weesp, NL<br />

KRUSE, Cornelis G., Solvay Pharmaceuticals B.V. IPSI Department<br />

C.J. Van Houtenlaan 36, 1381 CP Weesp, NL<br />

SHADID, Belal, Solvay Pharmaceuticals B.V. IPSI Department C.J.<br />

Van Houtenlaan 36, 1381 CP Weesp, NL<br />

(51) MKP<br />

C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>7402 *<br />

C07D 491/04 (2006.01)<br />

A61K 31/47<strong>09</strong> (2006.01)<br />

A61K 31/4741 (2006.01)<br />

A61P 31/14 (2006.01)<br />

(86) PCT/EP2007062436 16.11.2007.<br />

(96) EP 07822656.0 16.11.2007.<br />

(87) WO2008059046, 22.05.2008. 200821<br />

(97) EP 2<strong>09</strong>7402, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

(31) 06124359 (32) 17.11.2006. (33) EP<br />

(54) MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS<br />

(71) Tibotec Pharmaceuticals Ltd., Eastgate Village, Eastgate Little<br />

Island Co Cork, IE<br />

(72) RABOISSON, Pierre Jean-Marie Bernard, Rue Jolie 3, 1331<br />

Rosieres, BE<br />

DE KOCK, Herman Augustinus, Wolfseind 10, 2370 Arendonk, BE<br />

MC GOWAN, David Craig, Van Crombrugghelaan 163, 1150<br />

Brussel, BE<br />

VAN DE VREKEN, Wim, Willem Van Doornyckstraat 49, 9120<br />

Haasdonk, BE<br />

HU, Lili, Vrouw van Mechelenstraat 28, 2800 Mechelen, BE<br />

(51) MKP<br />

C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>9782 *<br />

A61K 31/472 (2006.01)<br />

A61P 3/00 (2006.01)<br />

(86) PCT/EP2007064220 19.12.2007.<br />

(96) EP 07857842.4 19.12.2007.<br />

(87) WO2008074834, 26.06.2008. 200826<br />

(97) EP 2<strong>09</strong>9782, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />

(31) 0625654 (32) 21.12.2006. (33) GB<br />

(54) ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF<br />

STEAROYL-COA DESATURASE (SCD)<br />

(71) SmithKline Beecham Corporation, One Franklin Pla<strong>za</strong> P.O. Box<br />

7929, Philadelphia, PA 19101, US<br />

(72) BOUILLOT, Anne Marie Jeanne, Laboratoire GlaxoSmithKline<br />

Centre de Recherches Z.A. de Courtaboeuf 25 Avenue de Quebec,<br />

91940 Les Ulis, FR<br />

ISSN 1331-2030

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