09/2009 - Državni zavod za intelektualno vlasništvo
09/2009 - Državni zavod za intelektualno vlasništvo
09/2009 - Državni zavod za intelektualno vlasništvo
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3456 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />
(51) MKP<br />
C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>1942 *<br />
C07D 241/20 (2006.01)<br />
A61K 31/501 (2006.01)<br />
A61P 25/00 (2006.01)<br />
(86) PCT/EP2007060748 10.10.2007.<br />
(96) EP 07821116.6 10.10.2007.<br />
(87) WO2008043775, 17.04.2008. 200816<br />
(97) EP 2<strong>09</strong>1942, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />
(31) 06122173 (32) 12.10.2006. (33) EP<br />
(54) SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A<br />
MEDICINE<br />
(71) JANSSEN PHARMACEUTICA N.V., Turnhoutsebaan 30, 2340<br />
Beerse, BE<br />
(72) ANDRÉS-GIL, José Ignacio, Johnson & Johnson Pharmaceutical<br />
Research & Development Division of Janssen-Cilag S.A. Calle<br />
Jarama, 75 Poligono Industrial, E-45007 Toledo, ES<br />
ALCÁZAR-VACA, Manuel Jesús, Johnson & Johnson<br />
Pharmaceutical Research & Development Division of Janssen-Cilag<br />
S.A. Calle Jarama, 75 Poligono Industrial, E-45007 Toledo, ES<br />
LINARES DE LA MORENA, Maria Lourdes, Johnson & Johnson<br />
Pharmaceutical Research & Development Division of Janssen-Cilag<br />
S.A. Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />
MARTINEZ GONZALEZ, Sonia, Johnson & Johnson<br />
Pharmaceutical Research & Development Division of Janssen-Cilag<br />
S.A. Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />
OYARZABAL SANTAMARINA, Julen, C/Góngora, 12, 45280 Olias<br />
del Rey (Toledo), ES<br />
PASTOR-FERNÁNDEZ, Joaquin, Johnson & Johnson<br />
Pharmaceutical Research & Development Division of Janssen-Cilag<br />
S.A. Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />
VEGA-RAMIRO, Juan Antonio, Johnson & Johnson Pharmaceutical<br />
Research & Development Division of Janssen-Cilag S.A. Calle<br />
Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />
DELGADO-JIMÉNEZ, Francisca, Johnson & Johnson<br />
Pharmaceutical Research & Development Division of Janssen-Cilag<br />
S.A Calle Jarama, 75 Poligono Industrial, 45007 Toledo, ES<br />
DRINKENBURG, Wilhelmus Helena Ignatius Maria, Janssen<br />
Pharmaceutica N.V. Turnhoutseweg 30, 2340 Beerse, BE<br />
(51) MKP<br />
C07D 401/12 (2006.01) (97) EP 2086961 *<br />
C07D 401/14 (2006.01)<br />
A61K 31/4427 (2006.01)<br />
(86) PCT/EP2007062274 13.11.2007.<br />
(96) EP 07822546.3 13.11.2007.<br />
(87) WO2008058961, 22.05.2008. 200821<br />
(97) EP 2086961, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />
(31) 06124131 (32) 15.11.2006. (33) EP<br />
(54) HETEROCYCLIC DERIVATIVES AS CETP INHIBITORS<br />
(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />
(72) IMASE, Hidetomo, Tsukuba Research Institute Okubo 8, Tsukuba<br />
Ibaraki 300-2611, JP<br />
KISHIDA, Masashi, Tsukuba Research Institute Okubo 8, Tsukuba<br />
Ibaraki 300-2611, JP<br />
TAHRI, Abdellah, Rue Maurice Albert Raskin 30, 1070 Anderlecht,<br />
BE<br />
VENDEVILLE, Sandrine Marie Helene, Rue du Bemel 142, 1150<br />
Woluwe-Saint-Pierre, BE<br />
(51) MKP<br />
C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>1938 *<br />
A61K 31/501 (2006.01)<br />
A61P 25/18 (2006.01)<br />
(86) PCT/EP2007063338 05.12.2007.<br />
(96) EP 07847833.6 05.12.2007.<br />
(87) WO2008068277, 12.06.2008. 200824<br />
(97) EP 2<strong>09</strong>1938, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />
(31) 06125685 (32) 08.12.2006. (33) EP<br />
(54) PIPERIDINYLAMINO-PYRIDAZINES AND THEIR USE AS FAST<br />
DISSOCIATING DOPAMINE 2 RECEPTOR ANTAGONISTS<br />
(71) JANSSEN PHARMACEUTICA N.V., Turnhoutsebaan 30, 2340<br />
Beerse, BE<br />
(72) MACDONALD, Gregor James, Janssen Pharmaceutica N.V.<br />
Turnhoutseweg 30, 2340 Beerse, BE<br />
ANDRÉS-GIL, José Ignacio, c/o Johnson & Johnson<br />
Pharmaceutical Research and Development Division of Janssen-<br />
Cilag, S.A. Calle Jarama, 75 / Poligono Industrial, 45007 Toledo,<br />
ES<br />
VAN DEN KEYBUS, Frans Alfons Maria, Janssen Pharmaceutica<br />
N.V. Turnhoutseweg 30, 2340 Beerse, BE<br />
BARTOLOMÉ-NEBREDA, José Manuel, c/o Johnson & Johnson<br />
Pharmaceutical Research and Development Division of Janssen-<br />
Cilag, S.A. Calle Jarama, 75 / Poligono Industrial, 45007 Toledo,<br />
ES<br />
VAN GOOL, Michiel Luc Maria, c/o Johnson & Johnson<br />
Pharmaceutical Research and Development Division of Janssen-<br />
Cilag, S.A. Calle Jarama, 75 / Poligono Industrial, 45007 Toledo,<br />
ES<br />
(51) MKP<br />
C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>1939 *<br />
A61K 31/473 (2006.01)<br />
A61P 25/28 (2006.01)<br />
A61P 25/30 (2006.01)<br />
A61P 25/24 (2006.01)<br />
(86) PCT/EP2007064169 19.12.2007.<br />
(96) EP 07857792.1 19.12.2007.<br />
(87) WO2008074816, 26.06.2008. 200826<br />
(97) EP 2<strong>09</strong>1939, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />
(31) 06126584 (32) 20.12.2006. (33) EP<br />
875808 P 20.12.2006. US<br />
(54) COMPOUNDS WITH A COMBINATION OF CANNABINOID-CB1<br />
ANTAGONISM AND ACETYLCHOLINESTERASE INHIBITION<br />
(71) Solvay Pharmaceuticals B.V., C.J. van Houtenlaan 36, 1381 CP<br />
Weesp, NL<br />
(72) LANGE, Josephus H.M., Solvay Pharmaceuticals B.V. IPSI<br />
Department C.J. Van Houtenlaan 36, 1381 CP Weesp, NL<br />
KRUSE, Cornelis G., Solvay Pharmaceuticals B.V. IPSI Department<br />
C.J. Van Houtenlaan 36, 1381 CP Weesp, NL<br />
SHADID, Belal, Solvay Pharmaceuticals B.V. IPSI Department C.J.<br />
Van Houtenlaan 36, 1381 CP Weesp, NL<br />
(51) MKP<br />
C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>7402 *<br />
C07D 491/04 (2006.01)<br />
A61K 31/47<strong>09</strong> (2006.01)<br />
A61K 31/4741 (2006.01)<br />
A61P 31/14 (2006.01)<br />
(86) PCT/EP2007062436 16.11.2007.<br />
(96) EP 07822656.0 16.11.2007.<br />
(87) WO2008059046, 22.05.2008. 200821<br />
(97) EP 2<strong>09</strong>7402, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />
(31) 06124359 (32) 17.11.2006. (33) EP<br />
(54) MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS<br />
(71) Tibotec Pharmaceuticals Ltd., Eastgate Village, Eastgate Little<br />
Island Co Cork, IE<br />
(72) RABOISSON, Pierre Jean-Marie Bernard, Rue Jolie 3, 1331<br />
Rosieres, BE<br />
DE KOCK, Herman Augustinus, Wolfseind 10, 2370 Arendonk, BE<br />
MC GOWAN, David Craig, Van Crombrugghelaan 163, 1150<br />
Brussel, BE<br />
VAN DE VREKEN, Wim, Willem Van Doornyckstraat 49, 9120<br />
Haasdonk, BE<br />
HU, Lili, Vrouw van Mechelenstraat 28, 2800 Mechelen, BE<br />
(51) MKP<br />
C07D 401/12 (2006.01) (97) EP 2<strong>09</strong>9782 *<br />
A61K 31/472 (2006.01)<br />
A61P 3/00 (2006.01)<br />
(86) PCT/EP2007064220 19.12.2007.<br />
(96) EP 07857842.4 19.12.2007.<br />
(87) WO2008074834, 26.06.2008. 200826<br />
(97) EP 2<strong>09</strong>9782, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, En<br />
(31) 0625654 (32) 21.12.2006. (33) GB<br />
(54) ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF<br />
STEAROYL-COA DESATURASE (SCD)<br />
(71) SmithKline Beecham Corporation, One Franklin Pla<strong>za</strong> P.O. Box<br />
7929, Philadelphia, PA 19101, US<br />
(72) BOUILLOT, Anne Marie Jeanne, Laboratoire GlaxoSmithKline<br />
Centre de Recherches Z.A. de Courtaboeuf 25 Avenue de Quebec,<br />
91940 Les Ulis, FR<br />
ISSN 1331-2030