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09/2009 - Državni zavod za intelektualno vlasništvo

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HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601 3455<br />

(31) 852604 P (32) 18.10.2006. (33) US<br />

(54) NOVEL INHIBITORS OF CHYMASE<br />

(71) JANSSEN PHARMACEUTICA N.V., Turnhoutsebaan 30, 2340<br />

Beerse, BE<br />

(72) GRECO, Michael N., 1634 Clearbrook Road, Lansdale,<br />

Pennsylvania 19446, US<br />

HAWKINS, Michael J., 318 Heckler Street, Ambler, Pennsylvania<br />

19002, US<br />

POWELL, Eugene, 4801 Woodspring Drive, Pipersville, PA 18947-<br />

1064, US<br />

DE GARAVILLA, Lawrence, 9<strong>09</strong> Noble Drive, Downingtown,<br />

Pennsylvania 19335, US<br />

MARYANOFF, Bruce E., P.O. Box 239, New Hope, Pennsylvania<br />

18938, US<br />

(51) MKP<br />

C07D 317/58 (2006.01) (97) EP 2089373 *<br />

C07D 405/12 (2006.01)<br />

(86) PCT/JP2007069645 02.10.2007.<br />

(96) EP 07829383.4 02.10.2007.<br />

(87) WO2008044667, 17.04.2008. 200816<br />

(97) EP 2089373, 19.08.20<strong>09</strong>. 20<strong>09</strong>34, En<br />

(31) 2006271172 (32) 02.10.2006. (33) JP<br />

(54) STAT3/5 ACTIVATION INHIBITOR<br />

(71) OTSUKA PHARMACEUTICAL CO., LTD., 9, Kanda Tsukasamachi<br />

2-chome, Chiyoda-ku Tokyo 101-8535, JP<br />

(72) SEKIGUCHI, Kazuo, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

SUZUKI, Takashi, c/o OTSUKA PHARMACEUTICAL CO., LTD. 11-<br />

1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

OHBUCHI, Yutaka, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

OKUNO, Mitsuhiro, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

OHI, Naoto, c/o OTSUKA PHARMACEUTICAL CO., LTD. 11-1,<br />

Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

OHNISHI, Kenji, c/o OTSUKA PHARMACEUTICAL CO., LTD. 11-1,<br />

Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

MOTOYAMA, Masaaki, c/o OTSUKA PHARMACEUTICAL CO.,<br />

LTD. 11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

YOSHIDA, Kenji, c/o OTSUKA PHARMACEUTICAL CO., LTD. 11-<br />

1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

KODAMA, Takeshi, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

SUGIYAMA, Kazuhisa, c/o OTSUKA PHARMACEUTICAL CO.,<br />

LTD. 11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

AKAMATSU, Seiji, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

KIYONO, Kunihiko, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

YANAGIHARA, Yasuo, c/o OTSUKA PHARMACEUTICAL CO.,<br />

LTD. 11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

WATANABE, Takashi, c/o OTSUKA PHARMACEUTICAL CO.,<br />

LTD. 11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

HAYASHI, Kazuhiko, c/o OTSUKA PHARMACEUTICAL CO., LTD.<br />

11-1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

TANAKA, Hideo, c/o OTSUKA PHARMACEUTICAL CO., LTD. 11-<br />

1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

SUMIDA, Takumi, c/o OTSUKA PHARMACEUTICAL CO., LTD. 11-<br />

1, Karasaki 1-chome, Otsu-shi Shiga 520-0106, JP<br />

(51) MKP<br />

C07D 327/02 (2006.01) (97) EP 2089374 *<br />

C07C 323/20 (2006.01)<br />

(86) PCT/FR2007001831 06.11.2007.<br />

(96) EP 07870250.3 06.11.2007.<br />

(87) WO2008068403, 12.06.2008. 200824<br />

(97) EP 2089374, 19.08.20<strong>09</strong>. 20<strong>09</strong>34, Fr<br />

(31) 06<strong>09</strong>815 (32) 08.11.2006. (33) FR<br />

(54) METHOD FOR THE SYNTHESIS OF N- [3- [ (2-<br />

METHOXYPHÉNYL) SULFANY] -2- METHYLPROPY]-3,4-<br />

DIHYDRO-2H-1,5-BENZOXATHIEPIN-3-AMINE.

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