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09/2009 - Državni zavod za intelektualno vlasništvo

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3454 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />

(86) PCT/AT2007000529 23.11.2007.<br />

(96) EP 07845264.6 23.11.2007.<br />

(87) WO2008061270, 29.05.2008. 200822<br />

(97) EP 2<strong>09</strong>9773, 16.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>38, De<br />

(31) 19582006 (32) 24.11.2006. (33) AT<br />

(54) NOVEL METHOD FOR PRODUCING 4,4'-(1-METHYL-1,2-<br />

ETHANEDIYL)-BIS-(2,6-PIPERAZINEDIONE)<br />

(71) Cyathus Exquirere Pharmaforschungs Gmbh, Rudolfsplatz 2/8,<br />

1010 Wien, AT<br />

(72) KOCH, Andreas, Auf der Gugl 44, 4020 Linz, AT<br />

NEUFELLNER, Erwin, Hanriederstrasse 22, 4020 Linz, AT<br />

(51) MKP<br />

C07D 249/08 (2006.01) (97) EP 2<strong>09</strong>1926 *<br />

C07D 401/12 (2006.01)<br />

C07D 403/12 (2006.01)<br />

C07D 413/12 (2006.01)<br />

A61K 31/55 (2006.01)<br />

A61P 35/00 (2006.01)<br />

(86) PCT/US2007084154 08.11.2007.<br />

(96) EP 07844993.1 08.11.2007.<br />

(87) WO2008063912, 29.05.2008. 200822<br />

(97) EP 2<strong>09</strong>1926, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) 858964 P (32) 13.11.2006. (33) US<br />

(54) SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS<br />

KSP INHIBITORS<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) XIA, Yi, Novartis Vaccines and Diagnostics, Inc. P.O. Box 8<strong>09</strong>7,<br />

Emeryville, California 94662-8<strong>09</strong>7, US<br />

MENDENHALL, Kris G., Novartis Vaccines and Diagnostics, Inc.<br />

P.O. Box 8<strong>09</strong>7, Emeryville, California 94662-8<strong>09</strong>7, US<br />

BARSANTI, Paul A., Novartis Vaccines and Diagnostics, Inc. P.O.<br />

Box 8<strong>09</strong>7, Emeryville, California 94662-8<strong>09</strong>7, US<br />

WALTER, Annette O., Novartis Vaccines and Diagnostics, Inc. P.O.<br />

Box 8<strong>09</strong>7, Emeryville, California 94662-8<strong>09</strong>7, US<br />

DUHL, David, Novartis Vaccines and Diagnostics, Inc. P.O. Box<br />

8<strong>09</strong>7, Emeryville, California 94662-8<strong>09</strong>7, US<br />

RENHOWE, Paul A., Novartis Vaccines and Diagnostics, Inc. P.O.<br />

Box 8<strong>09</strong>7, Emeryville, California 94662-8<strong>09</strong>7, US<br />

(51) MKP<br />

C07D 261/02 (2006.01) (97) EP 2<strong>09</strong>4673 *<br />

C07D 413/12 (2006.01)<br />

A61K 31/4155 (2006.01)<br />

A61P 35/00 (2006.01)<br />

(86) PCT/US2007023941 14.11.2007.<br />

(96) EP 07840052.0 14.11.2007.<br />

(87) WO2008060569, 22.05.2008. 200821<br />

(97) EP 2<strong>09</strong>4673, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 600332 (32) 15.11.2006. (33) US<br />

(54) COMPOUNDS AND METHODS FOR INHIBITING THE<br />

INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS<br />

(71) Infinity Discovery, Inc., 780 Memorial Drive, Cambridge, MA 02139,<br />

US<br />

(72) CASTRO, Alfredo C., 43 Wildwood St., Winchester, MA 01890, US<br />

HOLSON, Edward B., 66 Forest St., Newton Highlands, MA 02461,<br />

US<br />

HOPKINS, Brian T., 169 Washington St. 13, Newton, MA 02458,<br />

US<br />

KONEY, Nii O., 276 Chestnut Hill Ave. 2, Brighton, MA 02135, US<br />

SNYDER, Daniel A., 373 Highland Ave. 312, Somerville, MA 02144,<br />

US<br />

TIBBITTS, Thomas T., 67 Graniteville Road, Westford, MA 01886-<br />

2233, US<br />

(51) MKP<br />

C07D 271/06 (2006.01) (97) EP 2014653<br />

C07D 413/10 (2006.01)<br />

C07D 413/14 (2006.01)<br />

A61K 31/4245 (2006.01)<br />

A61P 29/00 (2006.01)<br />

A61P 37/06 (2006.01)<br />

(96) EP 07290748.8 15.06.2007.<br />

(97) EP 2014653, 14.01.20<strong>09</strong>. 20<strong>09</strong>03, En<br />

(54) Novel dicarboxylic acid derivatives as S1P1 receptor agonists<br />

(71) BIOPROJET, 30, rue des Francs-Bourgeois, 75003 Paris, FR<br />

Sun Pharma Advanced Research Company Limited, 17/B Mahal<br />

Industrial Estate Off Mahakali Caves Road, Andheri (East) Mumbai<br />

400 <strong>09</strong>3, IN<br />

(72) Capet, Marc, Les Petites Rivieres, 35520 Melesse, FR<br />

Levoin, Nicolas, 58 Avenue du Général de Gaulle, 35310 Mordelles,<br />

FR<br />

Berrebi-Bertrand, Isabelle, 11 rue de Vergéal, 35740 Pace, FR<br />

Robert, Philippe, 9 Chemin de la Reine Iseult, 35740 Pace, FR<br />

Schwartz, Jean-Charles, 9 Villa Seurat, 75014 Paris, FR<br />

Lecomte, Jeanne-Marie, 30 rue des Francs-Bourgeois, 75003 Paris,<br />

FR<br />

Aradhye, Jayraj Dilipbhai, E/58, Ayodhyanagar Society VIP Road,<br />

Karelibaugh Baroda 390018, IN<br />

Pillai, Muthukumaran Natarajan, C/106, Shantivan society, New<br />

Sama Road Near Abilasha, Char Rastha Baroda 390008, IN<br />

Panchal, Bhavesh Mohanbhai, 20, Gokul Park B/H Govardham<br />

Society - Opp. APC, Valabh Vidyanagar 388120, IN<br />

Jivani, Jignesh Kantilal, "Jignesh" - 10, Gopalnagar Rajkot 360 002,<br />

IN<br />

Samanta, Biswajit, 104, Akhand Sagar Appartment Near PF Office,<br />

Akota Baroda 390 020, IN<br />

Pal, Ranjan Kumar, A/4 Shreeji Park Duplex-Opp., L & T Colony<br />

B/H Nandanvan Society New Sama Road, Baroda 390 008, IN<br />

Thennati, Rajamannar, G-114-G Tower Avishkar Complex Olod<br />

Padra Road, Baroda, 390 015, IN<br />

(51) MKP<br />

C07D 295/20 (2006.01) (97) EP 2<strong>09</strong>1929 *<br />

C07C 275/44 (2006.01)<br />

C07C 335/08 (2006.01)<br />

C07C 335/16 (2006.01)<br />

C07D 471/10 (2006.01)<br />

C07D 215/40 (2006.01)<br />

C07D 317/66 (2006.01)<br />

C07D 217/06 (2006.01)<br />

C07D 471/04 (2006.01)<br />

C07D 211/52 (2006.01)<br />

C07D 307/68 (2006.01)<br />

C07D 243/08 (2006.01)<br />

C07C 335/12 (2006.01)<br />

C07C 335/14 (2006.01)<br />

C07D 413/04 (2006.01)<br />

(86) PCT/EP2007002504 21.03.2007.<br />

(96) EP 07723461.5 21.03.2007.<br />

(87) WO2007107352, 08.11.2007. 204507<br />

(97) EP 2<strong>09</strong>1929, 26.08.20<strong>09</strong>. 20<strong>09</strong>35, En<br />

(31) PCT/EP2006/002604 (32) 21.03.2006. (33) WO<br />

(54) AGENTS THAT DISRUPT CELLULAR REPLICATION AND<br />

THEIR USE IN INHIBITING PATHOLOGICAL CONDITIONS<br />

(71) The European Molecular Biology Laboratory, Meyerhofstrasse 1,<br />

69117 Heidelberg, DE<br />

(72) REID, George, Boxbergring 1, 69126 Heidelberg, DE<br />

GANNON, Frank, Karlsluststrasse 11, 69126 Heidleberg, DE<br />

POLYCARPOU-SCHWARZ, Maria, Am Lindenried 25, 69118<br />

Heidelberg, DE<br />

(51) MKP<br />

C07D 307/20 (2006.01) (97) EP 2089371 *<br />

C07D 493/04 (2006.01)<br />

(86) PCT/EP2007062119 <strong>09</strong>.11.2007.<br />

(96) EP 07822416.9 <strong>09</strong>.11.2007.<br />

(87) WO2008055970, 15.05.2008. 200820<br />

(97) EP 2089371, 19.08.20<strong>09</strong>. 20<strong>09</strong>34, En<br />

(31) 06123752 (32) <strong>09</strong>.11.2006. (33) EP<br />

(54) METHODS FOR THE PREPARATION OF<br />

HEXAHYDROFUROÝ2,3-B¨FURAN-3-OL<br />

(71) Tibotec Pharmaceuticals Ltd., Eastgate Village, Eastgate Little<br />

Island Co Cork, IE<br />

(72) LEMAIRE, Sébastien François Emmanuel, avenue des pagodes,<br />

20, 1020 Bruxelles, BE<br />

HORVATH, Andras, Smalvoortstraat 46 bus 2, 2300 Turnhout, BE<br />

AELTERMAN, Wim Albert Alex, Oude Lillebaan 7, 2275 Gierle, BE<br />

RAMMELOO, Thomas Joachim Landewald, Secretaris van de<br />

Venlaan 14, Vosselaar, 2350, BE<br />

(51) MKP<br />

C07D 307/80 (2006.01) (97) EP 2<strong>09</strong>7399 *<br />

C07D 307/81 (2006.01)<br />

A61K 31/343 (2006.01)<br />

(86) PCT/US2007022244 18.10.2007.<br />

(96) EP 07839664.5 18.10.2007.<br />

(87) WO2008048668, 24.04.2008. 200817<br />

(97) EP 2<strong>09</strong>7399, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

ISSN 1331-2030

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