09/2009 - Državni zavod za intelektualno vlasništvo

3452 HR - Patenti - Hrvatski glasnik intelektualnog vlasništva 16, 2009, 9, 3373 – 3601
(54) 2-[1-PHENYL-5-HYDROXY OR METHOXY-4ALPHA-METHYL-
HEXAHYDROCLOPENTA[F]INDAZOL-5-YL]ETHYL PHENYL
DERIVATIVES AS GLUCOCORTICOID RECEPTOR LIGANDS
(71) Merck & Co., Inc., 126 East Lincoln Avenue, Rahway, NJ 07065-
0907, US
(72) BUNGARD, Christopher J., 126 East Lincoln Avenue, Rahway, NJ
07065-0907, US
MANIKOWSKI, Jesse J., 126 East Lincoln Avenue, Rahway, NJ
07065-0907, US
PERKINS, James J., 126 East Lincoln Avenue, Rahway, NJ 07065-
0907, US
MEISSNER, Robert, 126 East Lincoln Avenue, Rahway, NJ 07065-
0907, US
(86) PCT/EP2007062804 26.11.2007.
(96) EP 07822860.8 26.11.2007.
(87) WO2008065068, 05.06.2008. 200823
(97) EP 2097386, 09.09.2009. 200937, En
(31) 06124802 (32) 27.11.2006. (33) EP
(54) SUBSTITUTED DIHYDROIMIDAZOLES AND THEIR USE IN THE
TREATMENT OF TUMORS
(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
(72) CHAMOIN, Sylvie, 87A, avenue de Bâle, 68300 Saint Louis, FR
ROTH, Hans-Jörg, Malvenweg 6, 5264 Gipf-Oberfrick, CH
ZIMMERMANN, Juerg, Schönenbachstr. 20, 4153 Reinach, CH
ZOLLER, Thomas, 19, rue des Coquelicots, 68280 Andolsheim, FR
(51) MKP
C07D 231/56 (2006.01) (97) EP 2099767 *
C07D 401/12 (2006.01)
C07D 403/12 (2006.01)
C07D 409/12 (2006.01)
A61K 31/416 (2006.01)
A61P 29/02 (2006.01)
(86) PCT/US2007083085 31.10.2007.
(96) EP 07854528.2 31.10.2007.
(87) WO2008057857, 15.05.2008. 200820
(97) EP 2099767, 16.09.2009. 200938, En
(31) 855953 P (32) 01.11.2006. (33) US
(54) MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1,
AND/OR NF- B ACTIVITY AND USE THEREOF
(71) Bristol-Myers Squibb Company, Route 206 and Province Line
Road, Princeton, NJ 08543-4000, US
(72) SHEPPECK, James E., Bristol-Myers Squibb Company Route 206
& Province Line Road, Princeton, New Jersey 08543, US
GILMORE, John L., Bristol-Myers Squibb Company Route 206 &
Province Line Road, Princeton, New Jersey 08543, US
DHAR, T.G. Murali, Bristol-Myers Squibb Company Route 206 &
Province Line Road, Princeton, New Jersey 08543, US
XIAO, Hai-Yun, Bristol-Myers Squibb Company Route 206 &
Province Line Road, Princeton, New Jersey 08543, US
WANG, Jianmin, 1208 Brook Circle, Blacksburg, Virginia 24060, US
YANG, Bingwei Vera, Bristol-Myers Squibb Company Route 206 &
Province Line Road, Princeton, New Jersey 08543, US
DOWEYKO, Lidia M., Bristol-Myers Squibb Company Route 206 &
Province Line Road, Princeton, New Jersey 08543, US
(51) MKP
C07D 231/56 (2006.01) (97) EP 2091922 *
C07D 401/10 (2006.01)
C07D 403/10 (2006.01)
A61K 31/416 (2006.01)
A61P 5/44 (2006.01)
(86) PCT/US2007022449 23.10.2007.
(96) EP 07867264.9 23.10.2007.
(87) WO2008060391, 22.05.2008. 200821
(97) EP 2091922, 26.08.2009. 200935, En
(31) 853655 P (32) 23.10.2006. (33) US
923337 P 13.04.2007. US
(54) 2-[1-PHENYL-5-HYDROXY-4ALPHA-METHYL-
HEXAHYDROCYCLOPENTA[F]INDAZOL-5-YL]ETHYL PHENYL
DERIVATIVES AS GLUCOCORTICOID RECEPTOR LIGANDS
(71) Merck & Co., Inc., 126 East Lincoln Avenue, Rahway, NJ 07065-
0907, US
(72) BUNGARD, Christopher J., 126 East Lincoln Avenue, Rahway, NJ
07065-0907, US
MANIKOWSKI, Jesse J., 126 East Lincoln Avenue, Rahway, NJ
07065-0907, US
PERKINS, James J., 126 East Lincoln Avenue, Rahway, NJ 07065-
0907, US
MEISSNER, Robert, 126 East Lincoln Avenue, Rahway, NJ 07065-
0907, US
(51) MKP
C07D 233/40 (2006.01) (97) EP 2097386 *
C07D 401/12 (2006.01)
C07D 403/06 (2006.01)
C07D 403/12 (2006.01)
C07D 403/14 (2006.01)
C07D 405/12 (2006.01)
A61K 31/4178 (2006.01)
A61P 35/00 (2006.01)
(51) MKP
C07D 233/64 (2006.01) (97) EP 2099768 *
C07D 241/04 (2006.01)
C07D 241/08 (2006.01)
C07D 277/28 (2006.01)
C07D 285/12 (2006.01)
C07C 237/20 (2006.01)
C07F 9/09 (2006.01)
A61K 31/426 (2006.01)
A61K 31/433 (2006.01)
A61K 31/661 (2006.01)
A61K 31/167 (2006.01)
A61P 25/28 (2006.01)
(86) PCT/US2007017384 02.08.2007.
(96) EP 07811077.2 02.08.2007.
(87) WO2008019090, 14.02.2008. 200807
(97) EP 2099768, 16.09.2009. 200938, En
(31) 821432 P (32) 04.08.2006. (33) US
821425 P 04.08.2006. US
827941 P 03.10.2006. US
827928 P 03.10.2006. US
(54) AGONISTS OF THE SPHINGOSINE-1-PHOSPHATE RECEPTOR
(71) Praecis Pharmaceuticals Incorporated, 830 Winter Street, Waltham,
MA 02451-1420, US
(72) EVINDAR, Ghotas, 31 Middlesex Circle, Apt. 19, Waltham, MA
02452, US
DENG, Hongfeng, 11 Brucewood Road, Acton, MA 01720, US
(51) MKP
C07D 235/14 (2006.01) (97) EP 2094670 *
C07D 401/04 (2006.01)
C07D 401/06 (2006.01)
C07D 401/12 (2006.01)
C07D 403/12 (2006.01)
C07D 405/12 (2006.01)
C07D 407/12 (2006.01)
C07D 409/12 (2006.01)
C07D 413/06 (2006.01)
C07D 413/12 (2006.01)
C07D 417/12 (2006.01)
C07D 471/04 (2006.01)
C07D 473/40 (2006.01)
C07D 487/04 (2006.01)
C07D 491/056 (2006.01)
(86) PCT/GB2007004267 08.11.2007.
(96) EP 07824500.8 08.11.2007.
(87) WO2008056150, 15.05.2008. 200820
(97) EP 2094670, 02.09.2009. 200936, En
(31) 865364 P (32) 10.11.2006. (33) US
895699 P 19.03.2007. US
947795 P 03.07.2007. US
953838 P 03.08.2007. US
(54) HETEROCYCLYC SULFONAMIDES HAVING EDG-I
ANTAGONISTIC ACTIVITY
(71) AstraZeneca AB, , 151 85 Södertälje, SE
(72) GREWAL, Gurmit, AstraZeneca R & D Boston 35 Gatehouse Drive,
Waltham, Massachusetts 02451, US
HENNESSY, Edward, AstraZeneca R & D Boston 35 Gatehouse
Drive, Waltham, Massachusetts 02451, US
KAMHI, Victor, AstraZeneca R & D Boston 35 Gatehouse Drive,
Waltham, Massachusetts 02451, US
LI, Danyang, AstraZeneca R & D Boston 35 Gatehouse Drive,
Waltham, Massachusetts 02451, US
LYNE, Paul, AstraZeneca R & D Boston 35 Gatehouse Drive,
Waltham, Massachusetts 02451, US
OZA, Vibha, AstraZeneca R & D Boston 35 Gatehouse Drive,
Waltham, Massachusetts 02451, US
SAEH, Jamal Carlos, AstraZeneca R & D Boston 35 Gatehouse
Drive, Waltham, Massachusetts 02451, US
ISSN 1331-2030