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09/2009 - Državni zavod za intelektualno vlasništvo

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HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601 3447<br />

(86) PCT/FR2007002028 10.12.2007.<br />

(96) EP 07871823.6 10.12.2007.<br />

(87) WO2008087278, 24.07.2008. 200830<br />

(97) EP 2<strong>09</strong>7374, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, Fr<br />

(31) 0610803 (32) 12.12.2006. (33) FR<br />

(54) 5-ALKYLOXY-INDOLIN-2-ONE DERIVATIVES, PREPARATION<br />

THEREOF AND APPLICATION THEREOF IN THERAPY AS<br />

SELECTIVE LIGANDS OF V2 VASOPRESSIN RECEPTORS<br />

(71) Sanofi-Aventis, 174 Avenue de France, 75013 Paris, FR<br />

(72) FOULON, Loic, c/o Sanofi-aventis Département Brevets 174,<br />

avenue de France, F-75013 Paris, FR<br />

ROCHARD, Pierrick, c/o Sanofi-aventis Département Brevets 174,<br />

avenue de France, F-75013 Paris, FR<br />

SERRADEIL-LE GAL, Claudine, c/o Sanofi-aventis Département<br />

Brevets 174, avenue de France, F-75013 Paris, FR<br />

VALETTE, Gérard, c/o Sanofi-aventis Département Brevets 174,<br />

avenue de France, F-75013 Paris, FR<br />

(51) MKP<br />

C07D 2<strong>09</strong>/42 (2006.01) (97) EP 2086933 *<br />

A61K 31/404 (2006.01)<br />

A61P 25/00 (2006.01)<br />

A61P 15/00 (2006.01)<br />

A61P 3/04 (2006.01)<br />

A61P 35/00 (2006.01)<br />

(86) PCT/FR2007001707 17.10.2007.<br />

(96) EP 07858467.9 17.10.2007.<br />

(87) WO2008049996, 02.05.2008. 200818<br />

(97) EP 2086933, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, Fr<br />

(31) 06<strong>09</strong>114 (32) 18.10.2006. (33) FR<br />

(54) NOVEL INDOLE DERIVATIVES, PROCESS FOR THE<br />

PREPARATION THEREOF AND PHARMACEUTICAL<br />

COMPOSITIONS CONTAINING THEM<br />

(71) Les Laboratoires Servier, 35, rue de Verdun, 92284 Suresnes<br />

Cedex, FR<br />

(72) MARCHAND, Pascal, 16, rue du Bois Hardy, 44100 Nantes, FR<br />

BABONNEAU, Vincent, 6, allée des Genets, 35235 Thorigne-<br />

Fouillard, FR<br />

PIESSARD, Sylvie, 147, rue Bonne Garde, 44100 Nantes, FR<br />

DUFLOS, Muriel, 37 ter, route de Nantes La Croix Rouge, F-44640<br />

Vue, FR<br />

BOUTIN, Jean Albert, 28, rue Roger Salengro, F-92150 Suresnes,<br />

FR<br />

AUDINOT, Valérie, 31, avenue Blanche de Castille, F-78300<br />

Poissy, FR<br />

DELAGRANGE, Philippe, 23, avenue Victor Hugo, 92130 Issy les<br />

Moulineaux, FR<br />

CAIGNARD, Daniel-Henri, 17, avenue des Coteaux, 95000<br />

Boisemont, FR<br />

(51) MKP<br />

C07D 2<strong>09</strong>/52 (2006.01) (97) EP 2<strong>09</strong>4657 *<br />

A61K 31/403 (2006.01)<br />

A61P 25/18 (2006.01)<br />

(86) PCT/EP2007063841 12.12.2007.<br />

(96) EP 07848087.8 12.12.2007.<br />

(87) WO2008074716, 26.06.2008. 200826<br />

(97) EP 2<strong>09</strong>4657, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 0625198 (32) 18.12.2006. (33) GB<br />

(54) AZABICYCLIC COMPOUNDS AS SEROTONINE, DOPAMINE<br />

AND NOREPINEPHRINE RE-UPTAKE INHIBITORS<br />

(71) Glaxo Group Limited, Glaxo Wellcome House Berkeley Avenue,<br />

Greenford Middlesex UB6 0NN, GB<br />

(72) BONANOMI, Giorgio, GlaxoSmithKline SpA Via Alessandro<br />

Fleming 2, 37135 Verona, IT<br />

MICHELI, Fabrizio, GlaxoSmithKline SpA Via Alessandro Fleming<br />

2, 37135 Verona, IT<br />

TERRENI, Silvia, GlaxoSmithKline SpA Via Alessandro Fleming 2,<br />

37135 Verona, IT<br />

(51) MKP<br />

C07D 2<strong>09</strong>/58 (2006.01) (97) EP 2<strong>09</strong>4658 *<br />

(86) PCT/US2007083745 06.11.2007.<br />

(96) EP 07844898.2 06.11.2007.<br />

(87) WO2008063867, 29.05.2008. 200822<br />

(97) EP 2<strong>09</strong>4658, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 866484 P (32) 20.11.2006. (33) US<br />

(54) TETRAHYDROCYCLOPENTA[B]INDOLE COMPOUNDS AS<br />

ANDROGEN RECEPTOR MODULATORS<br />

(71) ELI LILLY AND COMPANY, Lilly Corporate Center, Indianapolis,<br />

Indiana 46285, US<br />

(72) GAVARDINAS, Konstantinos, 3642 Marie Court West, Monrovia,<br />

Indiana 46157, US<br />

GREEN, Jonathan Edward, 7464 Glendale Drive, Avon, Indiana<br />

46123, US<br />

JADHAV, Prabhakar Kondaji, 7422 Fox Hollow Ridge, Zionsville,<br />

Indiana 46077, US<br />

MATTHEWS, Donald Paul, 7736 Wawasee Drive, Indianapolis,<br />

Indiana 46250, US<br />

(51) MKP<br />

C07D 211/58 (2006.01) (97) EP 2<strong>09</strong>85<strong>09</strong> *<br />

A61K 31/4468 (2006.01)<br />

A61K 31/453 (2006.01)<br />

A61K 31/454 (2006.01)<br />

A61K 31/4545 (2006.01)<br />

A61K 31/496 (2006.01)<br />

A61K 31/506 (2006.01)<br />

A61K 31/5377 (2006.01)<br />

A61P 3/04 (2006.01)<br />

A61P 3/06 (2006.01)<br />

A61P 3/10 (2006.01)<br />

A61P 9/10 (2006.01)<br />

A61P 9/12 (2006.01)<br />

A61P 25/08 (2006.01)<br />

A61P 25/14 (2006.01)<br />

A61P 25/18 (2006.01)<br />

A61P 25/20 (2006.01)<br />

A61P 25/22 (2006.01)<br />

A61P 25/24 (2006.01)<br />

A61P 25/28 (2006.01)<br />

(86) PCT/JP2007069561 05.10.2007.<br />

(96) EP 07829299.2 05.10.2007.<br />

(87) WO2008044632, 17.04.2008. 200816<br />

(97) EP 2<strong>09</strong>85<strong>09</strong>, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

(31) 2006275227 (32) 06.10.2006. (33) JP<br />

2007151270 07.06.2007. JP<br />

(54) 1-NAPHTHYL ALKYLPIPERIDINE DERIVATIVE<br />

(71) Taisho Pharmaceutical Co. Ltd., 24-1 Takata 3-chome Toshima-ku,<br />

Tokyo 170-8633, JP<br />

(72) SEKIGUCHI, Yoshinori, c/o TAISHO PHARMACEUTICAL CO.,<br />

LTD. 24-1, Takada 3-chome, Toshima-ku, Tokyo 170-8633, JP<br />

KANUMA, Kosuke, c/o TAISHO PHARMACEUTICAL CO., LTD. 24-<br />

1, Takada 3-chome, Toshima-ku, Tokyo 170-8633, JP<br />

SAKAGAMI, Kazunari, c/o TAISHO PHARMACEUTICAL CO., LTD.<br />

24-1, Takada 3-chome, Toshima-ku, Tokyo 170-8633, JP<br />

HAYASHI, Masato, c/o TAISHO PHARMACEUTICAL CO., LTD. 24-<br />

1, Takada 3-chome, Toshima-ku, Tokyo 170-8633, JP<br />

KASHIWA, Shuhei, c/o TAISHO PHARMACEUTICAL CO., LTD.<br />

24-1, Takada 3-chome, Toshima-ku, Tokyo 170-8633, JP<br />

OMODERA, Katsunori, c/o TAISHO PHARMACEUTICAL CO., LTD.<br />

24-1, Takada 3-chome, Toshima-ku, Tokyo 170-8633, JP<br />

(51) MKP<br />

C07D 213/02 (2006.01) (97) EP 2<strong>09</strong>7378 *<br />

C07D 239/34 (2006.01)<br />

C07D 239/48 (2006.01)<br />

C07D 239/50 (2006.01)<br />

C07D 251/14 (2006.01)<br />

A61K 31/44 (2006.01)<br />

A61K 31/505 (2006.01)<br />

A61K 31/506 (2006.01)<br />

A61K 31/53 (2006.01)<br />

A61P 1/16 (2006.01)<br />

A61P 9/02 (2006.01)<br />

A61P 9/04 (2006.01)<br />

A61P 9/10 (2006.01)<br />

(86) PCT/US2007083449 02.11.2007.<br />

(96) EP 07871337.7 02.11.2007.<br />

(87) WO2008105968, 04.<strong>09</strong>.2008. 200836<br />

(97) EP 2<strong>09</strong>7378, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

(31) 864178 P (32) 03.11.2006. (33) US<br />

(54) NOVEL SEH INHIBITORS AND THEIR USE<br />

(71) Smithkline Beecham Corporation, One Franklin Pla<strong>za</strong> PO Box<br />

7929, Philadelphia, PA 19101, US<br />

(72) DING, Yun, 830 Winter Street, Waltham, MA 02541, US<br />

MARINO, Joseph, Paul, Jr., 7<strong>09</strong> Swedeland Road, King Of Prussia,<br />

PA 19406, US<br />

LI, Peng, 7<strong>09</strong> Swedeland Road, King Of Prussia, PA 19406, US<br />

ISSN 1331-2030

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