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09/2009 - Državni zavod za intelektualno vlasništvo

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3464 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />

BLUHM, Harald, Dreihausener Weg 2, 59757 Arnsberg-Neheim, DE<br />

ESSERS, Michael, Kalmuentener Strasse 81b, 51467 Bergisch<br />

Gladbach, DE<br />

KROTH, Heiko, Marie-Curie-Weg 3, 69181 Leimen, DE<br />

GEGE, Christian, Elsenzstrasse 7, 69256 Mauer, DE<br />

TAVERAS, Arthur, 6 Joslin Lane, Southborough, Massachusetts<br />

01772, US<br />

D'ANDREA, Stanley, Bristol-Myers Squibb Co. 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

MEANWELL, Nicholas A., Bristol-Myers Squibb Co. 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

SCOLA, Paul Michael, Bristol-Myers Squibb Co. 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>7416 *<br />

(86) PCT/US2007025799 17.12.2007.<br />

(96) EP 07863038.1 17.12.2007.<br />

(87) WO2008076425, 26.06.2008. 200826<br />

(97) EP 2<strong>09</strong>7416, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />

(31) 875706 P (32) 18.12.2006. (33) US<br />

(54) AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL<br />

HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND<br />

USES THEREOF<br />

(71) Amgen, Inc, Patent Operations, M/S 28-2-C One Amgen Center<br />

Drive, Thousand Oaks, California 91320-1799, US<br />

(72) ALLEN, Jennifer R., 5255 Via Capote, Newbury Park, CA 91320,<br />

US<br />

BISWAS, Kaustav, 26003 Alizia Canyon Drive, Unit B, Calabasas,<br />

CA 91302, US<br />

CAO, Guo-Qiang, 4235 Via Rio, Thousand Oaks, CA 91320, US<br />

GOLDEN, Jennifer E., 3168 Tecopa Springs Lane, Simi Valley, CA<br />

93063, US<br />

MERCEDE, Stephanie, 1336 Moorpark Road, No. 183, Thousand<br />

Oaks, CA 91360, US<br />

PETERKIN, Tanya, 6130 Nevada Avenue, Apt. E311, Woodland<br />

Hills, CA 91367, US<br />

REED, Anthony, 3101 Peninsula Road, Apt. 304, Oxnard, CA<br />

93035, US<br />

TEGLEY, Christopher M., 478 Thunderhead Street, Thousand<br />

Oaks, CA 91360, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2086979 *<br />

A61K 31/5025 (2006.01)<br />

A61K 31/519 (2006.01)<br />

A61P 35/00 (2006.01)<br />

(86) PCT/US2007083773 06.11.2007.<br />

(96) EP 07863964.8 06.11.2007.<br />

(87) WO2008058126, 15.05.2008. 200820<br />

(97) EP 2086979, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) 864566 P (32) 06.11.2006. (33) US<br />

892523 P 01.03.2007. US<br />

957988 P 24.08.2007. US<br />

(54) IMIDAZOÝ1,2-B¨PYRIDAZINE AND PYRAZOLOÝ1,5-<br />

A¨PYRIMIDINE DERIVATIVES AND THEIR USE AS PROTEIN<br />

KINASE INHIBITORS<br />

(71) SuperGen, Inc., 4140 Dublin Boulevard, Suite 200, Dublin,<br />

California 94568, US<br />

(72) BEARSS, David J., 4001 Ironwood Drive, Cedar Hills, Utah 84062,<br />

US<br />

LIU, Xiao-Hui, 2028 Ashley Mesa Lane, Sandy, Utah 84<strong>09</strong>2, US<br />

VANKAYALAPATI, Hariprasad, 11558 South Sugar Berry Road,<br />

Draper, Utah 84020, US<br />

XU, Yong, 7557 Sandy Woods Lane, Midvale, Utah 84047, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2086980 *<br />

C07D 498/04 (2006.01)<br />

A61K 31/407 (2006.01)<br />

A61P 31/12 (2006.01)<br />

(86) PCT/US2007084788 15.11.2007.<br />

(96) EP 07864438.2 15.11.2007.<br />

(87) WO2008064061, 29.05.2008. 200822<br />

(97) EP 2086980, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) 866125 P (32) 16.11.2006. (33) US<br />

939768 14.11.2007. US<br />

(54) MACROCYCLIC PEPTIDES AS HEPATITIS C VIRUS<br />

INHIBITORS<br />

(71) Bristol-Myers Squibb Company, Route 206 and Province Line<br />

Road, Princeton, NJ 08543-4000, US<br />

(72) WANG, Alan Xiangdong, Bristol-Myers Squibb Co. 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

ZHENG, Barbara Zhizhen, Bristol-Myers Squibb Co. 5 Research<br />

Parkway, Wallingford, Connecticut 06492, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2086981 *<br />

A61K 31/55 (2006.01)<br />

A61P 35/00 (2006.01)<br />

(86) PCT/US2007023948 14.11.2007.<br />

(96) EP 07867449.6 14.11.2007.<br />

(87) WO2008063525, 29.05.2008. 200822<br />

(97) EP 2086981, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />

(31) 859340 P (32) 16.11.2006. (33) US<br />

(54) COMPOUNDS FOR INHIBITING MITOTIC PROGRESSION<br />

(71) Millennium Pharmaceuticals, Inc., 40 Landsdowne Street,<br />

Cambridge, MA 02139, US<br />

(72) CLAIBORNE, Christopher F., 23 Sparks Street, Cambridge, MA<br />

02138, US<br />

SELLS, Todd B., 32 Ray Avenue, Bellingham, MA 02019, US<br />

STROUD, Stephen G., 53 Tesla Avenue, Medford, MA 02155, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>4705 *<br />

A61K 31/5025 (2006.01)<br />

A61P 3/04 (2006.01)<br />

A61P 25/04 (2006.01)<br />

(86) PCT/US2007087404 13.12.2007.<br />

(96) EP 07869220.9 13.12.2007.<br />

(87) WO2008076810, 26.06.2008. 200826<br />

(97) EP 2<strong>09</strong>4705, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />

(31) 869933 P (32) 14.12.2006. (33) US<br />

(54) AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR<br />

MODULATORS<br />

(71) Bristol-Myers Squibb Company, Route 206 and Province Line<br />

Road, Princeton, NJ 08543-4000, US<br />

(72) EWING, William R., Bristol-Myers Squibb Co. 311 Pennington-<br />

Rocky Hill Road, Pennington, New Jersey 08534, US<br />

ZHU, Yeheng, Bristol-Myers Squibb Co. 311 Pennington-Rocky Hill<br />

Road, Pennington, New Jersey 08534, US<br />

SULSKY, Richard B., 2 Coventry Square, West Trenton, New<br />

Jersey 08628, US<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>4706 *<br />

A61K 31/5025 (2006.01)<br />

A61P 25/00 (2006.01)<br />

A61P 3/00 (2006.01)<br />

C07D 495/04 (2006.01)<br />

(86) PCT/FR2007001889 19.11.2007.<br />

(96) EP 07870295.8 19.11.2007.<br />

(87) WO2008068424, 12.06.2008. 200824<br />

(97) EP 2<strong>09</strong>4706, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, Fr<br />

(31) 0610371 (32) 23.11.2006. (33) FR<br />

(54) SUBSTITUTED 2,5-DFFLYDRO-3H-PYRAZOLO[4,3-<br />

C]PYRIDAZIN-3-ONE DERIVATIVES, PREPARATION THEREOF<br />

AND USE OF SAME AS CANNABINOID CB1 RECEPTOR<br />

LIGANDS<br />

(71) Sanofi-Aventis, 174 Avenue de France, 75013 Paris, FR<br />

(72) CONGY, Christian, Sanofi-Aventis Département Brevets 174,<br />

avenue de France, 75013 Paris, FR<br />

DOS SANTOS, Victor, Sanofi-Aventis Département Brevets 174,<br />

avenue de France, 75013 Paris, FR<br />

RINALDI-CARMONA, Murielle, Sanofi-Aventis Département<br />

Brevets 174, avenue de France, 75013 Paris, FR<br />

ROUQUETTE, Arnaud, Sanofi-Aventis Département Brevets 174,<br />

avenue de France, 75013 Paris, FR<br />

VAN BROECK, Didier, Sanofi-Aventis Département Brevets 174,<br />

avenue de France, 75013 Paris, FR<br />

(51) MKP<br />

C07D 487/04 (2006.01) (97) EP 2089392 *<br />

A61K 31/519 (2006.01)<br />

A61P 15/10 (2006.01)<br />

ISSN 1331-2030

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