09/2009 - Državni zavod za intelektualno vlasništvo
09/2009 - Državni zavod za intelektualno vlasništvo
09/2009 - Državni zavod za intelektualno vlasništvo
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3464 HR - Patenti - Hrvatski glasnik <strong>intelektualno</strong>g vlasništva 16, 20<strong>09</strong>, 9, 3373 – 3601<br />
BLUHM, Harald, Dreihausener Weg 2, 59757 Arnsberg-Neheim, DE<br />
ESSERS, Michael, Kalmuentener Strasse 81b, 51467 Bergisch<br />
Gladbach, DE<br />
KROTH, Heiko, Marie-Curie-Weg 3, 69181 Leimen, DE<br />
GEGE, Christian, Elsenzstrasse 7, 69256 Mauer, DE<br />
TAVERAS, Arthur, 6 Joslin Lane, Southborough, Massachusetts<br />
01772, US<br />
D'ANDREA, Stanley, Bristol-Myers Squibb Co. 5 Research<br />
Parkway, Wallingford, Connecticut 06492, US<br />
MEANWELL, Nicholas A., Bristol-Myers Squibb Co. 5 Research<br />
Parkway, Wallingford, Connecticut 06492, US<br />
SCOLA, Paul Michael, Bristol-Myers Squibb Co. 5 Research<br />
Parkway, Wallingford, Connecticut 06492, US<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>7416 *<br />
(86) PCT/US2007025799 17.12.2007.<br />
(96) EP 07863038.1 17.12.2007.<br />
(87) WO2008076425, 26.06.2008. 200826<br />
(97) EP 2<strong>09</strong>7416, <strong>09</strong>.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>37, En<br />
(31) 875706 P (32) 18.12.2006. (33) US<br />
(54) AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL<br />
HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND<br />
USES THEREOF<br />
(71) Amgen, Inc, Patent Operations, M/S 28-2-C One Amgen Center<br />
Drive, Thousand Oaks, California 91320-1799, US<br />
(72) ALLEN, Jennifer R., 5255 Via Capote, Newbury Park, CA 91320,<br />
US<br />
BISWAS, Kaustav, 26003 Alizia Canyon Drive, Unit B, Calabasas,<br />
CA 91302, US<br />
CAO, Guo-Qiang, 4235 Via Rio, Thousand Oaks, CA 91320, US<br />
GOLDEN, Jennifer E., 3168 Tecopa Springs Lane, Simi Valley, CA<br />
93063, US<br />
MERCEDE, Stephanie, 1336 Moorpark Road, No. 183, Thousand<br />
Oaks, CA 91360, US<br />
PETERKIN, Tanya, 6130 Nevada Avenue, Apt. E311, Woodland<br />
Hills, CA 91367, US<br />
REED, Anthony, 3101 Peninsula Road, Apt. 304, Oxnard, CA<br />
93035, US<br />
TEGLEY, Christopher M., 478 Thunderhead Street, Thousand<br />
Oaks, CA 91360, US<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2086979 *<br />
A61K 31/5025 (2006.01)<br />
A61K 31/519 (2006.01)<br />
A61P 35/00 (2006.01)<br />
(86) PCT/US2007083773 06.11.2007.<br />
(96) EP 07863964.8 06.11.2007.<br />
(87) WO2008058126, 15.05.2008. 200820<br />
(97) EP 2086979, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />
(31) 864566 P (32) 06.11.2006. (33) US<br />
892523 P 01.03.2007. US<br />
957988 P 24.08.2007. US<br />
(54) IMIDAZOÝ1,2-B¨PYRIDAZINE AND PYRAZOLOÝ1,5-<br />
A¨PYRIMIDINE DERIVATIVES AND THEIR USE AS PROTEIN<br />
KINASE INHIBITORS<br />
(71) SuperGen, Inc., 4140 Dublin Boulevard, Suite 200, Dublin,<br />
California 94568, US<br />
(72) BEARSS, David J., 4001 Ironwood Drive, Cedar Hills, Utah 84062,<br />
US<br />
LIU, Xiao-Hui, 2028 Ashley Mesa Lane, Sandy, Utah 84<strong>09</strong>2, US<br />
VANKAYALAPATI, Hariprasad, 11558 South Sugar Berry Road,<br />
Draper, Utah 84020, US<br />
XU, Yong, 7557 Sandy Woods Lane, Midvale, Utah 84047, US<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2086980 *<br />
C07D 498/04 (2006.01)<br />
A61K 31/407 (2006.01)<br />
A61P 31/12 (2006.01)<br />
(86) PCT/US2007084788 15.11.2007.<br />
(96) EP 07864438.2 15.11.2007.<br />
(87) WO2008064061, 29.05.2008. 200822<br />
(97) EP 2086980, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />
(31) 866125 P (32) 16.11.2006. (33) US<br />
939768 14.11.2007. US<br />
(54) MACROCYCLIC PEPTIDES AS HEPATITIS C VIRUS<br />
INHIBITORS<br />
(71) Bristol-Myers Squibb Company, Route 206 and Province Line<br />
Road, Princeton, NJ 08543-4000, US<br />
(72) WANG, Alan Xiangdong, Bristol-Myers Squibb Co. 5 Research<br />
Parkway, Wallingford, Connecticut 06492, US<br />
ZHENG, Barbara Zhizhen, Bristol-Myers Squibb Co. 5 Research<br />
Parkway, Wallingford, Connecticut 06492, US<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2086981 *<br />
A61K 31/55 (2006.01)<br />
A61P 35/00 (2006.01)<br />
(86) PCT/US2007023948 14.11.2007.<br />
(96) EP 07867449.6 14.11.2007.<br />
(87) WO2008063525, 29.05.2008. 200822<br />
(97) EP 2086981, 12.08.20<strong>09</strong>. 20<strong>09</strong>33, En<br />
(31) 859340 P (32) 16.11.2006. (33) US<br />
(54) COMPOUNDS FOR INHIBITING MITOTIC PROGRESSION<br />
(71) Millennium Pharmaceuticals, Inc., 40 Landsdowne Street,<br />
Cambridge, MA 02139, US<br />
(72) CLAIBORNE, Christopher F., 23 Sparks Street, Cambridge, MA<br />
02138, US<br />
SELLS, Todd B., 32 Ray Avenue, Bellingham, MA 02019, US<br />
STROUD, Stephen G., 53 Tesla Avenue, Medford, MA 02155, US<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>4705 *<br />
A61K 31/5025 (2006.01)<br />
A61P 3/04 (2006.01)<br />
A61P 25/04 (2006.01)<br />
(86) PCT/US2007087404 13.12.2007.<br />
(96) EP 07869220.9 13.12.2007.<br />
(87) WO2008076810, 26.06.2008. 200826<br />
(97) EP 2<strong>09</strong>4705, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, En<br />
(31) 869933 P (32) 14.12.2006. (33) US<br />
(54) AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR<br />
MODULATORS<br />
(71) Bristol-Myers Squibb Company, Route 206 and Province Line<br />
Road, Princeton, NJ 08543-4000, US<br />
(72) EWING, William R., Bristol-Myers Squibb Co. 311 Pennington-<br />
Rocky Hill Road, Pennington, New Jersey 08534, US<br />
ZHU, Yeheng, Bristol-Myers Squibb Co. 311 Pennington-Rocky Hill<br />
Road, Pennington, New Jersey 08534, US<br />
SULSKY, Richard B., 2 Coventry Square, West Trenton, New<br />
Jersey 08628, US<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2<strong>09</strong>4706 *<br />
A61K 31/5025 (2006.01)<br />
A61P 25/00 (2006.01)<br />
A61P 3/00 (2006.01)<br />
C07D 495/04 (2006.01)<br />
(86) PCT/FR2007001889 19.11.2007.<br />
(96) EP 07870295.8 19.11.2007.<br />
(87) WO2008068424, 12.06.2008. 200824<br />
(97) EP 2<strong>09</strong>4706, 02.<strong>09</strong>.20<strong>09</strong>. 20<strong>09</strong>36, Fr<br />
(31) 0610371 (32) 23.11.2006. (33) FR<br />
(54) SUBSTITUTED 2,5-DFFLYDRO-3H-PYRAZOLO[4,3-<br />
C]PYRIDAZIN-3-ONE DERIVATIVES, PREPARATION THEREOF<br />
AND USE OF SAME AS CANNABINOID CB1 RECEPTOR<br />
LIGANDS<br />
(71) Sanofi-Aventis, 174 Avenue de France, 75013 Paris, FR<br />
(72) CONGY, Christian, Sanofi-Aventis Département Brevets 174,<br />
avenue de France, 75013 Paris, FR<br />
DOS SANTOS, Victor, Sanofi-Aventis Département Brevets 174,<br />
avenue de France, 75013 Paris, FR<br />
RINALDI-CARMONA, Murielle, Sanofi-Aventis Département<br />
Brevets 174, avenue de France, 75013 Paris, FR<br />
ROUQUETTE, Arnaud, Sanofi-Aventis Département Brevets 174,<br />
avenue de France, 75013 Paris, FR<br />
VAN BROECK, Didier, Sanofi-Aventis Département Brevets 174,<br />
avenue de France, 75013 Paris, FR<br />
(51) MKP<br />
C07D 487/04 (2006.01) (97) EP 2089392 *<br />
A61K 31/519 (2006.01)<br />
A61P 15/10 (2006.01)<br />
ISSN 1331-2030