PDF (2,8 MB) - Ãrad priemyselného vlastnÃctva SR
PDF (2,8 MB) - Ãrad priemyselného vlastnÃctva SR
PDF (2,8 MB) - Ãrad priemyselného vlastnÃctva SR
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VESTNÍK ÚRADU PRIEMYSELNÉHO VLASTNÍCTVA <strong>SR</strong> 6 - 2010 - SK (preklady patentov)<br />
(51) C07D 417/00, C07D 413/00, C07D 405/00,<br />
A61K 31/427<br />
(11) E 6836<br />
(96) 03768730.8, 7.11.2003<br />
(97) 1562941, 23.12.2009<br />
(24) 23.12.2009<br />
(31) 425352 P, 473743 P<br />
(32) 7.11.2002, 27.5.2003<br />
(33) US, US<br />
(73) Kosan Biosciences, Inc., Princeton, NJ, US;<br />
(72) LI Yong, Palo Alto, CA, US; SUNDERMANN<br />
Kurt, Burlingame, CA, US; TANG Li, Foster City,<br />
CA, US; MYLES David, Kensington, CA, US;<br />
(74) Bušová Eva, JUDr., Bratislava, SK;<br />
(86) PCT/US2003/035411<br />
(87) WO 2004/043954<br />
(54) Trans-9,10-dehydroepotilón C a D, jeho analógy<br />
a spôsoby ich prípravy<br />
(51) C07D 487/00, C07D 471/00, A61K 31/40,<br />
A61K 31/435<br />
(11) E 6850<br />
(96) 03739358.4, 27.6.2003<br />
(97) 1519939, 9.12.2009<br />
(24) 9.12.2009<br />
(31) 394337 P<br />
(32) 5.7.2002<br />
(33) US<br />
(73) Targacept, Inc., Winston-Salem, NC, US;<br />
(72) BHATTI Balwinder S., Winston-Salem, NC, US;<br />
MILLER Craig H., Winston-Salem, NC, US;<br />
SCHMITT Jeffrey D., Winston- Salem, NC, US;<br />
(74) Hörmannová Zuzana, Ing., Bratislava, SK;<br />
(86) PCT/US2003/020524<br />
(87) WO 2004/005293<br />
(54) N-aryl-diazaspirocyklické zlúčeniny, spôsoby<br />
ich prípravy a použitie týchto zlúčenín<br />
(51) C07D 419/00, C07D 413/00, C07D 493/00,<br />
A61K 31/425, C07D 417/00, C07D 313/00,<br />
C07D 303/00, C07D 277/00<br />
(11) E 6852<br />
(96) 06026750.7, 22.8.2003<br />
(97) 1767535, 2.12.2009<br />
(24) 2.12.2009<br />
(31) 405823 P, 408589 P, 423129 P, 456159 P,<br />
402004, 435408, 496741 P<br />
(32) 23.8.2002, 6.9.2002, 1.11.2002, 20.3.2003,<br />
28.3.2003, 9.5.2003, 21.8.2003<br />
(33) US, US, US, US, US, US, US<br />
(73) Sloan-Kettering Institute For Cancer Research,<br />
New York, New York, US;<br />
(72) Danishefsky Samuel J., Engelwood NJ, US; Rivkin<br />
Alexey, Hoboken NJ, US; Yoshimura Fumihiko,<br />
Kita-ku Sapporo, JP; Gabarda Ortega Ana<br />
Esther, New York, NY, US; Cho Young Shin, Cambridge,<br />
MA, US; Chou Ting-Chao, Paramus NJ,<br />
US; Dong Huajin, Beijing, CN;<br />
(74) Hörmannová Zuzana, Ing., Bratislava, SK;<br />
(54) Syntéza epotilónov, ich medziproduktov, analógov<br />
a ich použitie<br />
(51) C07D 487/00, A61K 31/38, A61K 31/395,<br />
A61P 31/00, C07D 401/00, C07D 409/00,<br />
C07K 5/00<br />
(11) E 6876<br />
(96) 04750236.4, 16.4.2004<br />
(97) 1615613, 4.11.2009<br />
(24) 4.11.2009<br />
(31) 418759<br />
(32) 18.4.2003<br />
(33) US<br />
(73) Enanta Pharmaceuticals, Inc., Watertown, MA, US;<br />
(72) Nakajima Suanne, Cambridge, MA, US; Sun Ying,<br />
Waltham, MA, US; Tang Datong, Malden, MA,<br />
US; Xu Gouyou, Auburndale, MA, US; Porter<br />
Brian, Cambridge, MA, US; OR Yat Sun, Watertown,<br />
MA, US; Wang Zhe, Hockessin, DE, US;<br />
Miao Zhenwei, Medway, MA, US;<br />
(74) Čechvalová Dagmar, Bratislava, SK;<br />
(86) PCT/US2004/011841<br />
(87) WO 2004/093798<br />
(54) Chinoxalinylové makrocyklické zlúčeniny ako<br />
inhibítory serín proteázy hepatitídy C<br />
(51) C07D 491/00, C07D 495/00, C07D 493/00,<br />
C07D 471/00, A61K 31/407, A61P 25/00<br />
(11) E 6848<br />
(96) 03810963.3, 5.11.2003<br />
(97) 1560835, 2.9.2009<br />
(24) 2.9.2009<br />
(31) 10252667<br />
(32) 11.11.2002<br />
(33) DE<br />
(73) Grünenthal GmbH, Aachen, DE;<br />
(72) HINZE Claudia, Aachen, DE; AULENBACHER<br />
Otto, Herzogenrath, DE; SUNDERMANN Bernd,<br />
Aachen, DE; OBERBÖRSCH Stefan, Aachen,<br />
DE; FRIDERICHS Elmar, Stolberg, DE; ENGL-<br />
BERGER Werner, Stolberg, DE; KÖGEL Babette-Yvonne,<br />
Langerwehe-Hamich, DE; LINZ Klaus,<br />
Wachtberg, DE; SCHICK Hans, Berlin-Weissensee,<br />
DE; SONNENSCHEIN Helmut, Berlin,<br />
DE; HENKEL Birgitta, Berlin, DE; ROSE Valerie<br />
Sarah, Saffron Walden, Essex, GB; LIPKIN<br />
Michael Jonathan, Saffron Walden, Essex, GB;<br />
(74) Tomeš Pavol, Ing., Bratislava, SK;<br />
(86) PCT/EP2003/012305<br />
(87) WO 2004/043967<br />
(54) Spirocyklické deriváty cyklohexánu<br />
(51) C07F 9/00<br />
(11) E 6904<br />
(96) 04816640.9, 10.8.2004<br />
(97) 1656386, 9.12.2009<br />
(24) 9.12.2009<br />
(31) MU08372003<br />
(32) 21.8.2003<br />
(33) IN<br />
(73) Sun Pharmaceuticals Industries Ltd., Andheri (East),<br />
Mumbai, IN;<br />
(72) Patel Vijaykumar Muljibhai, Baroda, India, IN;<br />
Chitturi Trinadha Rao, Baroda, India, IN; Thennati<br />
Rajamannar, BarodaA, India, IN;<br />
(74) Majlingová Marta, Ing., Bratislava, SK;<br />
(86) PCT/IN2004/000238<br />
(87) WO 2005/044831<br />
(54) Spôsob prípravy zlúčenín kyseliny bisfosfónovej