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PDF (2,8 MB) - Úrad priemyselného vlastníctva SR

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VESTNÍK ÚRADU PRIEMYSELNÉHO VLASTNÍCTVA <strong>SR</strong> 6 - 2010 - SK (preklady patentov)<br />

(51) C07D 417/00, C07D 413/00, C07D 405/00,<br />

A61K 31/427<br />

(11) E 6836<br />

(96) 03768730.8, 7.11.2003<br />

(97) 1562941, 23.12.2009<br />

(24) 23.12.2009<br />

(31) 425352 P, 473743 P<br />

(32) 7.11.2002, 27.5.2003<br />

(33) US, US<br />

(73) Kosan Biosciences, Inc., Princeton, NJ, US;<br />

(72) LI Yong, Palo Alto, CA, US; SUNDERMANN<br />

Kurt, Burlingame, CA, US; TANG Li, Foster City,<br />

CA, US; MYLES David, Kensington, CA, US;<br />

(74) Bušová Eva, JUDr., Bratislava, SK;<br />

(86) PCT/US2003/035411<br />

(87) WO 2004/043954<br />

(54) Trans-9,10-dehydroepotilón C a D, jeho analógy<br />

a spôsoby ich prípravy<br />

(51) C07D 487/00, C07D 471/00, A61K 31/40,<br />

A61K 31/435<br />

(11) E 6850<br />

(96) 03739358.4, 27.6.2003<br />

(97) 1519939, 9.12.2009<br />

(24) 9.12.2009<br />

(31) 394337 P<br />

(32) 5.7.2002<br />

(33) US<br />

(73) Targacept, Inc., Winston-Salem, NC, US;<br />

(72) BHATTI Balwinder S., Winston-Salem, NC, US;<br />

MILLER Craig H., Winston-Salem, NC, US;<br />

SCHMITT Jeffrey D., Winston- Salem, NC, US;<br />

(74) Hörmannová Zuzana, Ing., Bratislava, SK;<br />

(86) PCT/US2003/020524<br />

(87) WO 2004/005293<br />

(54) N-aryl-diazaspirocyklické zlúčeniny, spôsoby<br />

ich prípravy a použitie týchto zlúčenín<br />

(51) C07D 419/00, C07D 413/00, C07D 493/00,<br />

A61K 31/425, C07D 417/00, C07D 313/00,<br />

C07D 303/00, C07D 277/00<br />

(11) E 6852<br />

(96) 06026750.7, 22.8.2003<br />

(97) 1767535, 2.12.2009<br />

(24) 2.12.2009<br />

(31) 405823 P, 408589 P, 423129 P, 456159 P,<br />

402004, 435408, 496741 P<br />

(32) 23.8.2002, 6.9.2002, 1.11.2002, 20.3.2003,<br />

28.3.2003, 9.5.2003, 21.8.2003<br />

(33) US, US, US, US, US, US, US<br />

(73) Sloan-Kettering Institute For Cancer Research,<br />

New York, New York, US;<br />

(72) Danishefsky Samuel J., Engelwood NJ, US; Rivkin<br />

Alexey, Hoboken NJ, US; Yoshimura Fumihiko,<br />

Kita-ku Sapporo, JP; Gabarda Ortega Ana<br />

Esther, New York, NY, US; Cho Young Shin, Cambridge,<br />

MA, US; Chou Ting-Chao, Paramus NJ,<br />

US; Dong Huajin, Beijing, CN;<br />

(74) Hörmannová Zuzana, Ing., Bratislava, SK;<br />

(54) Syntéza epotilónov, ich medziproduktov, analógov<br />

a ich použitie<br />

(51) C07D 487/00, A61K 31/38, A61K 31/395,<br />

A61P 31/00, C07D 401/00, C07D 409/00,<br />

C07K 5/00<br />

(11) E 6876<br />

(96) 04750236.4, 16.4.2004<br />

(97) 1615613, 4.11.2009<br />

(24) 4.11.2009<br />

(31) 418759<br />

(32) 18.4.2003<br />

(33) US<br />

(73) Enanta Pharmaceuticals, Inc., Watertown, MA, US;<br />

(72) Nakajima Suanne, Cambridge, MA, US; Sun Ying,<br />

Waltham, MA, US; Tang Datong, Malden, MA,<br />

US; Xu Gouyou, Auburndale, MA, US; Porter<br />

Brian, Cambridge, MA, US; OR Yat Sun, Watertown,<br />

MA, US; Wang Zhe, Hockessin, DE, US;<br />

Miao Zhenwei, Medway, MA, US;<br />

(74) Čechvalová Dagmar, Bratislava, SK;<br />

(86) PCT/US2004/011841<br />

(87) WO 2004/093798<br />

(54) Chinoxalinylové makrocyklické zlúčeniny ako<br />

inhibítory serín proteázy hepatitídy C<br />

(51) C07D 491/00, C07D 495/00, C07D 493/00,<br />

C07D 471/00, A61K 31/407, A61P 25/00<br />

(11) E 6848<br />

(96) 03810963.3, 5.11.2003<br />

(97) 1560835, 2.9.2009<br />

(24) 2.9.2009<br />

(31) 10252667<br />

(32) 11.11.2002<br />

(33) DE<br />

(73) Grünenthal GmbH, Aachen, DE;<br />

(72) HINZE Claudia, Aachen, DE; AULENBACHER<br />

Otto, Herzogenrath, DE; SUNDERMANN Bernd,<br />

Aachen, DE; OBERBÖRSCH Stefan, Aachen,<br />

DE; FRIDERICHS Elmar, Stolberg, DE; ENGL-<br />

BERGER Werner, Stolberg, DE; KÖGEL Babette-Yvonne,<br />

Langerwehe-Hamich, DE; LINZ Klaus,<br />

Wachtberg, DE; SCHICK Hans, Berlin-Weissensee,<br />

DE; SONNENSCHEIN Helmut, Berlin,<br />

DE; HENKEL Birgitta, Berlin, DE; ROSE Valerie<br />

Sarah, Saffron Walden, Essex, GB; LIPKIN<br />

Michael Jonathan, Saffron Walden, Essex, GB;<br />

(74) Tomeš Pavol, Ing., Bratislava, SK;<br />

(86) PCT/EP2003/012305<br />

(87) WO 2004/043967<br />

(54) Spirocyklické deriváty cyklohexánu<br />

(51) C07F 9/00<br />

(11) E 6904<br />

(96) 04816640.9, 10.8.2004<br />

(97) 1656386, 9.12.2009<br />

(24) 9.12.2009<br />

(31) MU08372003<br />

(32) 21.8.2003<br />

(33) IN<br />

(73) Sun Pharmaceuticals Industries Ltd., Andheri (East),<br />

Mumbai, IN;<br />

(72) Patel Vijaykumar Muljibhai, Baroda, India, IN;<br />

Chitturi Trinadha Rao, Baroda, India, IN; Thennati<br />

Rajamannar, BarodaA, India, IN;<br />

(74) Majlingová Marta, Ing., Bratislava, SK;<br />

(86) PCT/IN2004/000238<br />

(87) WO 2005/044831<br />

(54) Spôsob prípravy zlúčenín kyseliny bisfosfónovej

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