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Fragment based drug design

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Optimalizace Hitů<br />

•Znalost způsobu, jak se fragment váže na<br />

proteinový cíl umožňuje fragment zvětšovat.<br />

• Používají se počítačové metody<br />

• Docking<br />

• „Experimentální“ metody Isostar, Superstar,<br />

Gold, GoldMine, Hermes

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