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ELS-tíðindi - nóvember 2000

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76 <strong>ELS</strong> <strong>tíðindi</strong> 11/<strong>2000</strong><br />

(21) 5548<br />

(22) 27.6.<strong>2000</strong><br />

(41) 27.6.<strong>2000</strong><br />

(51) C07D 249/06; A61K 31/475; A61K<br />

31/495; A61K 31/41; A61K 31/415;<br />

A61K 31/425; A61K 31/47; C07D<br />

521/00; C07D 231/14; C07D 401/04;<br />

C07D 403/04; C07D 417/04; C07D<br />

405/04; C07D 413/04; C07D 409/04<br />

(54) N - [(setinn fimm -atóma dí - eða<br />

tríaza díómettað hring) karbónýl]<br />

gúanidín afleiður til meðhöndlunar á<br />

blóðþurrð.<br />

(71) Pfizer Products Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Ernest S. Hamanaka; Angel<br />

Guzman-Perez; Roger B. Ruggeri;<br />

Ronald T. Wester; Christian J.<br />

Mularski; Groton, Connecticut,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 27.2.98, US, 60/076,362<br />

(85) 27.6.<strong>2000</strong><br />

(86) 5.2.99, PCT/IB99/00206<br />

(21) 5561<br />

(22) 14.7.<strong>2000</strong><br />

(41) 14.7.<strong>2000</strong><br />

(51) A61K 7/48<br />

(54) Fegrunarsamsetning sem inniheldur<br />

efnasamband með virkniörvandi<br />

interleukíni-6.<br />

(71) Sanofi-Synthelabo, 174, Avenue<br />

de France, 75013 París, Frakklandi.<br />

(72) Pierre Casellas, Montpellier; Jean-<br />

Marie Derocq, Murviel les<br />

Montpellier; Jean-Marie Pereillo,<br />

Portet sur Garonne; Frakklandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 11.2.98, FR, 98/01637<br />

(85) 14.7.<strong>2000</strong><br />

(86) 3.2.99, PCT/FR99/00220<br />

(21) 5562<br />

(22) 14.7.<strong>2000</strong><br />

(41) 14.7.<strong>2000</strong><br />

(51) C07C 231/00<br />

(54) Nýjar díhýdroxýhexanósýru afleiður.<br />

(71) Pfizer Products Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) John Charles Kath, Waterford;<br />

Matthew Frank Brown, Pawcatuck;<br />

Christopher Stanley Poss,<br />

North Stonington; Connecticut,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 5.2.98, US, 60/073,801<br />

(85) 14.7.<strong>2000</strong><br />

(86) 18.1.99, PCT/IB99/00067<br />

(21) 5563<br />

(22) 17.7.<strong>2000</strong><br />

(41) 17.7.<strong>2000</strong><br />

(51) G06F<br />

(54) Stækkanlegt samþættingarkerfi fyrir<br />

dreifða framtaksnotkun.<br />

(71) Saga Software, Inc., 11190 Sunrise<br />

Valley Drive, Reston, Virginia 20191,<br />

Bandaríkjunum.<br />

(72) Hon-Siew Yee, Herndon; John Timothy<br />

Taylor, Leesburg; Gary Alan Gordon,<br />

McLean; Virginia, Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 18.11.98, US, 60/108,993<br />

5.10.99, US, 09/4 12,595<br />

5.10.99, US, 09/4 12,633<br />

(85) 17.7.<strong>2000</strong><br />

(86) 18.11.99, PCT/US99/27238<br />

(21) 5567<br />

(22) 20.7.<strong>2000</strong><br />

(41) 20.7.<strong>2000</strong><br />

(51) C12N 15/60; C12N 15/52; C12N 9/88;<br />

C12N 15/76; C12P 19/62; C12P 17/18;<br />

C12Q 1/527; C12N 1/21<br />

(54) Streptomyces avermitilis gen sem<br />

stýrir hlutfallinu milli B2:B1<br />

avermektína.<br />

(71) Pfizer Products Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Kim Jonelle Stutzman-Engwall, East<br />

Lyme, Connecticut, Bandaríkjunum;<br />

Yoshihiro Katoh, Aichi-ken, Japan;<br />

Hamish Alastair Irvine McArthur,<br />

Gales Ferry, Connecticut,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 13.2.98, US, 60/074,636<br />

(85) 20.7.<strong>2000</strong><br />

(86) 25.1.99, PCT/IB99/00130<br />

(21) 5568<br />

(22) 20.7.<strong>2000</strong><br />

(41) 20.7.<strong>2000</strong><br />

(51) A61K 31/535<br />

(54) Lyfjafræðilega virkt morfólínól.<br />

(71) Glaxo Group Limited, Glaxo<br />

Wellcome House, Berkeley Avenue,<br />

Greenford, Middlesex UB6 ONN,<br />

Bretlandi.<br />

(72) Phillip Frederick Morgan; David Lee<br />

Musso; John Joseph Partridge;<br />

Research Triangle Park, North Carolina,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 21.1.98, GB, 9801230.5<br />

22.1.98, US, 60/072,180<br />

(85) 20.7.<strong>2000</strong><br />

(86) 20.1.99, PCT/US99/01134<br />

(21) 5569<br />

(22) 20.7.<strong>2000</strong><br />

(41) 20.7.<strong>2000</strong><br />

(51) A61K 9/00; A61K 47/12; A61K 31/52<br />

(54) Lyfjasamsetningar.<br />

(71) Glaxo Group Limited, Glaxo<br />

Wellcome House, Berkeley Avenue,<br />

Greenford, Middlesex UB6 ONN,<br />

Bretlandi.<br />

(72) Nikki Thoennes Brooks, Glen Allen,<br />

Virginia, Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 6.2.98, GB, 9802472.2<br />

(85) 20.7.<strong>2000</strong><br />

(86) 4.2.99, PCT/EP99/00663<br />

(21) 5571<br />

(22) 24.7.<strong>2000</strong><br />

(41) 24.7.<strong>2000</strong><br />

(51) A61K 31/565; A61K 31/57<br />

(54) Lyfjasamsetningar sem valvíst bæta<br />

upp estrógenskort í miðtaugakerfinu.<br />

(71) Jenapharm GmbH & Co. KG, Otto-<br />

Schott-Strasse 15, D-07745 Jena,<br />

Þýskalandi.<br />

(72) Vladimir Patchev, Jena; Michael<br />

Oettel, Jena; Ina Thieme,<br />

Graitschen; Sigfrid Schwarz, Jena;<br />

Wolfgang Römer, Jena; Þýskalandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 20.2.98, DE, 19807264.3<br />

15.5.98, DE, 19821831.1<br />

(85) 24.7.<strong>2000</strong><br />

(86) 10.2.99, PCT/DE99/00353<br />

(21) 5575<br />

(22) 25.7.<strong>2000</strong><br />

(41) 25.7.<strong>2000</strong><br />

(51) C07D 487/04; A61K 31/50<br />

(54) Setið 1,2,4-tríasóló[3,4-a]pýridasín.<br />

(71) Merck Sharp & Dohme Limited,<br />

Hertford Road, Hoddesdon,<br />

Hertfordshire EN11 9BU, Bretlandi.<br />

(72) William Robert Carling; Tamara<br />

Ladduwahetty; Angus Murray<br />

Macleod; Kevin John Merchant;<br />

Kevin William Moore; Francine<br />

Sternfeld; Leslie Joseph Street;<br />

Harlow, Essex, Bretlandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 25.2.98, GB, 9803992.8<br />

6.5.98, GB, PCT/GB98/0130<br />

12.11.98, GB, 9824896.6<br />

(85) 25.7.<strong>2000</strong><br />

(86) 17.2.99, PCT/GB99/00485

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