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ELS-tíðindi - janúar 2002 - Einkaleyfastofan

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68 <strong>ELS</strong> <strong>tíðindi</strong> 1/02<br />

(21) 6158<br />

(22) 13.11.2001<br />

(41) 13.11.2001<br />

(51) C07D 401/12; C07D 401/14; A61K<br />

31/495<br />

(54) Pýrazínón þrombín latar.<br />

(71) Merck & Co., Inc., 126 East Lincoln<br />

Avenue, Rahway, New Jersey<br />

07065-0907, Bandaríkjunum.<br />

(72) Christopher S. Burgey; Kyle A.<br />

Robinson; Peter D. Williams; Craig<br />

A. Coburn; Terry A. Lyle; Philip E.<br />

Sanderson; Rahway, New Jersey,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 4.6.99, US, 60/137,538<br />

16.7.99, US, 60/144,291<br />

(85) 13.11.2001<br />

(86) 1.6.2000, PCT/US00/15140<br />

(21) 6159<br />

(22) 13.11.2001<br />

(41) 13.11.2001<br />

(51) C07D 453/02; A61K 31/439; A61P<br />

1/08<br />

(54) Fjölgervingar af kristölluðu<br />

asabísýkló (2,2,2) oktan-3-amín<br />

sítrati og lyfjasamsetningar.<br />

(71) Pfizer Product Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Michael James Castaldi; George<br />

Joseph Quallich; Lewin Theophilus<br />

Wint; Groton, Connecticut,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 1.6.99, US, 60/136,992<br />

(85) 13.11.2001<br />

(86) 18.5.2000, PCT/IB00/00665<br />

(21) 6160<br />

(22) 13.11.2001<br />

(41) 13.11.2001<br />

(51) C07H 17/08; A61K 31/70; A61P 31/04<br />

(54) Dífosfat salt af 4"-setinni-9-deoxó-<br />

9A-asa-9A-hómóerýtrómysín afleiðu<br />

og lyfjasamsetning þar af.<br />

(71) Pfizer Product Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Robert John Rafka; Colman Brendan<br />

Ragan; Douglas John Meldrum<br />

Allen; Groton, Connecticut,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 30.6.99, US, 60/141,681<br />

(85) 13.11.2001<br />

(86) 13.6.2000, PCT/IB00/00785<br />

(21) 6161<br />

(22) 13.11.2001<br />

(41) 13.11.2001<br />

(51) C07D 453/02; A61K 31/435; A61P<br />

25/28<br />

(54) Fjölgervingar af kristölluðu (2benshýdrýl-1-azabísýkló<br />

[2,2,2]okt-<br />

3-ýl)-(5-ísóprópýl-2-metoxýbensýl)ammóníumklóríði<br />

sem NK-1 viðtaka<br />

mótlyf.<br />

(71) Pfizer Product Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Douglas John Meldrum Allen; Troy<br />

Anthony Appleton; Michael Jon<br />

Gumkowski; David Joseph<br />

Muehlbauer; Timothy Norris; Groton,<br />

Connecticut, Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 22.6.99, US, 60/140,233<br />

(85) 13.11.2001<br />

(86) 6.6.2000, PCT/IB00/00756<br />

(21) 6163<br />

(22) 16.11.2001<br />

(41) 16.11.2001<br />

(51) A61K 47/48<br />

(54) Lyfjakomplex.<br />

(71) Pfizer Inc., 235 East 42nd Street,<br />

New York, New York 10017,<br />

Bandaríkjunum.<br />

(72) Anne Billotte, Sandwich, Kent,<br />

Bretlandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 29.6.99, GB, 9915231.6<br />

(85) 16.11.2001<br />

(86) 2.6.2000, PCT/IB00/00746<br />

(21) 6164<br />

(22) 16.11.2001<br />

(41) 16.11.2001<br />

(51) A61K 31/451; A61K 31/4523; C07D<br />

401/10; A61K 31/453; C07D 405/14;<br />

C07D 401/14; C07D 211/22; C07D<br />

405/12; C07D 211/26; C07D 417/10;<br />

A61P 9/00<br />

(54) Málmpróteasa latar.<br />

(71) Pfizer Inc., 235 East 42nd Street,<br />

New York, New York 10017,<br />

Bandaríkjunum.<br />

(72) Kevin Neil Dack; Michael Jonathan<br />

Fray; Gavin Alistair Whitlock; Mark<br />

Llewellyn Lewis; Nicholas Murray<br />

Thomson; Sandwich, Kent,<br />

Bretlandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 3.6.99, GB, 9912961.1<br />

(85) 16.11.2001<br />

(86) 18.5.2000, PCT/IB00/00667<br />

(21) 6165<br />

(22) 16.11.2001<br />

(41) 16.11.2001<br />

(51) C07H 19/167; A61K 31/70; A61P 11/00;<br />

A61P 9/00<br />

(54) Púrín afleiður.<br />

(71) Pfizer Inc., 235 East 42nd Street,<br />

New York, New York 10017,<br />

Bandaríkjunum.<br />

(72) Sandra Marina Monaghan,<br />

Sandwich, Kent, Bretlandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 14.10.99, GB, 9924363.6<br />

(85) 16.11.2001<br />

(86) 6.10.2000, PCT/IB00/01444<br />

(21) 6166<br />

(22) 19.11.2001<br />

(41) 19.11.2001<br />

(51) C07D 239/42; C07D 409/04; C07D<br />

401/04; C07D 403/12; A61K 31/505;<br />

A61K 31/506; A61P 9/14<br />

(54) 5-sýanó-2-amínópýrimidín afleiður.<br />

(71) Celltech R&D Limited, 208 Bath<br />

Road, Slough, Berkshire SL1 3WE,<br />

Bretlandi.<br />

(72) Mark James Batchelor, Watlington,<br />

Oxfordshire; David Festus Charles<br />

Moffat, Maidenhead, Berkshire;<br />

Jeremy Martin Davis, Wokingham,<br />

Berkshire; Martin Clive Hutchings,<br />

Wokingham, Berkshire; Bretlandi.<br />

(74) Sigurjónsson & Thor, ehf.,<br />

Skólavörðustíg 16, 101 Reykjavík.<br />

(30) 18.6.99, GB, 9914258.0<br />

(85) 19.11.2001<br />

(86) 19.6.2000, PCT/GB00/02382<br />

(21) 6168<br />

(22) 20.11.2001<br />

(41) 20.11.2001<br />

(51) F16K 31/12<br />

(54) Vökvaflæði- og þrýstistýrikerfi og<br />

aðferð.<br />

(71) M-I L.L.C., P.O. Box 42842, Houston,<br />

Texas 77242-2842, Bandaríkjunum.<br />

(72) Roger Suter, Edmond, Oklahoma;<br />

Lester L. Cain; Bandaríkjunum.<br />

(74) A&P Árnason ehf., Efstaleiti 5, 103<br />

Reykjavík.<br />

(30) 21.5.99, US, 09/316,579<br />

(85) 20.11.2001<br />

(86) 28.4.2000, PCT/US00/11404<br />

(21) 6169<br />

(22) 21.11.2001<br />

(41) 21.11.2001<br />

(51) E04C 2/34<br />

(54) Léttur byggingarþáttur á formi hols<br />

meginhluta með uppbyggingu<br />

sexhyrnds yfirborðs.<br />

(71) Peter Küppers, Kaiserstiege 143,<br />

D-48599 Gronau, Þýskalandi.<br />

(72) Peter Küppers, Gronau, Þýskalandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 27.5.99, DE, 199 24 332.8<br />

10.5.2000, DE, 100 22 742.2<br />

(85) 21.11.2001<br />

(86) 25.5.2000, PCT/DE00/01683

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