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輔舒酮TM 優氟TM吸入劑50微公克/劑量

輔舒酮TM 優氟TM吸入劑50微公克/劑量

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TM TM 50 /<br />

FLIXOTIDE TM Evohaler TM 50 g<br />

023755 <br />

TM TM 250 /<br />

FLIXOTIDE TM Evohaler TM 250 g<br />

023753 <br />

<br />

50 /( 250 /)<br />

50 mcg( 250 mcg) fluticasone propionate<br />

<br />

<br />

<br />

FLIXOTIDE 50 Evohaler 120 <br />

FLIXOTIDE 250 Evohaler 60 120 <br />

<br />

<br />

FLIXOTIDE <br />

<br />

(adrenal reserve)<br />

<br />

PEF 60% 30%<br />

()<br />

<br />

<br />

<br />

<br />

<br />

<br />

(PEF 80% 20%)<br />

<br />

(PEF 60-80% 20-30%)<br />

<br />

<br />

(PEF 60% 30%)


FLIXOTIDE <br />

<br />

<br />

<br />

<br />

<br />

<br />

4 7 <br />

24 <br />

<br />

<br />

<br />

<br />

16 <br />

100 1000 mcg<br />

FLIXOTIDE <br />

100 mcg 250 mcg<br />

250 mcg 500 mcg<br />

500 mcg 1000 mcg<br />

<br />

fluticasone propionate beclomethasone<br />

dipropionate <br />

4 <br />

50 mcg 200 mcg<br />

fluticasone propionate 50 mcg 100 mcg<br />

<br />

<br />

<br />

<br />

<br />

<br />

<br />

-<br />

<br />

<br />

(peak flow)<br />

FLIXOTIDE


FLIXOTIDE <br />

<br />

<br />

()<br />

(Cushing’s syndrome)<br />

<br />

()<br />

<br />

<br />

<br />

<br />

FLIXOTIDE <br />

FLIXOTIDE <br />

<br />

<br />

<br />

antihistamine /<br />

FLIXOTIDE <br />

FLIXOTIDE ()<br />

<br />

<br />

fluticasone propionate ritonavir <br />

<br />

fluticasone propionate ritonavir <br />

<br />

()<br />

<br />

()<br />

FLIXOTIDE <br />

FLIXOTIDE


fluticasone propionate <br />

<br />

P450 3A4 fluticasone propionate <br />

<br />

ritonavir (<br />

P450 3A4 ) fluticasone propionate <br />

<br />

fluticasone propionate ritonavir <br />

<br />

fluticasone propionate ritonavir <br />

<br />

P450 3A4 (erythromycin)<br />

(ketoconazole)fluticasone propionate <br />

P450 3A4 (<br />

ketoconazole) fluticasone propionate <br />

<br />

<br />

fluticasone propionate <br />

<br />

<br />

fluticasone propionate <br />

<br />

fluticasone propionate<br />

fluticasone propionate <br />

fluticasone propionate <br />

fluticasone propionate <br />

<br />

<br />

FLIXOTIDE <br />

<br />

(1/10)(<br />

1/100


FLIXOTIDE<br />

(COPD )<br />

<br />

<br />

<br />

()(/<br />

)<br />

<br />

()<br />

(Cushing’s syndrome)<br />

<br />

<br />

<br />

<br />

()<br />

<br />

<br />

(hoarseness)<br />

(paradosical bronchospasm)<br />

<br />

(paradosical bronchospasm)<br />

FLIXOTIDE Evohaler <br />

<br />

<br />

<br />

<br />

--<br />

<br />

<br />

()(<br />

1000 1000 )<br />

/<br />

<br />

<br />

<br />

<br />

FLIXOTIDE


fluticasone propionate <br />

fluticasone propionate <br />

fluticasone propionate Accuhaler/Diskus<br />

fluticasone propionate Diskhaler fluticasone propionate Evohaler <br />

7.8%9.0% 10.9% COPD <br />

fluticasone propionate <br />

<br />

<br />

1%<br />

<br />

<br />

Fluticasone propionate ( 300 )<br />

(91%)<br />

<br />

Fluticasone propionate<br />

P450 CYP3A4 CYP3A4 <br />

CYP3A4 fluticasone propionate <br />

<br />

<br />

Fluticasone propionate (1150 /) 8 <br />

Fluticasone propionate 0.2%<br />

5% Fluticasone propionate <br />

<br />

<br />

<br />

Fluticasone propionate <br />

<br />

HFA134a CFC <br />

<br />

<br />

<br />

Hydroxyfluoroalkane 134a, 1, 1, 1, 2-tetrafluoroethane (HFA 134a)


FLIXOTIDE Evohaler 2~30<br />

<br />

<br />

<br />

50 mcg/dose( 250 mcg/dose)60120 <br />

FLIXOTIDE Evohaler fluticasone propionate CFC <br />

HFA134a<br />

<br />

<br />

<br />

<br />

<br />

<br />

1. <br />

2. <br />

3. <br />

4.


5. <br />

6. salmeterol <br />

fluticasone propionate<br />

7.


8. 30 <br />

3 7<br />

9. <br />

<br />

56 7 <br />

<br />

2 <br />

<br />

<br />

<br />

<br />

1. <br />

2. <br />

3. <br />

4. <br />

<br />

: GDS26/IPI06<br />

: 11 January 2008<br />

Glaxo Wellcome S.A.<br />

<br />

Avenida Extremadura, 3, 09400, Aranda De Duero, Burgos, Spain<br />

GlaxoSmithKline Australia Pty. Ltd.<br />

<br />

<br />

<br />

1061 Monutain Highway, Boronia, Victoria 3155, Australia

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