European Patent Bulletin 2012/09 - European Patent Office
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European Patent Bulletin 2012/09 - European Patent Office

European Patent Bulletin 2012/09 - European Patent Office European Patent Bulletin 2012/09 - European Patent Office

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(C07D) I.1(1) C07D 403/14 → (51) C07D 401/12 C07D 405/04 → (51) C07D 207/16 C07D 405/04 → (51) C07D 213/64 (51) C07D 405/06 (11) 2 421 856 A1* C07D 409/06 C07D 205/06 A61K 31/496 A61P 25/00 A61P 29/00 (25) En (26) En (21) 10716672.0 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032086 22.04.2010 (87) WO 2010/124112 2010/43 28.10.2010 (30) 22.04.2009 US 171649 P 22.04.2009 US 171658 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS DIAMIDES D'AZÉTIDINYLE INHIBITEURS DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Sui-po, Exton PA 19341, US ZHANG, Yue-mei, Spring House PA 19477, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, Carpmaels & Ransford One Southampton Row, GB- London WC1B 5HA, GB C07D 405/06 → (51) C07D 207/16 C07D 405/06 → (51) C07D 401/10 C07D 405/06 → (51) C07D 405/12 (51) C07D 405/12 (11) 2 421 857 A2* C07D 405/06 (25) En (26) En (21) 10722163.2 (22) 23.03.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) GB 2010/000545 23.03.2010 (87) WO 2010/109185 2010/39 30.09.2010 (88) 05.05.2011 (30) 23.03.2009 IN MU06672009 (54) VERFAHREN ZUR HERSTELLUNG VON DOXAZOSIN UND SALZEN DARAUS Process for the preparation of doxazosin and salts thereof Procédé de préparation de la doxazosine et de ses sels (71) CIPLA LIMITED, Mumbai Central, Mumbai 400 008, IN Europäisches Patentblatt European Patent Bulletin Bulletin européen des brevets (72) RAO, Dharmaraj Ramachandra, Maharashtra, IN KANKAN, Rajendra Narayanrao, Mumbai 400 076, IN BIRARI, Dilip Ramdas, Maharashtra, IN (74) Ono, Shusuke, A.A. Thornton & Co. 235 High Holborn, London WC1V 7LE, GB C07D 405/12 → (51) C07D 205/04 C07D 405/12 → (51) C07D 207/16 C07D 405/12 → (51) C07D 211/60 C07D 405/12 → (51) C07D 213/81 C07D 405/14 → (51) C07D 205/04 C07D 405/14 → (51) C07D 207/16 C07D 405/14 → (51) C07D 401/12 C07D 407/04 → (51) C07D 401/04 (51) C07D 409/06 (11) 2 421 858 A1* A61K 31/5415 A61P 31/00 (25) En (26) En (21) 10713994.1 (22) 20.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055176 20.04.2010 (87) WO 2010/122012 2010/43 28.10.2010 (30) 20.04.2009 EP 09158229 20.04.2009 US 202918 P (54) THIOXANTHENDERIVATE ZUR BEHAND- LUNG VON INFEKTIONSKRANKHEITEN THIOXANTHENE DERIVATIVES FOR THE TREATMENT OF INFECTIOUS DISEASES DÉRIVÉS DE THIOXANTHÈNE POUR LE TRAITEMENT DE MALADIES INFEC- TIEUSES (71) BKG Pharma ApS, Birgit Kjoldgaard Giwercman Vintervej 2, 2920 Charlottenlund, DK (72) GIWERCMAN, Birgit, Kjældgaard, DK-2920 Charlottenlund, DK (74) Bender, Mikkel, et al, Chas. Hude A/S Patent H.C. Andersens Boulevard 33, 1780 Copenhagen, DK C07D 409/06 → (51) C07D 205/04 C07D 409/06 → (51) C07D 401/06 C07D 409/06 → (51) C07D 401/10 C07D 409/06 → (51) C07D 405/06 C07D 409/10 → (51) C07D 401/10 C07D 409/12 → (51) C07D 205/04 C07D 409/12 → (51) C07D 401/12 C07D 409/14 → (51) C07D 205/04 C07D 409/14 → (51) C07D 207/16 C07D 409/14 → (51) C07D 401/04 C07D 409/14 → (51) C07D 401/12 C07D 413/06 → (51) C07D 401/10 C07D 413/12 → (51) C07D 205/04 C07D 413/12 → (51) C07D 207/16 86 Anmeldungen Applications Demandes (09/2012) 29.02.2012 C07D 413/12 → (51) C07D 213/81 C07D 413/12 → (51) C07D 231/14 C07D 413/12 → (51) C07D 401/12 C07D 413/14 → (51) C07D 205/04 C07D 413/14 → (51) C07D 231/14 C07D 413/14 → (51) C07D 401/12 C07D 413/14 → (51) C07D 403/14 (51) C07D 417/04 (11) 2 421 859 A1* C07F 9/38 A61K 31/496 A61P 7/02 A61P 9/10 (25) En (26) En (21) 10719097.7 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) IB 2010/051742 21.04.2010 (87) WO 2010/122504 2010/43 28.10.2010 (30) 22.04.2009 PCT/IB2009/051647 (54) THIAZOLDERIVATE UND IHRE VERWEN- DUNG ALS P2Y12-REZEPTORANTAGO- NISTEN THIAZOLE DERIVATIVES AND THEIR USE AS P2Y12 RECEPTOR ANTAGONISTS DÉRIVÉS DE THIAZOLE ET LEURS UTILI- SATION COMME ANTAGONISTES DU RECEPTEUR P2Y12 (71) Actelion Pharmaceuticals Ltd., Gewerbestrasse 16, 4123 Allschwil, CH (72) CAROFF, Eva, CH-4123 Allschwil, CH HILPERT, Kurt, CH-4123 Allschwil, CH HUBLER, Francis, CH-4123 Allschwil, CH LEHMANN, David, CH-4123 Allschwil, CH MEYER, Emmanuel, CH-4123 Allschwil, CH RENNEBERG, Dorte, CH-4123 Allschwil, CH (74) Gschwend, Thomas Peter, Actelion Pharmaceuticals Ltd Gewerbestrasse 16, CH-4123 Allschwil, CH C07D 417/06 → (51) C07D 205/04 C07D 417/06 → (51) C07D 401/06 C07D 417/06 → (51) C07D 401/10 (51) C07D 417/12 (11) 2 421 860 A1* C07D 417/14 A61K 31/496 A61P 25/00 A61P 29/00 (25) En (26) En (21) 10715456.9 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032045 22.04.2010 (87) WO 2010/124082 2010/43 28.10.2010 (30) 22.04.2009 US 171649 P 22.04.2009 US 171658 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS AZÉTIDINYL DIAMIDES EN TANT QU'IN- HIBITEURS DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US

(C07D) I.1(1) FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Sui-po, Exton PA 19341, US ZHANG, Yue-mei, Spring House PA 19477, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, Carpmaels & Ransford One Southampton Row, London WC1B 5HA, GB C07D 417/12 → (51) C07D 205/04 C07D 417/12 → (51) C07D 213/81 C07D 417/12 → (51) C07D 401/12 (51) C07D 417/14 (11) 2 421 861 A1* A01N 43/80 (25) En (26) En (21) 10719453.2 (22) 19.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/031546 19.04.2010 (87) WO 2010/123791 2010/43 28.10.2010 (30) 22.04.2009 US 171573 P 08.03.2010 US 311512 P (54) FESTE FORMEN EINES AZOCYCLISCHEN AMIDS SOLID FORMS OF AN AZOCYCLIC AMIDE FORMES SOLIDES D'UN AMIDE AZOCY- CLIQUE (71) E. I. du Pont de Nemours and Company, 1007 Market Street, Wilmington, DE 19898, US (72) HANAGAN, Mary, Ann, Newark Delaware 19711, US OBERHOLZER, Matthew, Richard, Wilmington Delaware 19810, US PASTERIS, Robert, James, Newark Delaware 19713, US SHAPIRO, Rafael, Wilmington Delaware 19803, US (74) Beacham, Annabel Rose, Dehns St Bride's House 10 Salisbury Square, London EC4Y 8JD, GB C07D 417/14 → (51) C07D 205/04 C07D 417/14 → (51) C07D 401/12 C07D 417/14 → (51) C07D 417/12 C07D 453/02 → (51) C07D 231/14 (51) C07D 471/00 (11) 2 421 862 A1* (25) En (26) En (21) 10767711.4 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) US 2010/031916 21.04.2010 (87) WO 2010/124005 2010/43 28.10.2010 (30) 21.04.2009 US 171273 P (54) OCTAHYDROBENZOISOCHINOLINMODU- LATOREN VON DOPAMINREZEPTOREN UND IHRE VERWENDUNG Europäisches Patentblatt European Patent Bulletin Bulletin européen des brevets OCTAHYDROBENZOISOQUINOLINE MODULATORS OF DOPAMINE RECEPTORS AND USES THEREFOR MODULATEURS OCTAHYDROBENZOISO- QUINOLÉINES DE RÉCEPTEURS DE LA DOPAMINE, ET UTILISATIONS DE CES MODULATEURS (71) Purdue Research Foundation, 1281 Win Hentschel Boulevard, West Lafayette, IN 47906, US (72) NICHOLS, David, Earl, West Lafayette IN 47906, US WATTS, Val, Joseph, West Lafayette IN 47906, US (74) Chapman, Paul Gilmour, et al, Marks & Clerk LLP Aurora 120 Bothwell Street, Glasgow G2 7JS, GB (51) C07D 471/04 (11) 2 421 863 A1* A61K 31/4375 A61P 25/00 (25) En (26) En (21) 10714304.2 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055284 21.04.2010 (87) WO 2010/122064 2010/43 28.10.2010 (30) 21.04.2009 DK 200900516 27.04.2009 US 172822 P (54) SUBSTITUIERTE NAPHTHYRIDINDERI- VATE UND DEREN MEDIZINISCHE VER- WENDUNG SUBSTITUTED NAPHTHYRIDINE DERI- VATIVES AND THEIR MEDICAL USE DÉRIVÉS DE NAPHTYRIDINE SUBSTI- TUÉS ET LEUR UTILISATION MÉDICALE (71) NeuroSearch AS, Pederstrupvej 93, 2750 Ballerup, DK (72) BROWN, William, Dalby, DK-2750 Ballerup, DK JESSEN, Carsten, DK-2750 Ballerup, DK MATTSSON, Cecilia, S-413 46 Göteborg, SE SOTT, Richard, S-413 46 Göteborg, SE STRØBÆK, Dorte, DK-2750 Ballerup, DK (51) C07D 471/04 (11) 2 421 864 A1* A61K 31/4745 A61P 35/00 (25) Fr (26) Fr (21) 10723723.2 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) FR 2010/050773 22.04.2010 (87) WO 2010/122272 2010/43 28.10.2010 (30) 24.04.2009 FR 0901995 (54) 1-PYRAZOLO[4,3-C]ISOCHINOLINDERI- VATE, DEREN HERSTELLUNG UND DE- REN THERAPEUTISCHE VERWENDUNG 1-PYRAZOLO[4,3-C]ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF DERIVES DE 1-PYRAZOLO[4,3-c]ISOQUI- NOLEINES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE (71) SANOFI, 174, Avenue de France, 75013 Paris, FR (72) DELETTRE, Georges, F-75013 Paris, FR DEPRETS, Stéphanie, F-75013 Paris, FR HALLEY, Frank, F-75013 Paris, FR SCHIO, Laurent, F-75013 Paris, FR THOMPSON, Fabienne, F-75013 Paris, FR (74) Jacobson, Claude, et al, Cabinet Lavoix 2, Place d'Estienne d'Orves, 75441 Paris Cedex 09, FR C07D 471/04 → (51) A61P 35/00 C07D 471/04 → (51) C07D 498/04 87 Anmeldungen Applications Demandes (09/2012) 29.02.2012 (51) C07D 471/10 (11) 2 421 865 A1* A01N 43/90 (25) En (26) En (21) 10713606.1 (22) 30.03.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) EP 2010/054216 30.03.2010 (87) WO 2010/115780 2010/41 14.10.2010 (30) 08.04.2009 GB 0906164 (54) ALS PESTIZIDE VERWENDETE SPIROHE- TEROCYCLISCHE PYRROLIDINDIONDE- RIVATE SPIROHETEROCYCLIC PYRROLIDINE DIONE DERIVATIVES USED AS PESTICIDES DÉRIVÉS SPIRO-HÉTÉROCYCLIQUES DE PYRROLIDINE-DIONE UTILISÉS COMME PESTICIDES (71) Syngenta Participations AG, Schaffhauserstrasse, 4332 Stein, CH (72) MUEHLEBACH, Michel, CH-4332 Stein, CH HUETER, Ottmar Franz, CH-4332 Stein, CH (74) Herrmann, Jörg, Syngenta Crop Protection Münchwilen AG Intellectual Property Department Schaffhauserstrasse, CH-4332 Stein, CH (51) C07D 471/10 (11) 2 421 866 A1* A61K 31/4747 A61P 35/00 (25) En (26) En (21) 10716316.4 (22) 20.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055139 20.04.2010 (87) WO 2010/121995 2010/43 28.10.2010 (30) 23.04.2009 US 171970 P (54) 3,3'-SPIROINDOLINONDERIVATE UND DEREN VERWENDUNG GEGEN KREBS 3,3'-SPIROINDOLINONE DERIVATIVES AND THEIR USE FOR CANCER DÉRIVÉS 3,3'-SPIROINDOLINONE ET LEUR UTILISATION POUR LE CANCER (71) F.Hoffmann-La Roche AG, Grenzacherstrasse 124, 4070 Basel, CH (72) CHEN, Li, Shanghai 201203, CN HAN, Xingchun, Shanghai 201102, CN YANG, Song, Shanghai 201210, CN ZHANG, Zhuming, Hillsborough New Jersey 08844, US (74) Beyermann, Jochen Carl, et al, F. Hoffmann- La Roche AG CLP - Patent Department Grenzacherstrasse 124, 4070 Basel, CH C07D 471/14 → (51) A61P 35/00 C07D 471/14 → (51) C07D 498/04 (51) C07D 487/04 (11) 2 421 867 A2* C07D 403/12 A61P 19/02 A61P 37/02 (25) En (26) En (21) 10767652.0 (22) 20.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) US 2010/031773 20.04.2010 (87) WO 2010/123919 2010/43 28.10.2010 (88) 03.03.2011 (30) 03.02.2010 US 300887 P 20.04.2009 US 170858 P (54) PIPERIDINHEMMER DER JANUS-KINASE 3 PIPERIDINE INHIBITORS OF JANUS KINASE 3 INHIBITEURS PIPÉRIDINIQUES DE LA JANUS KINASE 3

(C07D) I.1(1)<br />

C07D 403/14 → (51) C07D 401/12<br />

C07D 405/04 → (51) C07D 207/16<br />

C07D 405/04 → (51) C07D 213/64<br />

(51) C07D 405/06 (11) 2 421 856 A1*<br />

C07D 4<strong>09</strong>/06 C07D 205/06<br />

A61K 31/496 A61P 25/00<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 10716672.0 (22) 22.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) US 2010/032086 22.04.2010<br />

(87) WO 2010/124112 2010/43 28.10.2010<br />

(30) 22.04.20<strong>09</strong> US 171649 P<br />

22.04.20<strong>09</strong> US 171658 P<br />

(54) AZETIDINYLDIAMIDE ALS MONOACYL-<br />

GLYCERINLIPASEINHIBITOREN<br />

AZETIDINYL DIAMIDES AS MONOACYL-<br />

GLYCEROL LIPASE INHIBITORS<br />

DIAMIDES D'AZÉTIDINYLE INHIBITEURS<br />

DE LA MONOACYLGLYCÉROL LIPASE<br />

(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) BIAN, Haiyan, Princeton NJ 08540, US<br />

CHEVALIER, Kristen, M., Collegeville PA<br />

19426, US<br />

CONNOLLY, Peter, J., Spring House PA<br />

19477, US<br />

FLORES, Christopher, M., Spring House PA<br />

19477, US<br />

LIN, Shu-chen, Doylestown PA 18902, US<br />

LIU, Li, Doylestown PA 18901, US<br />

MABUS, John, East Greenville PA 18041, US<br />

MACIELAG, Mark, J., Spring House PA<br />

19477, US<br />

MCDONNELL, Mark, E., Lansdale PA 19446,<br />

US<br />

PITIS, Philip, M., North Wales PA 19454, US<br />

ZHANG, Sui-po, Exton PA 19341, US<br />

ZHANG, Yue-mei, Spring House PA 19477,<br />

US<br />

ZHU, Bin, Spring House PA 19477, US<br />

CLEMENTE, Jose, Exton PA 19341, US<br />

(74) Warner, James Alexander, Carpmaels &<br />

Ransford One Southampton Row, GB-<br />

London WC1B 5HA, GB<br />

C07D 405/06 → (51) C07D 207/16<br />

C07D 405/06 → (51) C07D 401/10<br />

C07D 405/06 → (51) C07D 405/12<br />

(51) C07D 405/12 (11) 2 421 857 A2*<br />

C07D 405/06<br />

(25) En (26) En<br />

(21) 10722163.2 (22) 23.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) GB 2010/000545 23.03.2010<br />

(87) WO 2010/1<strong>09</strong>185 2010/39 30.<strong>09</strong>.2010<br />

(88) 05.05.2011<br />

(30) 23.03.20<strong>09</strong> IN MU066720<strong>09</strong><br />

(54) VERFAHREN ZUR HERSTELLUNG VON<br />

DOXAZOSIN UND SALZEN DARAUS<br />

Process for the preparation of doxazosin<br />

and salts thereof<br />

Procédé de préparation de la doxazosine<br />

et de ses sels<br />

(71) CIPLA LIMITED, Mumbai Central, Mumbai<br />

400 008, IN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(72) RAO, Dharmaraj Ramachandra, Maharashtra,<br />

IN<br />

KANKAN, Rajendra Narayanrao, Mumbai 400<br />

076, IN<br />

BIRARI, Dilip Ramdas, Maharashtra, IN<br />

(74) Ono, Shusuke, A.A. Thornton & Co. 235<br />

High Holborn, London WC1V 7LE, GB<br />

C07D 405/12 → (51) C07D 205/04<br />

C07D 405/12 → (51) C07D 207/16<br />

C07D 405/12 → (51) C07D 211/60<br />

C07D 405/12 → (51) C07D 213/81<br />

C07D 405/14 → (51) C07D 205/04<br />

C07D 405/14 → (51) C07D 207/16<br />

C07D 405/14 → (51) C07D 401/12<br />

C07D 407/04 → (51) C07D 401/04<br />

(51) C07D 4<strong>09</strong>/06 (11) 2 421 858 A1*<br />

A61K 31/5415 A61P 31/00<br />

(25) En (26) En<br />

(21) 10713994.1 (22) 20.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/055176 20.04.2010<br />

(87) WO 2010/12<strong>2012</strong> 2010/43 28.10.2010<br />

(30) 20.04.20<strong>09</strong> EP <strong>09</strong>158229<br />

20.04.20<strong>09</strong> US 202918 P<br />

(54) THIOXANTHENDERIVATE ZUR BEHAND-<br />

LUNG VON INFEKTIONSKRANKHEITEN<br />

THIOXANTHENE DERIVATIVES FOR THE<br />

TREATMENT OF INFECTIOUS DISEASES<br />

DÉRIVÉS DE THIOXANTHÈNE POUR LE<br />

TRAITEMENT DE MALADIES INFEC-<br />

TIEUSES<br />

(71) BKG Pharma ApS, Birgit Kjoldgaard<br />

Giwercman Vintervej 2, 2920 Charlottenlund,<br />

DK<br />

(72) GIWERCMAN, Birgit, Kjældgaard, DK-2920<br />

Charlottenlund, DK<br />

(74) Bender, Mikkel, et al, Chas. Hude A/S <strong>Patent</strong><br />

H.C. Andersens Boulevard 33, 1780<br />

Copenhagen, DK<br />

C07D 4<strong>09</strong>/06 → (51) C07D 205/04<br />

C07D 4<strong>09</strong>/06 → (51) C07D 401/06<br />

C07D 4<strong>09</strong>/06 → (51) C07D 401/10<br />

C07D 4<strong>09</strong>/06 → (51) C07D 405/06<br />

C07D 4<strong>09</strong>/10 → (51) C07D 401/10<br />

C07D 4<strong>09</strong>/12 → (51) C07D 205/04<br />

C07D 4<strong>09</strong>/12 → (51) C07D 401/12<br />

C07D 4<strong>09</strong>/14 → (51) C07D 205/04<br />

C07D 4<strong>09</strong>/14 → (51) C07D 207/16<br />

C07D 4<strong>09</strong>/14 → (51) C07D 401/04<br />

C07D 4<strong>09</strong>/14 → (51) C07D 401/12<br />

C07D 413/06 → (51) C07D 401/10<br />

C07D 413/12 → (51) C07D 205/04<br />

C07D 413/12 → (51) C07D 207/16<br />

86<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />

C07D 413/12 → (51) C07D 213/81<br />

C07D 413/12 → (51) C07D 231/14<br />

C07D 413/12 → (51) C07D 401/12<br />

C07D 413/14 → (51) C07D 205/04<br />

C07D 413/14 → (51) C07D 231/14<br />

C07D 413/14 → (51) C07D 401/12<br />

C07D 413/14 → (51) C07D 403/14<br />

(51) C07D 417/04 (11) 2 421 859 A1*<br />

C07F 9/38 A61K 31/496<br />

A61P 7/02 A61P 9/10<br />

(25) En (26) En<br />

(21) 10719<strong>09</strong>7.7 (22) 21.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) IB 2010/051742 21.04.2010<br />

(87) WO 2010/122504 2010/43 28.10.2010<br />

(30) 22.04.20<strong>09</strong> PCT/IB20<strong>09</strong>/051647<br />

(54) THIAZOLDERIVATE UND IHRE VERWEN-<br />

DUNG ALS P2Y12-REZEPTORANTAGO-<br />

NISTEN<br />

THIAZOLE DERIVATIVES AND THEIR USE<br />

AS P2Y12 RECEPTOR ANTAGONISTS<br />

DÉRIVÉS DE THIAZOLE ET LEURS UTILI-<br />

SATION COMME ANTAGONISTES DU<br />

RECEPTEUR P2Y12<br />

(71) Actelion Pharmaceuticals Ltd., Gewerbestrasse<br />

16, 4123 Allschwil, CH<br />

(72) CAROFF, Eva, CH-4123 Allschwil, CH<br />

HILPERT, Kurt, CH-4123 Allschwil, CH<br />

HUBLER, Francis, CH-4123 Allschwil, CH<br />

LEHMANN, David, CH-4123 Allschwil, CH<br />

MEYER, Emmanuel, CH-4123 Allschwil, CH<br />

RENNEBERG, Dorte, CH-4123 Allschwil, CH<br />

(74) Gschwend, Thomas Peter, Actelion Pharmaceuticals<br />

Ltd Gewerbestrasse 16, CH-4123<br />

Allschwil, CH<br />

C07D 417/06 → (51) C07D 205/04<br />

C07D 417/06 → (51) C07D 401/06<br />

C07D 417/06 → (51) C07D 401/10<br />

(51) C07D 417/12 (11) 2 421 860 A1*<br />

C07D 417/14 A61K 31/496<br />

A61P 25/00 A61P 29/00<br />

(25) En (26) En<br />

(21) 10715456.9 (22) 22.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) US 2010/032045 22.04.2010<br />

(87) WO 2010/124082 2010/43 28.10.2010<br />

(30) 22.04.20<strong>09</strong> US 171649 P<br />

22.04.20<strong>09</strong> US 171658 P<br />

(54) AZETIDINYLDIAMIDE ALS MONOACYL-<br />

GLYCERINLIPASEINHIBITOREN<br />

AZETIDINYL DIAMIDES AS MONOACYL-<br />

GLYCEROL LIPASE INHIBITORS<br />

AZÉTIDINYL DIAMIDES EN TANT QU'IN-<br />

HIBITEURS DE LA MONOACYLGLYCÉROL<br />

LIPASE<br />

(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) BIAN, Haiyan, Princeton NJ 08540, US<br />

CHEVALIER, Kristen, M., Collegeville PA<br />

19426, US<br />

CONNOLLY, Peter, J., Spring House PA<br />

19477, US

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