(C07D) I.1(1) HUTCHINSON, Douglas K., Antioch Illinois 60002-1863, US KATI, Warren M., Gurnee Illinois 60031, US KRUEGER, Allan C., Gurnee Illinois 60031, US LIU, Dachun, Waukegan, Illinois 60085, US LONGENECKER, Kenton L., Grayslake Illinois 60030, US PRATT, John K., Kenosha Wisconsin 53142, US STEWART, Kent D., Gurnee Illinois 60031, US WAGNER, Rolf, Antioch Illinois 60002, US MARING, Clarence, J., Palatine, Illinois 60067, US (74) Modiano, Micaela Nadia, et al, Modiano & Partners Thierschstrasse 11, 80538 München, DE C07D 401/04 → (51) C07D 205/04 C07D 401/04 → (51) C07D 207/16 (51) C07D 401/06 (11) 2 421 846 A1* C07D 401/14 A61K 31/444 A61K 31/496 A61K 31/5377 A61P 35/00 A61P 37/00 A61P 29/00 A61P 31/00 (25) En (26) En (21) 10714016.2 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR BA ME (86) EP 2010/055293 21.04.2010 (87) WO 2010/122069 2010/43 28.10.2010 (30) 21.04.2009 EP 09158327 (54) 5-ALKINYLPYRIDINE 5-ALKYNYL-PYRIDINES 5-ALCYNYLPYRIDINES (71) Boehringer Ingelheim International GmbH, Binger Strasse 173, 55216 Ingelheim am Rhein, DE (72) WUNBERG, Tobias, 55216 Ingelheim am Rhein, DE SCHNEIDER, Siegfried, 55216 Ingelheim am Rhein, DE VAN DER VEEN, Lars, 55216 Ingelheim am Rhein, DE (74) Hammann, Heinz, et al, Boehringer Ingelheim GmbH Corporate Patents Binger Strasse 173, 55216 Ingelheim am Rhein, DE (51) C07D 401/06 (11) 2 421 847 A1* C07D 417/06 C07D 205/04 C07D 401/12 C07D 409/06 A61K 31/496 A61P 25/00 A61P 29/00 (25) En (26) En (21) 10717365.0 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032092 22.04.2010 (87) WO 2010/124116 2010/43 28.10.2010 (30) 22.04.2009 US 171658 P 22.04.2009 US 171649 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS DIAMIDES D'AZÉTIDINYLE INHIBITRICES DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US Europäisches Patentblatt EuropeanPatentBulletinBulletin européen des brevets CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Yue-mei, Spring House PA 19477, US ZHANG, Sui-po, Exton PA 19341, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, Carpmaels & Ransford One Southampton Row, London WC1B 5HA, GB C07D 401/06 → (51) C07D 205/04 C07D 401/06 → (51) C07D 207/16 C07D 401/06 → (51) C07D 241/16 (51) C07D 401/10 (11) 2 421 848 A1* C07D 403/04 C07D 403/06 C07D 403/10 C07D 405/06 C07D 409/06 C07D 409/10 C07D 413/06 C07D 417/06 A61K 31/496 A61P 29/00 A61P 25/00 (25) En (26) En (21) 10715461.9 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032095 22.04.2010 (87) WO 2010/124119 2010/43 28.10.2010 (30) 22.04.2009 US 171649 P 22.04.2009 US 171658 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS AZÉTIDINYL DIAMIDES EN TANT QU'IN- HIBITEURS DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-Chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Sui-Po, Exton PA 19341, US ZHANG, Yue-Mei, Spring House PA 19477, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US 84 Anmeldungen Applications Demandes (09/2012) 29.02.2012 (74) Warner, James Alexander, et al, Carpmaels & Ransford One Southampton Row, GB- London WC1B 5HA, GB C07D 401/10 → (51) C07D 205/04 (51) C07D 401/12 (11) 2 421 849 A1* A61K 31/444 A61P 11/00 A61P 11/08 (25) En (26) En (21) 10715058.3 (22) 16.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) US 2010/031356 16.04.2010 (87) WO 2010/123766 2010/43 28.10.2010 (30) 23.04.2009 US 172039 P (54) DIAMIDVERBINDUNGEN, DIE ALS ANTA- GONISTEN AM MUSKARINREZEPTOR ALS AGONISTEN AM & 946; 2-ADRE- NERGEN REZEPTOR WIRKEN DIAMIDE COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY COMPOSES DIAMIDES AYANT UN ANTA- GONISTE DU RECEPTEUR MUSCARI- NIQUE ET UNE ACTIVITE AGONISTE DES RECEPTEURS ADRENERGIQUES BETA2 (71) Theravance, Inc., 901 Gateway Boulevard, South San Francisco, CA 94080, US (72) HUGHES, Adam, Belmont California 94002, US BYUN, Daniel, Alameda California 94501, US CHEN, Yan, Burlingame California 94010, US FLEURY, Melissa, San Mateo California 94404, US JACOBSEN, John, R., San Mateo California 94402, US STANGELAND, Eric, L., Pacifica California 94044, US WILSON, Richard, D., Orinda California 94563, US YEN, Rose, San Francisco California 94110, US (74) Scott, Susan Margaret, et al, Abel & Imray 20 Red Lion Street, London WC1R 4PQ, GB (51) C07D 401/12 (11) 2 421 850 A1* C07D 403/14 C07D 413/14 C07D 417/14 A61K 31/44 A61K 31/501 A61K 31/506 A61P 3/04 A61P 25/22 A61P 25/24 A61P 25/30 (25) En (26) En (21) 10715239.9 (22) 23.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) EP 2010/055449 23.04.2010 (87) WO 2010/122151 2010/43 28.10.2010 (30) 24.04.2009 GB 0907112 17.06.2009 GB 0910483 22.12.2009 GB 0922472 (54) ALS OREXINANTAGONISTEN VERWEN- DETE 3-AZABICYCLO[4.1.0]HEPTANE 3 -AZABICYCLO [4.1.0]HEPTANES USED AS OREXIN ANTAGONISTS 3 -AZABICYCLO [4.1.0]HEPTANES UTILISÉS COMME ANTAGONISTES DE L'OREXINE (71) Glaxo Group Limited, Glaxo Wellcome House Berkeley Avenue Greenford, Middlesex UB6 0NN, GB (72) AMANTINI, David, I-37135 Verona, IT FERRONI, Francesco, I-37135 Verona, IT GIANOTTI, Massimo, I-37135 Verona, IT PAVONE, Francesca, I-37135 Verona, IT
(C07D) I.1(1) DI FABIO, Romano, 37135 Verona, IT (74) Lawrence, Geoffrey Mark Prouse, GlaxoSmithKline Corporate Intellectual Property (CN925.1) 980 Great West Road, Brentford Middlesex TW8 9GS, GB (51) C07D 401/12 (11) 2 421 851 A1* C07D 403/12 C07D 403/14 C07D 409/12 C07D 417/12 C07D 417/14 C07D 495/04 A61K 31/496 A61P 25/00 A61P 29/00 (25) En (26) En (21) 10716203.4 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032068 22.04.2010 (87) WO 2010/124102 2010/43 28.10.2010 (30) 22.04.2009 US 171658 P 22.04.2009 US 171649 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS AZÉTIDINYL DIAMIDES EN TANT QU'IN- HIBITEURS DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica, N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-Chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Sui-Po, Exton PA 19341, US ZHANG, Yue-Mei, Spring House PA 19477, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, et al, Carpmaels & Ransford One Southampton Row, London WC1B 5HA, GB (51) C07D 401/12 (11) 2 421 852 A1* C07D 401/14 C07D 403/12 C07D 403/14 C07D 405/14 C07D 409/12 C07D 409/14 C07D 413/12 C07D 417/12 A61K 31/496 A61P 29/00 A61P 25/00 (25) En (26) En (21) 10719479.7 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032098 22.04.2010 (87) WO 2010/124121 2010/43 28.10.2010 (30) 22.04.2009 US 171660 P (54) HETEROAROMATISCHE UND AROMATI- SCHE PIPERAZINYLAZETIDINYLAMIDE ALS MONOACYLGLYCERINLIPASEINHI- BITOR HETEROAROMATIC AND AROMATIC PIPERAZINYL AZETIDINYL AMIDES AS Europäisches Patentblatt EuropeanPatentBulletinBulletin européen des brevets MONOACYLGLYCEROL LIPASE INHIBITOR PIPÉRAZINYL AZÉTIDINYL AMIDES HÉTÉROAROMATIQUES ET AROMATI- QUES EN TANT QU'INHIBITEUR DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) CHEVALIER, Kristen, M., Collegeville PA 19426, US DAX, Scott, L., Landenberg PA 19350, US FLORES, Christopher, M., Spring House PA 19477, US LIU, Li, Doylestown PA 18901, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Landsdale PA 19446, US NELEN, Marina, I., Exton PA 19341, US PROUTY, Stephen, PA 19104, US TODD, Matthew, Exton PA 19341, US ZHANG, Sui-Po, Exton PA 19341, US ZHU, Bin, Spring House PA 19477, US NULTON, Erica, L., Exton PA 19341, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, Carpmaels & Ransford One Southampton Row, London WC1B 5HA, GB C07D 401/12 → (51) C07D 205/04 C07D 401/12 → (51) C07D 207/16 C07D 401/12 → (51) C07D 211/46 C07D 401/12 → (51) C07D 401/06 C07D 401/14 → (51) C07D 205/04 C07D 401/14 → (51) C07D 207/16 C07D 401/14 → (51) C07D 401/06 C07D 401/14 → (51) C07D 401/12 C07D 403/04 → (51) C07D 207/16 C07D 403/04 → (51) C07D 211/96 C07D 403/04 → (51) C07D 401/04 C07D 403/04 → (51) C07D 401/10 (51) C07D 403/06 (11) 2 421 853 A1* (25) En (26) En (21) 09751896.3 (22) 09.11.2009 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2009/064850 09.11.2009 (87) WO 2010/121673 2010/43 28.10.2010 (30) 22.04.2009 IT MI20090678 (54) SYNTHESE VON 3-{[(2R)-1-METHYLPYR- ROLIDIN-2-YL]METHYL}-5- [2-(PHENYL- SULFONYL)ETHYL]-1H-INDOL SYNTHESIS OF 3-{[(2R)-1-METHYLPYR- ROLIDIN-2-YL]METHYL}-5-[2-(PHENYL- SULFONYL)ETHYL]-1H-INDOLE SYNTHÈSE DE 3-{[(2R)-1-MÉTHYLPYR- ROLIDIN-2-YL]MÉTHYL}-5-[2-(PHÉNYL- SULFONYL)ÉTHYL]-1H-INDOLE (71) F.I.S. Fabbrica Italiana Sintetici S.p.A., Viale Milano, 26, 36075 Alte di Montecchio Maggiore, IT (72) SERAFINI, Siro, I-36100 Vicenza, IT CASTELLIN, Andrea, I-35035 Mestrino Padova, IT DAL SANTO, Claudio, I-36040 Sarego Vicenza, IT 85 Anmeldungen Applications Demandes (09/2012) 29.02.2012 (74) Long, Giorgio, et al, Jacobacci & Partners S.p.A. Via Senato 8, 20121 Milano, IT C07D 403/06 → (51) C07D 205/04 C07D 403/06 → (51) C07D 207/16 C07D 403/06 → (51) C07D 401/10 C07D 403/10 → (51) C07D 205/04 C07D 403/10 → (51) C07D 401/10 C07D 403/12 → (51) C07D 205/04 C07D 403/12 → (51) C07D 207/16 C07D 403/12 → (51) C07D 401/12 C07D 403/12 → (51) C07D 487/04 (51) C07D 403/14 (11) 2 421 854 A1* C07D 413/14 A61K 31/5513 A61K 31/553 A61P 29/00 (25) En (26) En (21) 10714295.2 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055227 21.04.2010 (87) WO 2010/122038 2010/43 28.10.2010 (30) 24.04.2009 US 172288 P (54) HEMMER DER BRUTON-TYROSINKINASE INHIBITORS OF BRUTON'S TYROSINE KINASE INHIBITEURS DE LA TYROSINE KINASE DE BRUTON (71) F.Hoffmann-La Roche AG, Grenzacherstrasse 124, 4070 Basel, CH (72) DEWDNEY, Nolan James, Repulse Bay, HK HAWLEY, Ronald Charles, Glen Ridge New Jersey 07028, US KONDRU, Rama K., Morris Plains New Jersey 07950, US LAI, Yingjie, Cupertino California 95014, US LOU, Yan, Clifton New Jersey 07012, US (74) Sauer, Frank, F. Hoffmann-La Roche AG Patent Department Grenzacherstrasse 124, 4070 Basel, CH (51) C07D 403/14 (11) 2 421 855 A1* A61K 31/4178 A61P 31/14 (25) En (26) En (21) 10715243.1 (22) 23.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055482 23.04.2010 (87) WO 2010/122162 2010/43 28.10.2010 (30) 24.04.2009 EP 09158676 (54) DIARYLETHER DIARYL ETHERS ETHERS DE DIARYLE (71) Tibotec Pharmaceuticals, Eastgate Village Eastgate Little Island, Co Cork, IE (72) DEMIN, Samuël, Dominique, B-2800 Mechelen, BE MC GOWAN, David, B-1150 Brussel, BE LAST, Stefaan, Julien, B-2547 Lint, BE RABOISSON, Pierre, Jean-Marie, Bernard, B- 1331 Rosieres, BE (74) Daelemans, Frank F.R., J&J Patent Law Department Turnhoutseweg 30, 2340 Beerse, BE C07D 403/14 → (51) C07D 205/04 C07D 403/14 → (51) C07D 207/16
(71) Glaxo Group Limited, Glaxo Wellcome House<br />
Berkeley Avenue Greenford, Middlesex UB6<br />
0NN, GB<br />
(72) AMANTINI, David, I-37135 Verona, IT<br />
FERRONI, Francesco, I-37135 Verona, IT<br />
GIANOTTI, Massimo, I-37135 Verona, IT<br />
PAVONE, Francesca, I-37135 Verona, IT
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