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European Patent Bulletin 2012/09 - European Patent Office

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(C07D) I.1(1)<br />

ANTAGONISTES CCR3 D'ARYLSULFONA-<br />

MIDES<br />

(71) Axikin Pharmaceuticals, Inc., 10835 Road to<br />

the Cure, Suite 250, San Diego, CA 92121,<br />

US<br />

(72) LY, Tai, Wei, San Diego CA 92131, US<br />

FORRESTER, Jared, Andrew, Castle Rock CO<br />

80108, US<br />

(74) Ritter, Thomas Kurt, et al, Jones Day Prinzregentenstraße<br />

11, 80538 München, DE<br />

C07D 295/26 → (51) C07D 211/96<br />

C07D 301/03 → (51) C07D 301/22<br />

C07D 301/04 → (51) C07D 301/22<br />

(51) C07D 301/10 (11) 2 421 839 A1*<br />

(25) En (26) En<br />

(21) 10714400.8 (22) 05.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/029948 05.04.2010<br />

(87) WO 2010/123675 2010/43 28.10.2010<br />

(30) 21.04.20<strong>09</strong> US 171207 P<br />

(54) VERFAHREN ZUR VERBESSERUNG DER<br />

EFFIZIENZ VON KATALYSATOREN FÜR<br />

DIE RHENIUMUNTERSTÜTZTE EPOXIDIE-<br />

RUNG UND EPOXIDIERUNGSVERFAH-<br />

REN, BEI DENEN DIESE ANGEWANDT<br />

WERDEN<br />

METHODS FOR ENHANCING THE EFFI-<br />

CIENCY OF RHENIUM-PROMOTED EPOX-<br />

IDATION CATALYSTS AND EPOXIDATION<br />

METHODS UTILIZING THESE<br />

PROCÉDÉS POUR AMÉLIORER L'EFFICA-<br />

CITÉ DE CATALYSEURS D'ÉPOXYDATION<br />

À PROMOTEUR RHÉNIUM ET PROCÉDÉS<br />

D'ÉPOXYDATION UTILISANT CES<br />

PROCÉDÉS<br />

(71) Dow Technology Investments LLC, 2020<br />

Dow Center, Midland, MI 48674, US<br />

(72) LIU, Albert Cheng-Yu, Charleston West<br />

Virginia 25311, US<br />

ZHANG, Liping, Lake Jackson Texas 77566,<br />

US<br />

(74) Raynor, John, et al, Beck Greener Fulwood<br />

House 12 Fulwood Place, London WC1V<br />

6HR, GB<br />

(51) C07D 301/10 (11) 2 421 840 A1*<br />

(25) En (26) En<br />

(21) 10718767.6 (22) 20.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/031668 20.04.2010<br />

(87) WO 2010/123842 2010/43 28.10.2010<br />

(30) 21.04.20<strong>09</strong> US 171248 P<br />

(54) VEREINFACHTES VERFAHREN ZUR HER-<br />

STELLUNG VON ALKYLENOXIDEN MIT<br />

BEI DER ALTERUNG HOCHEFFIZIENTEM<br />

KATALYSATOR<br />

SIMPLIFIED METHOD FOR PRODUCING<br />

ALKYLENE OXIDES WITH A HIGH EFFI-<br />

CIENCY CATALYST AS IT AGES<br />

PROCÉDÉ SIMPLIFIÉ DE PRODUCTION<br />

D'OXYDES D'ALKYLÈNE AVEC UN CATA-<br />

LYSEUR HAUTE EFFICACITÉ AU FUR ET À<br />

MESURE DE SON VIEILLISSEMENT<br />

(71) Dow Technology Investments LLC, 2020<br />

Dow Center, Midland, MI 48674, US<br />

(72) ZHANG, Liping, Lake Jackson Texas 77566,<br />

US<br />

SOO, Hwaili, Charleston West Virginia<br />

25314, US<br />

HENSTOCK, William, Charleston West<br />

Virginia 25314, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) Raynor, John, Beck Greener Fulwood House<br />

12 Fulwood Place, London WC1V 6HR, GB<br />

(51) C07D 301/10 (11) 2 421 841 A1*<br />

A61K 31/336<br />

(25) En (26) En<br />

(21) 10732499.8 (22) 20.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/031673 20.04.2010<br />

(87) WO 2010/123844 2010/43 28.10.2010<br />

(30) 21.04.20<strong>09</strong> US 171284 P<br />

(54) VERBESSERTES VERFAHREN ZUR HER-<br />

STELLUNG UND AUFRECHTERHALTUNG<br />

EINES SPEZIFISCHEN PARAMETERS FÜR<br />

DIE ALKYLENOXIDHERSTELLUNG MIT<br />

EINEM HOCHEFFIZIENTEN KATALYSA-<br />

TOR<br />

IMPROVED METHOD OF ACHIEVING AND<br />

MAINTAINING A SPECIFIED ALKYLENE<br />

OXIDE PRODUCTION PARAMETER WITH<br />

A HIGH EFFICIENCY CATALYST<br />

PROCÉDÉ PERFECTIONNÉ POUR<br />

OBTENIR ET MAINTENIR UN PARA-<br />

MÈTRE DE PRODUCTION D'OXYDE L'AL-<br />

KYLÈNE SPÉCIFIÉ AVEC UN CATALY-<br />

SEUR À HAUT RENDEMENT<br />

(71) Dow Technology Investments LLC, 2020<br />

Dow Center, Midland, MI 48674, US<br />

(72) ZHANG, Liping, Lake Jackson Texas 77566,<br />

US<br />

LIU, Albert, Charleston West Virginia 25311,<br />

US<br />

HABENSCHUSS, Michael, South Charleston<br />

West Virginia 25303, US<br />

(74) Raynor, John, Beck Greener Fulwood House<br />

12 Fulwood Place, London WC1V 6HR, GB<br />

(51) C07D 301/22 (11) 2 421 842 A1*<br />

C07D 301/03 C07D 301/04<br />

(25) En (26) En<br />

(21) 10719457.3 (22) 20.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/031694 20.04.2010<br />

(87) WO 2010/123856 2010/43 28.10.2010<br />

(30) 21.04.20<strong>09</strong> US 171104 P<br />

(54) EPOXIDATIONSREAKTIONEN UND BE-<br />

DINGUNGEN FÜR DEREN DURCHFÜH-<br />

RUNG<br />

EPOXIDATION REACTIONS AND<br />

OPERATING CONDITIONS THEREOF<br />

RÉACTIONS D'ÉPOXYDATION ET LEURS<br />

CONDITIONS D'EXPLOITATION<br />

(71) Dow Technology Investments LLC, 2020<br />

Dow Center, Midland, MI 48674, US<br />

(72) HABENSCHUSS, Michael, South Charleston<br />

WV 25303, US<br />

SOO, Hwaili, Charleston WV 25314, US<br />

HINMAN, Paul, Charleston WV 25314, US<br />

LIU, Albert, Charleston WV 25311, US<br />

(74) Raynor, John, Beck Greener Fulwood House<br />

12 Fulwood Place, London WC1V 6HR, GB<br />

(51) C07D 313/12 (11) 2 421 843 A2*<br />

A61K 31/335<br />

(25) En (26) En<br />

(21) 107<strong>09</strong>754.5 (22) 23.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/053783 23.03.2010<br />

(87) WO 2010/121877 2010/43 28.10.2010<br />

(88) 10.03.2011<br />

(30) 21.04.20<strong>09</strong> IT MI20<strong>09</strong>0659<br />

(54) VERFAHREN ZUR HERSTELLUNG VON<br />

OLOPATADIN<br />

83<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />

PROCESS FOR THE PREPARATION OF<br />

OLOPATADINE<br />

PROCÉDÉ DE PRÉPARATION DE L'OLO-<br />

PATADINE<br />

(71) F.I.S. Fabbrica Italiana Sintetici S.p.A., Viale<br />

Milano, 26, 36075 Alte di Montecchio Maggiore,<br />

IT<br />

(72) CASTELLIN, Andrea, I-35035 Mestrino PA-<br />

DOVA, IT<br />

FERRARI, Clark, I-36070 Brogliano VI-<br />

CENZA, IT<br />

GALVAGNI, Marco, I-37131 Verona, IT<br />

(74) Mozzi, Matteo, et al, Jacobacci & Partners<br />

S.p.A. Via Senato, 8, <strong>2012</strong>1 Milano, IT<br />

C07D 317/12 → (51) C07C 43/305<br />

C07D 317/58 → (51) C07C 233/08<br />

C07D 319/06 → (51) C07C 43/305<br />

(51) C07D 333/38 (11) 2 421 844 A1*<br />

C07D 333/40 A61K 31/381<br />

A61P 29/00 A61P 35/00<br />

A61P 37/00<br />

(25) En (26) En<br />

(21) 10714660.7 (22) 20.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) GB 2010/000790 20.04.2010<br />

(87) WO 2010/122294 2010/43 28.10.2010<br />

(30) 24.04.20<strong>09</strong> GB <strong>09</strong>07120<br />

(54) THIOPHENE ALS INHIBITOREN VON IKK-<br />

B-SERIN/THREONIN-PROTEINKINASE<br />

THIOPHENE INHIBITORS OF IKK-B<br />

SERINE-THREONINE PROTEIN KINASE<br />

INHIBITEURS THIOPHÈNES DE LA<br />

SÉRINE-THRÉONINE PROTÉINE KINASE<br />

IKK-<br />

(71) Chroma Therapeutics Ltd., 93 Milton Park,<br />

Abingdon Oxfordshire OX14 4RY, GB<br />

(72) DRUMMOND, Alan, Hastings, Abingdon,<br />

Oxfordshire OX14 4RY, GB<br />

TESTAR, Richard, James, Abingdon,<br />

Oxfordshire OX14 4RY, GB<br />

(74) Simons, Amanda Louise, J.A. Kemp & Co.<br />

14 South Square Gray's Inn, London WC1R<br />

5JJ, GB<br />

C07D 333/40 → (51) C07D 333/38<br />

(51) C07D 401/04 (11) 2 421 845 A1*<br />

C07D 403/04 C07D 407/04<br />

C07D 4<strong>09</strong>/14 A61K 31/513<br />

A61P 31/12<br />

(25) En (26) En<br />

(21) 10712220.2 (22) 25.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/028561 25.03.2010<br />

(87) WO 2010/111437 2010/39 30.<strong>09</strong>.2010<br />

(30) 25.03.20<strong>09</strong> US 163157 P<br />

(54) ANTIVIRALE VERBINDUNGEN UND AN-<br />

WENDUNGEN DAVON<br />

ANTIVIRAL COMPOUNDS AND USES<br />

THEREOF<br />

COMPOSÉS ANTIVIRAUX ET LEURS<br />

UTILISATIONS<br />

(71) Abbott Laboratories, 100 Abbott Park Rd.,<br />

Abbott Park, IL 60064, US<br />

(72) ROCKWAY, Todd W., Gurnee Illinois 60030,<br />

US<br />

BETEBENNER, David A., Libertyville Illinois<br />

60048, US<br />

DEGOEY, David A., Salem Wisconsin 53168,<br />

US<br />

FLENTGE, Charles A., Salem Wisconsin<br />

53168, US

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