European Patent Bulletin 2012/09 - European Patent Office
European Patent Bulletin 2012/09 - European Patent Office European Patent Bulletin 2012/09 - European Patent Office
(C07C) I.1(1) LANDWIRTSCHAFTLICHEN FORMULIE- RUNGEN NITROGEN CONTAININIG ISETHIONIC ACID SALT IN REGISTERABLE, STABLE AGRICULTURAL FORMULATIONS AZOTE CONTENANT UN SEL D'ACIDE ISÉTHIONIQUE PRÉSENT DANS DES PRÉPARATIONS AGRICOLES STABLES, HOMOLOGABLES (71) Huntsman Petrochemical LLC, 10003 Woodloch Forest Drive, The Woodlands, TX 77380, US (72) TANN, R., Scott, Sugar Land, TX 77478, US STRIDDE, Howard, M., Shiner, TX 77984, US (74) Van Steenlandt, Wim August Maria, et al, Huntsman (Europe) BVBA Intellectual Property Department Everslaan 45, 3078 Everberg, BE C07C 233/10 → (51) C07C 233/08 C07C 233/19 → (51) C07C 233/08 C07C 233/21 → (51) C07C 233/08 C07C 233/48 → (51) C07C 233/08 C07C 233/54 → (51) C07C 233/08 (51) C07C 245/20 (11) 2 421 822 A1* C07C 37/14 C07C 39/15 C07C 39/19 (25) De (26) De (21) 10714884.3 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055347 22.04.2010 (87) WO 2010/122105 2010/43 28.10.2010 (30) 22.04.2009 EP 09158489 (54) VERFAHREN ZUR HERSTELLUNG EINES KREUZKUPPLUNGSPRODUKTES EINES BENZOLISCHEN DIAZONIUMSALZES METHOD FOR PRODUCING A CROSS- COUPLING PRODUCT OF A BENZENOID DIAZONIUM SALT PROCÉDÉ DE FABRICATION D'UN PRODUIT DE COUPLAGE CROISÉ D'UN SEL BENZÉNIQUE DE DIAZONIUM (71) Zylum Beteiligungsgesellschaft mbH & Co. Patente II KG, Berliner Strasse 1, 12529 Schönfeld/OT Waltersdorf, DE (72) BOEGE, Nicolas, 20149 Hamburg, DE KREIPL, Andreas, 20359 Hamburg, DE SCHMIDT, Bernd, 14482 Potsdam, DE HOELTER, Frank, 14473 Potsdam, DE BERGER, René, 14471 Potsdam, DE (74) Held, Stephan, Meissner, Bolte & Partner GbR Widenmayerstraße 48, D-80538 München, DE C07C 255/42 → (51) C07C 233/08 C07C 255/58 → (51) C07C 233/08 C07C 257/12 → (51) C07D 211/46 C07C 263/10 → (51) C07C 209/78 C07C 265/14 → (51) C07C 209/78 C07C 309/08 → (51) A01N 41/04 C07C 309/66 → (51) C07C 209/74 C07C 311/29 → (51) C07D 211/96 Europäisches Patentblatt European Patent Bulletin Bulletin européen des brevets (51) C07D 205/04 (11) 2 421 823 A1* C07D 401/10 C07D 401/12 C07D 403/12 C07D 403/14 C07D 405/12 C07D 409/14 A61K 31/496 A61P 25/00 C07D 417/12 A61P 29/00 C07D 417/14 C07D 491/048 (25) En (26) En (21) 10715457.7 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032049 22.04.2010 (87) WO 2010/124086 2010/43 28.10.2010 (30) 22.04.2009 US 171649 P 22.04.2009 US 171658 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS AZÉTIDINYL DIAMIDES SERVANT D'IN- HIBITEURS DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Sui-Po, Exton PA 19341, US ZHANG, Yue-mei, Spring House PA 19477, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, Carpmaels & Ransford One Southampton Row, GB- London WC1B 5HA, GB (51) C07D 205/04 (11) 2 421 824 A1* C07D 401/04 C07D 401/06 C07D 401/10 C07D 403/06 C07D 403/10 C07D 403/12 C07D 405/12 C07D 409/06 C07D 417/06 C07D 417/14 A61K 31/496 A61P 25/00 A61P 29/00 (25) En (26) En (21) 10715460.1 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032089 22.04.2010 (87) WO 2010/124114 2010/43 28.10.2010 (30) 22.04.2009 US 171658 P 22.04.2009 US 171649 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS DIAMIDES D'AZÉTIDINYLE UTILISÉES COMME INHIBITEUR DE LA MONOACYL- GLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE 80 Anmeldungen Applications Demandes (09/2012) 29.02.2012 (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Yue-mei, Spring House PA 19477, US ZHANG, Sui-po, Exton PA 19341, US CLEMENTE, Jose, Exton PA 19341, US ZHU, Bin, Spring House PA 19477, US (74) Warner, James Alexander, et al, Carpmaels & Ransford One Southampton Row, London WC1B 5HA, GB (51) C07D 205/04 (11) 2 421 825 A1* C07D 401/14 C07D 403/12 C07D 405/12 C07D 405/14 C07D 409/12 C07D 409/14 C07D 413/12 C07D 413/14 C07D 417/12 C07D 417/14 C07D 495/04 A61K 31/496 A61P 29/00 A61P 25/00 (25) En (26) En (21) 10716205.9 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/032082 22.04.2010 (87) WO 2010/124108 2010/43 28.10.2010 (30) 22.04.2009 US 171649 P 22.04.2009 US 171658 P (54) AZETIDINYLDIAMIDE ALS MONOACYL- GLYCERINLIPASEINHIBITOREN AZETIDINYL DIAMIDES AS MONOACYL- GLYCEROL LIPASE INHIBITORS AZÉTIDINYL DIAMIDES EN TANT QU'IN- HIBITEURS DE LA MONOACYLGLYCÉROL LIPASE (71) Janssen Pharmaceutica N.V., Turnhoutseweg 30, 2340 Beerse, BE (72) BIAN, Haiyan, Princeton NJ 08540, US CHEVALIER, Kristen, M., Collegeville PA 19426, US CONNOLLY, Peter, J., Spring House PA 19477, US FLORES, Christopher, M., Spring House PA 19477, US LIN, Shu-chen, Doylestown PA 18902, US LIU, Li, Doylestown PA 18901, US MABUS, John, East Greenville PA 18041, US MACIELAG, Mark, J., Spring House PA 19477, US MCDONNELL, Mark, E., Lansdale PA 19446, US PITIS, Philip, M., North Wales PA 19454, US ZHANG, Sui-po, Exton PA 19341, US ZHANG, Yue-mei, Spring House PA 19477, US ZHU, Bin, Spring House PA 19477, US CLEMENTE, Jose, Exton PA 19341, US (74) Warner, James Alexander, Carpmaels & Ransford One Southampton Row, London WC1B 5HA, GB C07D 205/04 → (51) C07D 401/06
(C07D) I.1(1) C07D 205/06 → (51) C07D 405/06 (51) C07D 207/16 (11) 2 421 826 A1* C07D 401/04 C07D 401/06 C07D 401/12 C07D 401/14 C07D 403/04 C07D 403/06 C07D 403/12 C07D 403/14 C07D 405/04 C07D 405/06 C07D 405/12 C07D 405/14 C07D 409/14 C07D 413/12 (25) En (26) En (21) 10713457.9 (22) 13.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR RS (86) EP 2010/054792 13.04.2010 (87) WO 2010/121918 2010/43 28.10.2010 (30) 20.04.2009 EP 09158212 (54) PROLINDERIVATE ALS KATHEPSININHI- BITOREN PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS DÉRIVÉS DE PROLINE COMME INHIBI- TEURS DE LA CATHEPSINE (71) F.Hoffmann-La Roche AG, Grenzacherstrasse 124, 4070 Basel, CH (72) ALVAREZ SANCHEZ, Ruben, F-68128 Rosenau, FR BANNER, David, CH-4054 Basel, CH CECCARELLI, Simona M., CH-4057 Basel, CH GRETHER, Uwe, 79588 Efringen-Kirchen, DE HAAP, Wolfgang, 79540 Loerrach, DE HARTMAN, Peter, 79539 Loerrach, DE HARTMANN, Guido, 79539 Loerrach, DE HILPERT, Hans, CH-4142 Muenchenstein, CH KUEHNE, Holger, 79540 Loerrach, DE MAUSER, Harald, 79418 Schliengen, DE PLANCHER, Jean-Marc, F-68220 Hagenthalle-Bas, FR (74) Pomeranc, Didier, F. Hoffmann-La Roche AG Patent Department Grenzacherstrasse 124, 4070 Basel, CH (51) C07D 211/46 (11) 2 421 827 A2* C07C 257/12 C07D 401/12 (25) En (26) En (21) 10715333.0 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) GB 2010/050653 22.04.2010 (87) WO 2010/122340 2010/43 28.10.2010 (88) 09.09.2011 (30) 23.04.2009 US 171994 P (54) VERFAHREN ZUR HERSTELLUNG VON 4- (3-CHLOR-2-FLUORANILINO)-7-ME- THOXY-6-{-[1-(N-METHYLCARBAMOYL- METHYL)PIPERIDIN-4-YL]OXY}CHINAZO- LIN PROCESS FOR THE PREPARATION OF 4- (3-CHLORO-2-FLUORO- ANILINO)-7- METHOXY-6- { [1-(N-METHYLCARBA- MOYLMETHYL)- PIPERIDIN- 4-YL]OXY}- QUINAZOLINE PROCÉDÉ DE PRÉPARATION DE 4-(3- CHLORO-2-FLUORO- ANILINO)-7- MÉTHOXY-6- { [1-(N-MÉTHYLCARBA- MOYLMÉTHYL)- PIPÉRIDIN- 4-YL]OXY}- QUINAZOLINE (71) AstraZeneca AB, 151 85 Södertälje, SE (72) BOARDMAN, Kay, Alison, Macclesfield Cheshire SK10 2NA, GB CUNNINGHAM, Oliver, Robert, Macclesfield Cheshire SK10 2NA, GB Europäisches Patentblatt European Patent Bulletin Bulletin européen des brevets GOUNDRY, William, Macclesfield Cheshire SK10 2NA, GB LAFFAN, David, Dermot, Patrick, Macclesfield Cheshire SK10 2NA, GB (74) Bryant, Tracey, AstraZeneca AB, Global Intellectual Property, 151 85 Sodertalje, SE (51) C07D 211/60 (11) 2 421 828 A2* C07D 405/12 A61K 31/4468 A61P 9/04 A61P 9/02 A61P 9/10 A61P 11/00 A61P 13/12 (25) En (26) En (21) 10747951.1 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) IN 2010/000253 22.04.2010 (87) WO 2010/122580 2010/43 28.10.2010 (88) 16.12.2010 (30) 24.04.2009 IN MU10912009 (54) PIPERIDINDERIVATE ALS RENIN-INHIBI- TOREN PIPERIDINE DERIVATIVES AS INHI- BITORS OF RENIN DERIVATIFS DE PIPERIDINE COMME INHIBITEURS DE RÉNINE (71) Cadila Healthcare Limited, Zydus Tower Satellite Cross Roads, Ahmedabad 380 015, Gujarat, IN (72) THOMBARE, Pravain, Gujarat, IN DESAI, Jigar, Gujarat, IN JAIN, Mukul, R., Gujarat, IN (74) Jones, Helen M.M., Gill Jennings & Every LLP The Broadgate Tower 20 Primrose Street, London EC2A 2ES, GB (51) C07D 211/96 (11) 2 421 829 A2* C07D 241/04 C07D 243/08 C07D 403/04 C07D 487/04 C07D 295/26 C07C 311/29 A61K 31/445 A61P 25/28 A61P 11/06 (25) En (26) En (21) 10714821.5 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/031828 21.04.2010 (87) WO 2010/123956 2010/43 28.10.2010 (88) 09.09.2011 (30) 22.04.2009 US 171775 P (54) 2,5-DISUBSTITUIERTE ARYLSULFONA- MIDE ALS CCR3-ANTAGONISTEN 2,5-DISUBSTITUTED ARYLSULFO- NAMIDE CCR3 ANTAGONISTS ANTAGONISTES CCR3 D'ARYLSULFONA- MIDES 2,5-DISUBSTITUÉS (71) Axikin Pharmaceuticals, Inc., 10835 Road to the Cure, Suite 250, San Diego, CA 92121, US (72) LY, Tai, Wei, San Diego CA 92131, US TRAN, Marie Chantal, Siu-ying, Arcadia CA 91007, US RAAUM, Erik, Dean, Teton Village WY 83025, US (74) Ritter, Thomas Kurt, et al, Jones Day Prinzregentenstraße 11, 80538 München, DE (51) C07D 211/96 (11) 2 421 830 A2* C07D 241/04 C07D 241/08 C07D 295/26 A01N 43/62 A61K 31/18 A61P 11/02 A61P 25/28 A61P 29/00 (25) En (26) En 81 Anmeldungen Applications Demandes (09/2012) 29.02.2012 (21) 10714822.3 (22) 21.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR AL BA ME RS (86) US 2010/031832 21.04.2010 (87) WO 2010/123959 2010/43 28.10.2010 (88) 17.02.2011 (30) 22.04.2009 US 171626 P (54) 2,5-DISUBSTITUIERTE ARYLSULFONA- MID-CCR3-ANTAGONISTEN 2,5-DISUBSTITUTED ARYLSULFO- NAMIDE CCR3 ANTAGONISTS ANTAGONISTES CCR3 D'ARYLSULFONA- MIDES 2,5-DISUBSTITUÉS (71) Axikin Pharmaceuticals, Inc., 10835 Road to the Cure, Suite 250, San Diego, CA 92121, US (72) LY, Tai, Wei, San Diego CA 92131, US POTTER, Garrett, Thomas, San Diego CA 92122, US (74) Ritter, Thomas Kurt, et al, Jones Day Prinzregentenstraße 11, 80538 München, DE C07D 213/16 → (51) C07C 13/62 (51) C07D 213/64 (11) 2 421 831 A1* C07D 213/76 C07D 237/14 C07D 239/54 C07D 241/18 C07D 405/04 A61K 31/4412 A61K 31/50 A61K 31/513 A61K 31/4965 A61P 31/14 (25) En (26) En (21) 10715229.0 (22) 22.04.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) EP 2010/055309 22.04.2010 (87) WO 2010/122082 2010/43 28.10.2010 (30) 25.04.2009 US 172723 P (54) HETEROCYCLISCHE ANTIVIRALE VER- BINDUNGEN HETEROCYCLIC ANTIVIRAL COMPOUNDS COMPOSES ANTIVIRAUX HETEROCYCLI- QUES (71) F.Hoffmann-La Roche AG, Grenzacherstrasse 124, 4070 Basel, CH (72) LEE, Eun Kyung, San Jose California 95129, US SCHOENFELD, Ryan Craig, San Jose California 95117, US TALAMAS, Francisco Xavier, Mountain View California 94040, US (74) Halbig, Dirk, F. Hoffmann-La Roche AG Grenzacherstrasse 124, 4070 Basel, CH C07D 213/76 → (51) C07D 213/64 (51) C07D 213/81 (11) 2 421 832 A1* C07D 239/28 C07D 239/30 C07D 405/12 C07D 413/12 C07D 417/12 C07H 15/04 A01N 43/40 A01N 43/54 A01N 43/76 A01N 43/78 A01N 43/828 A01N 43/84 (25) En (26) En (21) 10706859.5 (22) 25.02.2010 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (86) US 2010/025342 25.02.2010 (87) WO 2010/099279 2010/35 02.09.2010 (30) 27.02.2009 US 156088 P (54) N-ALKOXYAMIDE VON 6-(SUBSTITUIER- TES PHENYL)-4-AMINOPICOLINATEN UND 2-(SUBSTITUIERTES PHENYL)-6- AMINO-4-PYRIMIDINCARBOXYLATEN
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(C07C) I.1(1)<br />
LANDWIRTSCHAFTLICHEN FORMULIE-<br />
RUNGEN<br />
NITROGEN CONTAININIG ISETHIONIC<br />
ACID SALT IN REGISTERABLE, STABLE<br />
AGRICULTURAL FORMULATIONS<br />
AZOTE CONTENANT UN SEL D'ACIDE<br />
ISÉTHIONIQUE PRÉSENT DANS DES<br />
PRÉPARATIONS AGRICOLES STABLES,<br />
HOMOLOGABLES<br />
(71) Huntsman Petrochemical LLC, 10003<br />
Woodloch Forest Drive, The Woodlands, TX<br />
77380, US<br />
(72) TANN, R., Scott, Sugar Land, TX 77478, US<br />
STRIDDE, Howard, M., Shiner, TX 77984,<br />
US<br />
(74) Van Steenlandt, Wim August Maria, et al,<br />
Huntsman (Europe) BVBA Intellectual<br />
Property Department Everslaan 45, 3078<br />
Everberg, BE<br />
C07C 233/10 → (51) C07C 233/08<br />
C07C 233/19 → (51) C07C 233/08<br />
C07C 233/21 → (51) C07C 233/08<br />
C07C 233/48 → (51) C07C 233/08<br />
C07C 233/54 → (51) C07C 233/08<br />
(51) C07C 245/20 (11) 2 421 822 A1*<br />
C07C 37/14 C07C 39/15<br />
C07C 39/19<br />
(25) De (26) De<br />
(21) 10714884.3 (22) 22.04.2010<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MK MT<br />
NL NO PL PT RO SE SI SK SM TR<br />
(86) EP 2010/055347 22.04.2010<br />
(87) WO 2010/122105 2010/43 28.10.2010<br />
(30) 22.04.20<strong>09</strong> EP <strong>09</strong>158489<br />
(54) VERFAHREN ZUR HERSTELLUNG EINES<br />
KREUZKUPPLUNGSPRODUKTES EINES<br />
BENZOLISCHEN DIAZONIUMSALZES<br />
METHOD FOR PRODUCING A CROSS-<br />
COUPLING PRODUCT OF A BENZENOID<br />
DIAZONIUM SALT<br />
PROCÉDÉ DE FABRICATION D'UN<br />
PRODUIT DE COUPLAGE CROISÉ D'UN<br />
SEL BENZÉNIQUE DE DIAZONIUM<br />
(71) Zylum Beteiligungsgesellschaft mbH & Co.<br />
<strong>Patent</strong>e II KG, Berliner Strasse 1, 12529<br />
Schönfeld/OT Waltersdorf, DE<br />
(72) BOEGE, Nicolas, 20149 Hamburg, DE<br />
KREIPL, Andreas, 20359 Hamburg, DE<br />
SCHMIDT, Bernd, 14482 Potsdam, DE<br />
HOELTER, Frank, 14473 Potsdam, DE<br />
BERGER, René, 14471 Potsdam, DE<br />
(74) Held, Stephan, Meissner, Bolte & Partner<br />
GbR Widenmayerstraße 48, D-80538 München,<br />
DE<br />
C07C 255/42 → (51) C07C 233/08<br />
C07C 255/58 → (51) C07C 233/08<br />
C07C 257/12 → (51) C07D 211/46<br />
C07C 263/10 → (51) C07C 2<strong>09</strong>/78<br />
C07C 265/14 → (51) C07C 2<strong>09</strong>/78<br />
C07C 3<strong>09</strong>/08 → (51) A01N 41/04<br />
C07C 3<strong>09</strong>/66 → (51) C07C 2<strong>09</strong>/74<br />
C07C 311/29 → (51) C07D 211/96<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
(51) C07D 205/04 (11) 2 421 823 A1*<br />
C07D 401/10 C07D 401/12<br />
C07D 403/12 C07D 403/14<br />
C07D 405/12 C07D 4<strong>09</strong>/14<br />
A61K 31/496 A61P 25/00<br />
C07D 417/12 A61P 29/00<br />
C07D 417/14 C07D 491/048<br />
(25) En (26) En<br />
(21) 10715457.7 (22) 22.04.2010<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MK MT<br />
NL NO PL PT RO SE SI SK SM TR<br />
AL BA ME RS<br />
(86) US 2010/032049 22.04.2010<br />
(87) WO 2010/124086 2010/43 28.10.2010<br />
(30) 22.04.20<strong>09</strong> US 171649 P<br />
22.04.20<strong>09</strong> US 171658 P<br />
(54) AZETIDINYLDIAMIDE ALS MONOACYL-<br />
GLYCERINLIPASEINHIBITOREN<br />
AZETIDINYL DIAMIDES AS MONOACYL-<br />
GLYCEROL LIPASE INHIBITORS<br />
AZÉTIDINYL DIAMIDES SERVANT D'IN-<br />
HIBITEURS DE LA MONOACYLGLYCÉROL<br />
LIPASE<br />
(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />
30, 2340 Beerse, BE<br />
(72) BIAN, Haiyan, Princeton NJ 08540, US<br />
CHEVALIER, Kristen, M., Collegeville PA<br />
19426, US<br />
CONNOLLY, Peter, J., Spring House PA<br />
19477, US<br />
FLORES, Christopher, M., Spring House PA<br />
19477, US<br />
LIN, Shu-chen, Doylestown PA 18902, US<br />
LIU, Li, Doylestown PA 18901, US<br />
MABUS, John, East Greenville PA 18041, US<br />
MACIELAG, Mark, J., Spring House PA<br />
19477, US<br />
MCDONNELL, Mark, E., Lansdale PA 19446,<br />
US<br />
PITIS, Philip, M., North Wales PA 19454, US<br />
ZHANG, Sui-Po, Exton PA 19341, US<br />
ZHANG, Yue-mei, Spring House PA 19477,<br />
US<br />
ZHU, Bin, Spring House PA 19477, US<br />
CLEMENTE, Jose, Exton PA 19341, US<br />
(74) Warner, James Alexander, Carpmaels &<br />
Ransford One Southampton Row, GB-<br />
London WC1B 5HA, GB<br />
(51) C07D 205/04 (11) 2 421 824 A1*<br />
C07D 401/04 C07D 401/06<br />
C07D 401/10 C07D 403/06<br />
C07D 403/10 C07D 403/12<br />
C07D 405/12 C07D 4<strong>09</strong>/06<br />
C07D 417/06 C07D 417/14<br />
A61K 31/496 A61P 25/00<br />
A61P 29/00<br />
(25) En (26) En<br />
(21) 10715460.1 (22) 22.04.2010<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MK MT<br />
NL NO PL PT RO SE SI SK SM TR<br />
AL BA ME RS<br />
(86) US 2010/032089 22.04.2010<br />
(87) WO 2010/124114 2010/43 28.10.2010<br />
(30) 22.04.20<strong>09</strong> US 171658 P<br />
22.04.20<strong>09</strong> US 171649 P<br />
(54) AZETIDINYLDIAMIDE ALS MONOACYL-<br />
GLYCERINLIPASEINHIBITOREN<br />
AZETIDINYL DIAMIDES AS MONOACYL-<br />
GLYCEROL LIPASE INHIBITORS<br />
DIAMIDES D'AZÉTIDINYLE UTILISÉES<br />
COMME INHIBITEUR DE LA MONOACYL-<br />
GLYCÉROL LIPASE<br />
(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />
30, 2340 Beerse, BE<br />
80<br />
Anmeldungen<br />
Applications<br />
Demandes (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />
(72) BIAN, Haiyan, Princeton NJ 08540, US<br />
CHEVALIER, Kristen, M., Collegeville PA<br />
19426, US<br />
CONNOLLY, Peter, J., Spring House PA<br />
19477, US<br />
FLORES, Christopher, M., Spring House PA<br />
19477, US<br />
LIN, Shu-chen, Doylestown PA 18902, US<br />
LIU, Li, Doylestown PA 18901, US<br />
MABUS, John, East Greenville PA 18041, US<br />
MACIELAG, Mark, J., Spring House PA<br />
19477, US<br />
MCDONNELL, Mark, E., Lansdale PA 19446,<br />
US<br />
PITIS, Philip, M., North Wales PA 19454, US<br />
ZHANG, Yue-mei, Spring House PA 19477,<br />
US<br />
ZHANG, Sui-po, Exton PA 19341, US<br />
CLEMENTE, Jose, Exton PA 19341, US<br />
ZHU, Bin, Spring House PA 19477, US<br />
(74) Warner, James Alexander, et al, Carpmaels &<br />
Ransford One Southampton Row, London<br />
WC1B 5HA, GB<br />
(51) C07D 205/04 (11) 2 421 825 A1*<br />
C07D 401/14 C07D 403/12<br />
C07D 405/12 C07D 405/14<br />
C07D 4<strong>09</strong>/12 C07D 4<strong>09</strong>/14<br />
C07D 413/12 C07D 413/14<br />
C07D 417/12 C07D 417/14<br />
C07D 495/04 A61K 31/496<br />
A61P 29/00 A61P 25/00<br />
(25) En (26) En<br />
(21) 10716205.9 (22) 22.04.2010<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MK MT<br />
NL NO PL PT RO SE SI SK SM TR<br />
AL BA ME RS<br />
(86) US 2010/032082 22.04.2010<br />
(87) WO 2010/124108 2010/43 28.10.2010<br />
(30) 22.04.20<strong>09</strong> US 171649 P<br />
22.04.20<strong>09</strong> US 171658 P<br />
(54) AZETIDINYLDIAMIDE ALS MONOACYL-<br />
GLYCERINLIPASEINHIBITOREN<br />
AZETIDINYL DIAMIDES AS MONOACYL-<br />
GLYCEROL LIPASE INHIBITORS<br />
AZÉTIDINYL DIAMIDES EN TANT QU'IN-<br />
HIBITEURS DE LA MONOACYLGLYCÉROL<br />
LIPASE<br />
(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />
30, 2340 Beerse, BE<br />
(72) BIAN, Haiyan, Princeton NJ 08540, US<br />
CHEVALIER, Kristen, M., Collegeville PA<br />
19426, US<br />
CONNOLLY, Peter, J., Spring House PA<br />
19477, US<br />
FLORES, Christopher, M., Spring House PA<br />
19477, US<br />
LIN, Shu-chen, Doylestown PA 18902, US<br />
LIU, Li, Doylestown PA 18901, US<br />
MABUS, John, East Greenville PA 18041, US<br />
MACIELAG, Mark, J., Spring House PA<br />
19477, US<br />
MCDONNELL, Mark, E., Lansdale PA 19446,<br />
US<br />
PITIS, Philip, M., North Wales PA 19454, US<br />
ZHANG, Sui-po, Exton PA 19341, US<br />
ZHANG, Yue-mei, Spring House PA 19477,<br />
US<br />
ZHU, Bin, Spring House PA 19477, US<br />
CLEMENTE, Jose, Exton PA 19341, US<br />
(74) Warner, James Alexander, Carpmaels &<br />
Ransford One Southampton Row, London<br />
WC1B 5HA, GB<br />
C07D 205/04 → (51) C07D 401/06