European Patent Bulletin 2012/09 - European Patent Office
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European Patent Bulletin 2012/09 - European Patent Office

European Patent Bulletin 2012/09 - European Patent Office European Patent Bulletin 2012/09 - European Patent Office

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(C07C) II.1(1) SULFONIC ACIDS, THEIR DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ACIDES SULFONIQUES, LEURS DERIVES AINSI QUE COMPOSITIONS PHARMA- CEUTIQUES LES CONTENANTS (73) Dompé S.P.A., Via Campo di Pile, I-67100 L'Aquila, IT (72) ALLEGRETTI, Marcello, I-67100 L'Aquila, IT ARAMINI, Andrea, I-67100 L'Aquila, IT CESTA, Maria Candida, I-67100 L'Aquila, IT BERTINI, Riccardo, I-67100 L'Aquila, IT BIZZARRI, Cinzia, I-67100 L'Aquila, IT COLOTTA, Francesco, I-67100 L'Aquila, IT (74) Bonvicini, Davide, et al, Perani & Partners Piazza San Babila, 5, 20122 Milano, IT C07C 309/29 → (51) C07C 309/24 C07C 311/16 → (51) C07C 309/24 C07C 311/21 → (51) C07C 309/24 (51) C07C 319/04 (11) 2 205 557 B1 C07C 323/56 C07C 323/54 C07C 323/61 C07B 45/06 (25) En (26) En (21) 08831702.9 (22) 19.09.2008 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR (43) 14.07.2010 (86) JP 2008/067580 19.09.2008 (87) WO 2009/038232 2009/13 26.03.2009 (30) 20.09.2007 JP 2007243279 (54) VERFAHREN ZUR HERSTELLUNG VON BETA-MERCAPTOCARBONSÄUREN METHOD FOR PRODUCING BETA- MERCAPTOCARBOXYLIC ACIDS PROCEDE DE PRODUCTION D'ACIDES BETA-MERCAPTOCARBOXYLIQUES (73) Showa Denko K.K., 13-9, Shiba Daimon 1chome Minato-ku, Tokyo 105-8518, JP (72) SHIBUYA, Akira, Kawasaki-shi Kanagawa 210-0865, JP AOKI, Hidemasa, Kawasaki-shi Kanagawa 210-0865, JP (74) Strehl Schübel-Hopf & Partner, Maximilianstrasse 54, 80538 München, DE (51) C07C 323/47 (11) 2 327 689 B1 C07C 323/65 C07C 391/02 C07F 9/50 C07C 251/66 C07C 251/68 C08F 2/50 (25) En (26) En (21) 10015054.9 (22) 26.11.2010 (84) AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR (43) 01.06.2011 (30) 27.11.2009 JP 2009269801 04.10.2010 JP 2010225063 (54) Oximesterverbindung und Photopolymerisationsinitiator, der diese Verbindung enthält Oxime ester compound and photopolymerization initiator containing the same Composé ester d'oxime et initiateur de photo-polymérisation le contenant (73) Adeka Corporation, 2-35, Higashiogu 7chome Arakawa-ku, Tokyo 116-8554, JP (72) Murata, Kiyoshi, Tokyo 116-8554, JP Oishi, Takeo, Tokyo 116-8554, JP Kimijima, Koichi, Tokyo 116-8554, JP (74) Forstmeyer, Dietmar, et al, BOETERS & LIECK Oberanger 32, 80331 München, DE C07C 323/54 → (51) C07C 319/04 Europäisches Patentblatt European Patent Bulletin Bulletin européen des brevets C07C 323/56 → (51) C07C 319/04 C07C 323/61 → (51) C07C 319/04 C07C 323/65 → (51) C07C 323/47 C07C 391/02 → (51) C07C 323/47 (51) C07D 205/04 (11) 1 667 966 B1 (25) En (26) En (21) 04781964.4 (22) 20.08.2004 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR AL HR LT LV MK (43) 14.06.2006 (86) US 2004/027379 20.08.2004 (87) WO 2005/021499 2005/10 10.03.2005 (30) 21.08.2003 US 496775 P (54) N-ALKYLIERTE DIAMINOPROPANDERI- VATE ALS MODULATOREN DER CHEMO- KINREZEPTORAKTIVITÄT N-ALKYLATED DIAMINOPROPANE DERI- VATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY DERIVES DE DIAMINOPROPANE N- ALKYLES EN TANT QUE MODULATEURS DE L'ACTIVITE DU RECEPTEUR DE LA CHIMIOKINE (73) Bristol-Myers Squibb Company, Route 206 and Province Line Road, Princeton, NJ 08543-4000, US (72) CARTER, Percy, H., Princeton, NJ 08540, US (74) Beacham, Annabel Rose, et al, Dehns St Bride's House 10 Salisbury Square, London EC4Y 8JD, GB C07D 207/263 → (51) C07C 309/24 (51) C07D 207/277 (11) 2 022 781 B1 C08F 26/00 C08G 63/66 C09K 8/00 (25) De (26) De (21) 08013824.1 (22) 01.08.2008 (84) DE ES FR GB IT NL NO (43) 11.02.2009 (30) 06.08.2007 DE 102007037017 (54) 1-Alkyl-5-oxo-pyrrolidin-3-carbonsäureester mit verbesserter biologischer Abbaubarkeit 1-Alkyl-5-oxo-pyrrolidine-3-carboxylic acid esters with improved biodegradability Esters d'acide 1-alkyl-5-oxo-pyrrolidine-3carboxylique ayant une biodégrabilité améliorée (73) Clariant Finance (BVI) Limited, Citco Building Wickhams Cay P.O. Box 662, Road Town, Tortola, VG (72) Leinweber, Dirk, 65779 Kelkheim, DE Rösch, Alexander, 67578 Gimbsheim, DE Feustel, Michael, 55278 Köngerheim, DE (74) Mikulecky, Klaus, et al, Clariant Produkte (Deutschland) GmbH Group Intellectual Property Am Unisys-Park 1, 65843 Sulzbach, DE (60) 11008153.6 C07D 207/333 → (51) C07C 309/24 (51) C07D 209/40 (11) 2 328 866 B1 A61K 31/404 A61P 35/00 A61P 25/00 (25) En (26) En (21) 09802595.0 (22) 21.07.2009 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (43) 08.06.2011 (86) IB 2009/053153 21.07.2009 656 Patente Patents Brevets (09/2012) 29.02.2012 (87) WO 2010/013168 2010/05 04.02.2010 (30) 01.08.2008 EP 08161646 01.08.2008 US 85432 P (54) 3',6-SUBSTITUIERTE INDIRUBINE UND IHRE BIOLOGISCHE ANWENDUNG 3',6-SUBSTITUTED INDIRUBINS AND THEIR BIOLOGICAL APPLICATIONS INDIRUBINES SUBSTITUÉES EN 3',6 ET LEURS APPLICATIONS BIOLOGIQUES (73) Centre National de la Recherche Scientifique (CNRS), 3, rue Michel-Ange, 75794 Paris Cedex 16, FR (72) MEIJER, Laurent, F-29680 Roscoff, FR SKALTSOUNIS, Leandros, 11253 Athens, GR MIKROS, Emmanuel, 15341 Ag. Paraskevi, GR MAGIATIS, Prokopios, 18902 Ambelakia, GR JOHNSON, Carl, Nashville, Tennessee 37235-1634, US (74) Peaucelle, Chantal, et al, Cabinet Armengaud Aîné 3, Avenue Bugeaud, 75116 Paris, FR (51) C07D 209/42 (11) 2 323 980 B1 C07D 401/12 C07D 403/12 C07D 405/12 C07D 405/14 A61K 31/404 A61P 11/00 (25) De (26) De (21) 09782239.9 (22) 26.08.2009 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (43) 25.05.2011 (86) EP 2009/061025 26.08.2009 (87) WO 2010/026096 2010/10 11.03.2010 (30) 02.09.2008 EP 08163526 (54) 7-(PIPERAZIN-1-YLMETHYL)-1H-INDOL- 2-CARBONSÄURE (PHENYL) -AMIDDERI- VATE UND VERWANDTE VERBINDUNGEN ALS P38 MAP-KINASE-INHIBITOREN ZUR BEHANDLUNG VON ATEMWEGSERKRAN- KUNGEN 7-(PIPERAZINE-1-YMETHYL)-1H- INDOLE-2-CARBOXYLIC ACID (PHENYL)- AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHI- BITORS FOR THE TREATMENT OF RESPIRATORY DISEASES DÉRIVÉS 7-(PIPÉRAZIN-1-YLMÉTHYL)- 1H-INDOL-2-ACIDE CARBOXYLIQUE (PHÉNYL) -AMIDES ET COMPOSÉS ANALOGUES UTILISÉS COMME INHIBI- TEURS DE LA P38 MAP-KINASE POUR LE TRAITEMENT DES MALADIES DES VOIES RESPIRATOIRES (73) Boehringer Ingelheim International GmbH, Binger Strasse 173, 55216 Ingelheim am Rhein, DE (72) WAGNER, Holger, 55216 Ingelheim am Rhein, DE JUNG, Birgit, 55216 Ingelheim am Rhein, DE HIMMELSBACH, Frank, 55216 Ingelheim am Rhein, DE GOEGGEL, Rolf, 55216 Ingelheim am Rhein, DE DAHMANN, Georg, 55216 Ingelheim am Rhein, DE (74) Hammann, Heinz, et al, Boehringer Ingelheim Pharma GmbH & Co. KG CD Patents Binger Strasse 173, 55216 Ingelheim Am Rhein, DE (51) C07D 209/88 (11) 2 323 982 B1 A61K 31/403 (25) En (26) En (21) 09789145.1 (22) 14.08.2009 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR (43) 25.05.2011

(C07D) II.1(1) (86) US 2009/004681 14.08.2009 (87) WO 2010/019271 2010/07 18.02.2010 (30) 15.08.2008 US 189059 P (54) FLUORESZENTE REGULATOREN DER RASSF1A-EXPRESSION UND DER PRO- LIFERATION HUMANER KREBSZELLEN FLUORESCENT REGULATORS OF RASSF1A EXPRESSION AND HUMAN CANCER CELL PROLIFERATION RÉGULATEURS FLUORESCENTS DE L'EXPRESSION DE RASSF1A ET DE LA PROLIFÉRATION DE CELLULES CANCÉ- REUSES HUMAINES (73) Georgetown University, Harris Building Suite 1500 3300 Whitehaven Street, Washington, DC 20007, US (72) BROWN, Milton, L., Brookeville MD 20833, US SHEIKH, Kathryn, D., Washington DC 20007, US PAIGE, Mikell, Fairfax VA 22030, US BANERJEE, Partha, Rockville MD 20852, US JAGADEESH, Shankar, Gaithersburg MD 20879, US (74) Bassett, Richard Simon, Potter Clarkson LLP Park View House 58 The Ropewalk, Nottingham NG1 5DD, GB (60) 12152000.1 (51) C07D 211/58 (11) 1 669 350 B1 C07D 401/06 C07D 401/14 C07D 401/02 C07D 401/12 C07D 409/12 A61K 31/4545 A61K 31/496 A61K 31/454 A61K 31/4523 A61K 31/4535 A61K 31/506 A61P 43/00 A61P 3/04 A61P 3/10 A61P 5/00 A61P 3/06 A61P 19/06 A61P 9/10 A61P 9/04 A61P 9/12 (25) Ja (26) En (21) 04787951.5 (22) 21.09.2004 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR LT LV (43) 14.06.2006 (86) JP 2004/013768 21.09.2004 (87) WO 2005/028438 2005/13 31.03.2005 (30) 22.09.2003 JP 2003330758 (54) PIPERIDINDERIVATE PIPERIDINE DERIVATIVES DERIVES DE PIPERIDINE (73) MSD K.K., Kitanomaru Square 1-13-12 Kudankita, Chiyoda-ku Tokyo 102-8667, JP (72) OHTAKE, N. Tsukuba Res. Inst. Banyu Pharmaceutical, Ibaraki 300-2611, JP MIZUTANI, Sayaka, c/o Tsukuba Research Institute, Tsukuba-shi Ibaraki 3002611, JP YOSHIMOTO, Ryo, c/o Tsukuba Research Institute, Tsukuba-shi, Ibaraki 3002611, JP TOKITA, Shigeru, c/o Tsukuba Research Institute, Tsukuba-shi, Ibaraki 3002611, JP KANATANI, Akio, c/o Tsukuba Research Institute, Tsukuba-shi, Ibaraki 3002611, JP (74) Rollins, Anthony John, et al, Merck Sharp & Dohme Limited European Patent Department Hertford Road, Hoddesdon Hertfordshire EN11 9BU, GB C07D 211/94 → (51) C08K 5/00 C07D 213/61 → (51) C07C 211/48 (51) C07D 213/64 (11) 1 772 450 B1 (25) Ja (26) En (21) 05758231.4 (22) 05.07.2005 Europäisches Patentblatt European Patent Bulletin Bulletin européen des brevets (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR AL BA HR MK YU (43) 11.04.2007 (86) JP 2005/012364 05.07.2005 (87) WO 2006/004100 2006/02 12.01.2006 (30) 06.07.2004 JP 2004198709 (54) VERFAHREN ZUR HERSTELLUNG EINER 1,2-DIHYDROPYRIDIN-2-ONVERBIN- DUNG METHOD FOR PRODUCING 1,2-DIHY- DROPYRIDINE-2-ONE COMPOUND PROCÉDÉ POUR LA FABRICATION D"UN COMPOSÉ DE 1,2-DIHYDROPYRIDINE-2- ONE (73) Eisai R&D Management Co., Ltd., 6-10, Koishikawa 4-chome, Bunkyo-ku, Tokyo 112-8088, JP (72) KAYANO, Akio, Kamisu-shi, Ibaraki, JP NISHIURA, Katsutoshi, Kamisu-shi, Ibaraki, JP (74) HOFFMANN EITLE, Patent- und Rechtsanwälte Arabellastraße 4, 81925 München, DE (51) C07D 213/75 (11) 1 203 766 B1 C07D 215/22 C07D 221/04 C07D 221/16 C07D 401/04 C07D 401/12 C07D 403/12 C07D 405/12 C07D 409/06 C07D 409/12 C07D 409/14 C07D 413/06 C07D 413/12 C07D 417/06 C07D 471/04 A61K 31/505 A61K 31/44 A61K 31/50 A61K 31/4704 A61P 29/00 A61P 35/00 (25) En (26) En (21) 01125494.3 (22) 06.11.2001 (84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR (43) 08.05.2002 (30) 06.11.2000 US 707068 09.10.2001 US 973142 (54) Carbonsäurederivate, die die Bindung von Integrinen an ihre Rezeptoren hemmen Carboxylic acid derivatives that inhibit the binding of integrins to their receptors Dérivés d'acides carboxyliques inhibant la liaison des intégrines à leurs récepteurs (73) ENCYSIVE PHARMACEUTICALS, INC., 4848 Loop Central Drive, Suite 700, Houston, TX 77081, US (72) Biediger, Ronald J., Houston, TX 77095, US Chen, Qi, Pearland, TX 77584, US Holland, George W., Houston, Texas 77007, US Kassir, Jamal M., Stafford, Texas 77477, US Li, Wen, Houston, TX 77057, US Market, Robert V., Pearland, TX 77581, US Scott, Ian L., Delanson, NY 12053, US Wu, Chengde, Pearland, TX 77584, US Decker, Radford E., Houston, TX 77018, US Li, Jian, Houston, TX 77382, US (74) Weber, Martin, et al, Jones Day Prinzregentenstraße 11, 80538 München, DE C07D 215/22 → (51) C07D 213/75 C07D 221/04 → (51) C07D 213/75 C07D 221/16 → (51) C07D 213/75 (51) C07D 239/38 (11) 2 205 569 B1 C07D 239/47 C07D 239/58 A61K 31/505 A61P 29/00 (25) En (26) En (21) 08833849.6 (22) 24.09.2008 657 Patente Patents Brevets (09/2012) 29.02.2012 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR (43) 14.07.2010 (86) US 2008/011053 24.09.2008 (87) WO 2009/042138 2009/14 02.04.2009 (30) 25.09.2007 US 995386 P (54) ALKYLTHIOPYRIMIDINE ALS CRTH2-AN- TAGONISTEN ALKYLTHIO PYRIMIDINES AS CRTH2 ANTAGONISTS ALKYLTHIOPYRIMIDINES EN TANT QU'ANTAGONISTES DE CRTH2 (73) Actimis Pharmaceuticals, Inc., 10835 Road to the Cure, Suite 200, San Diego, CA 92121, US (72) LY, Tai, Wei, San Diego CA 92121, US RAAUM, Erik, D., San Diego CA 92121, US TRAN, Marie, Chantal S.-Y, San Diego CA 92121, US (74) Ritter, Thomas Kurt, Jones Day Prinzregentenstraße 11, 80538 München, DE C07D 239/47 → (51) C07D 239/38 C07D 239/58 → (51) C07D 239/38 (51) C07D 239/90 (11) 1 953 148 B1 A61K 31/517 A61K 31/519 A61P 19/02 A61P 29/00 A61P 43/00 C07D 401/14 C07D 403/12 C07D 403/14 C07D 487/04 C07D 495/04 (25) Ja (26) En (21) 06822961.6 (22) 27.10.2006 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR AL BA HR MK RS (43) 06.08.2008 (86) JP 2006/322043 27.10.2006 (87) WO 2007/049820 2007/18 03.05.2007 (30) 28.10.2005 JP 2005315267 (54) HETEROCYCLISCHE AMIDVERBINDUNG UND ANWENDUNG DAVON HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF COMPOSE AMIDE HETEROCYCLIQUE ET UTILISATION DE CELUI-CI (73) Takeda Pharmaceutical Company Limited, 1- 1, Doshomachi 4-chome Chuo-ku, Osakashi, Osaka 541-0045, JP (72) NARA, Hiroshi, Osaka-shi, Osaka 532-8686, JP KAIEDA, Akira, Osaka-shi, Osaka 532-8686, JP SATO, Kenjiro, Osaka-shi, Osaka 532-8686, JP TERAUCHI, Jun, Osaka-shi, Osaka 532- 8686, JP (74) Dossmann, Gérard, et al, Casalonga & Partners Bayerstrasse 71-73, 80335 München, DE C07D 241/04 → (51) A61K 31/495 (51) C07D 249/08 (11) 2 212 301 B1 A61K 31/4196 A61P 35/00 (25) En (26) En (21) 08702736.3 (22) 16.01.2008 (84) AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR (43) 04.08.2010 (86) IN 2008/000024 16.01.2008 (87) WO 2009/069140 2009/23 04.06.2009 (30) 28.11.2007 IN DE24792007

(C07D) II.1(1)<br />

(86) US 20<strong>09</strong>/004681 14.08.20<strong>09</strong><br />

(87) WO 2010/019271 2010/07 18.02.2010<br />

(30) 15.08.2008 US 189059 P<br />

(54) FLUORESZENTE REGULATOREN DER<br />

RASSF1A-EXPRESSION UND DER PRO-<br />

LIFERATION HUMANER KREBSZELLEN<br />

FLUORESCENT REGULATORS OF<br />

RASSF1A EXPRESSION AND HUMAN<br />

CANCER CELL PROLIFERATION<br />

RÉGULATEURS FLUORESCENTS DE<br />

L'EXPRESSION DE RASSF1A ET DE LA<br />

PROLIFÉRATION DE CELLULES CANCÉ-<br />

REUSES HUMAINES<br />

(73) Georgetown University, Harris Building Suite<br />

1500 3300 Whitehaven Street, Washington,<br />

DC 20007, US<br />

(72) BROWN, Milton, L., Brookeville MD 20833,<br />

US<br />

SHEIKH, Kathryn, D., Washington DC 20007,<br />

US<br />

PAIGE, Mikell, Fairfax VA 22030, US<br />

BANERJEE, Partha, Rockville MD 20852, US<br />

JAGADEESH, Shankar, Gaithersburg MD<br />

20879, US<br />

(74) Bassett, Richard Simon, Potter Clarkson LLP<br />

Park View House 58 The Ropewalk,<br />

Nottingham NG1 5DD, GB<br />

(60) 12152000.1<br />

(51) C07D 211/58 (11) 1 669 350 B1<br />

C07D 401/06 C07D 401/14<br />

C07D 401/02 C07D 401/12<br />

C07D 4<strong>09</strong>/12 A61K 31/4545<br />

A61K 31/496 A61K 31/454<br />

A61K 31/4523 A61K 31/4535<br />

A61K 31/506 A61P 43/00<br />

A61P 3/04 A61P 3/10<br />

A61P 5/00 A61P 3/06<br />

A61P 19/06 A61P 9/10<br />

A61P 9/04 A61P 9/12<br />

(25) Ja (26) En<br />

(21) 04787951.5 (22) 21.<strong>09</strong>.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI<br />

SK TR<br />

LT LV<br />

(43) 14.06.2006<br />

(86) JP 2004/013768 21.<strong>09</strong>.2004<br />

(87) WO 2005/028438 2005/13 31.03.2005<br />

(30) 22.<strong>09</strong>.2003 JP 2003330758<br />

(54) PIPERIDINDERIVATE<br />

PIPERIDINE DERIVATIVES<br />

DERIVES DE PIPERIDINE<br />

(73) MSD K.K., Kitanomaru Square 1-13-12<br />

Kudankita, Chiyoda-ku Tokyo 102-8667, JP<br />

(72) OHTAKE, N. Tsukuba Res. Inst. Banyu Pharmaceutical,<br />

Ibaraki 300-2611, JP<br />

MIZUTANI, Sayaka, c/o Tsukuba Research<br />

Institute, Tsukuba-shi Ibaraki 3002611, JP<br />

YOSHIMOTO, Ryo, c/o Tsukuba Research<br />

Institute, Tsukuba-shi, Ibaraki 3002611, JP<br />

TOKITA, Shigeru, c/o Tsukuba Research<br />

Institute, Tsukuba-shi, Ibaraki 3002611, JP<br />

KANATANI, Akio, c/o Tsukuba Research<br />

Institute, Tsukuba-shi, Ibaraki 3002611, JP<br />

(74) Rollins, Anthony John, et al, Merck Sharp &<br />

Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 211/94 → (51) C08K 5/00<br />

C07D 213/61 → (51) C07C 211/48<br />

(51) C07D 213/64 (11) 1 772 450 B1<br />

(25) Ja (26) En<br />

(21) 05758231.4 (22) 05.07.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 11.04.2007<br />

(86) JP 2005/012364 05.07.2005<br />

(87) WO 2006/004100 2006/02 12.01.2006<br />

(30) 06.07.2004 JP 20041987<strong>09</strong><br />

(54) VERFAHREN ZUR HERSTELLUNG EINER<br />

1,2-DIHYDROPYRIDIN-2-ONVERBIN-<br />

DUNG<br />

METHOD FOR PRODUCING 1,2-DIHY-<br />

DROPYRIDINE-2-ONE COMPOUND<br />

PROCÉDÉ POUR LA FABRICATION D"UN<br />

COMPOSÉ DE 1,2-DIHYDROPYRIDINE-2-<br />

ONE<br />

(73) Eisai R&D Management Co., Ltd., 6-10,<br />

Koishikawa 4-chome, Bunkyo-ku, Tokyo<br />

112-8088, JP<br />

(72) KAYANO, Akio, Kamisu-shi, Ibaraki, JP<br />

NISHIURA, Katsutoshi, Kamisu-shi, Ibaraki,<br />

JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München,<br />

DE<br />

(51) C07D 213/75 (11) 1 203 766 B1<br />

C07D 215/22 C07D 221/04<br />

C07D 221/16 C07D 401/04<br />

C07D 401/12 C07D 403/12<br />

C07D 405/12 C07D 4<strong>09</strong>/06<br />

C07D 4<strong>09</strong>/12 C07D 4<strong>09</strong>/14<br />

C07D 413/06 C07D 413/12<br />

C07D 417/06 C07D 471/04<br />

A61K 31/505 A61K 31/44<br />

A61K 31/50 A61K 31/4704<br />

A61P 29/00 A61P 35/00<br />

(25) En (26) En<br />

(21) 01125494.3 (22) 06.11.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 08.05.2002<br />

(30) 06.11.2000 US 707068<br />

<strong>09</strong>.10.2001 US 973142<br />

(54) Carbonsäurederivate, die die Bindung von<br />

Integrinen an ihre Rezeptoren hemmen<br />

Carboxylic acid derivatives that inhibit the<br />

binding of integrins to their receptors<br />

Dérivés d'acides carboxyliques inhibant la<br />

liaison des intégrines à leurs récepteurs<br />

(73) ENCYSIVE PHARMACEUTICALS, INC., 4848<br />

Loop Central Drive, Suite 700, Houston, TX<br />

77081, US<br />

(72) Biediger, Ronald J., Houston, TX 77<strong>09</strong>5, US<br />

Chen, Qi, Pearland, TX 77584, US<br />

Holland, George W., Houston, Texas 77007,<br />

US<br />

Kassir, Jamal M., Stafford, Texas 77477, US<br />

Li, Wen, Houston, TX 77057, US<br />

Market, Robert V., Pearland, TX 77581, US<br />

Scott, Ian L., Delanson, NY 12053, US<br />

Wu, Chengde, Pearland, TX 77584, US<br />

Decker, Radford E., Houston, TX 77018, US<br />

Li, Jian, Houston, TX 77382, US<br />

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(51) C07D 239/38 (11) 2 205 569 B1<br />

C07D 239/47 C07D 239/58<br />

A61K 31/505 A61P 29/00<br />

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(43) 14.07.2010<br />

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(87) WO 20<strong>09</strong>/042138 20<strong>09</strong>/14 02.04.20<strong>09</strong><br />

(30) 25.<strong>09</strong>.2007 US 995386 P<br />

(54) ALKYLTHIOPYRIMIDINE ALS CRTH2-AN-<br />

TAGONISTEN<br />

ALKYLTHIO PYRIMIDINES AS CRTH2<br />

ANTAGONISTS<br />

ALKYLTHIOPYRIMIDINES EN TANT<br />

QU'ANTAGONISTES DE CRTH2<br />

(73) Actimis Pharmaceuticals, Inc., 10835 Road<br />

to the Cure, Suite 200, San Diego, CA<br />

92121, US<br />

(72) LY, Tai, Wei, San Diego CA 92121, US<br />

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(51) C07D 239/90 (11) 1 953 148 B1<br />

A61K 31/517 A61K 31/519<br />

A61P 19/02 A61P 29/00<br />

A61P 43/00 C07D 401/14<br />

C07D 403/12 C07D 403/14<br />

C07D 487/04 C07D 495/04<br />

(25) Ja (26) En<br />

(21) 06822961.6 (22) 27.10.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

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(43) 06.08.2008<br />

(86) JP 2006/322043 27.10.2006<br />

(87) WO 2007/049820 2007/18 03.05.2007<br />

(30) 28.10.2005 JP 2005315267<br />

(54) HETEROCYCLISCHE AMIDVERBINDUNG<br />

UND ANWENDUNG DAVON<br />

HETEROCYCLIC AMIDE COMPOUND AND<br />

USE THEREOF<br />

COMPOSE AMIDE HETEROCYCLIQUE ET<br />

UTILISATION DE CELUI-CI<br />

(73) Takeda Pharmaceutical Company Limited, 1-<br />

1, Doshomachi 4-chome Chuo-ku, Osakashi,<br />

Osaka 541-0045, JP<br />

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JP<br />

KAIEDA, Akira, Osaka-shi, Osaka 532-8686,<br />

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8686, JP<br />

(74) Dossmann, Gérard, et al, Casalonga & Partners<br />

Bayerstrasse 71-73, 80335 München,<br />

DE<br />

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A61K 31/4196 A61P 35/00<br />

(25) En (26) En<br />

(21) 08702736.3 (22) 16.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 04.08.2010<br />

(86) IN 2008/000024 16.01.2008<br />

(87) WO 20<strong>09</strong>/069140 20<strong>09</strong>/23 04.06.20<strong>09</strong><br />

(30) 28.11.2007 IN DE24792007

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