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European Patent Bulletin 2012/09 - European Patent Office

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(C07C) II.1(1)<br />

(60) 11179217.2 / 2 392 556<br />

11179239.6 / 2 392 557<br />

(51) C07C 41/03 (11) 2 059 495 B1<br />

C07C 43/11 C07C 67/26<br />

C07C 213/04 C07D 301/10<br />

C08G 65/26<br />

(25) De (26) De<br />

(21) 07801953.6 (22) 29.08.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL<br />

PT RO SE SI SK TR<br />

(43) 20.05.20<strong>09</strong><br />

(86) EP 2007/007531 29.08.2007<br />

(87) WO 2008/028587 2008/11 13.03.2008<br />

(30) 07.<strong>09</strong>.2006 DE 102006041903<br />

(54) VERFAHREN ZUR HERSTELLUNG VON<br />

ALKYLENOXIDANLAGERUNGSPRODUK-<br />

TEN<br />

METHOD FOR PRODUCING ALKYLENE<br />

OXIDE ADDITION PRODUCTS<br />

PROCÉDÉ DE PRÉPARATION DES<br />

PRODUITS D'ADDITION D'OXYDES D'AL-<br />

KYLÈNE<br />

(73) Cognis IP Management GmbH, Henkelstrasse<br />

67, 40589 Düsseldorf, DE<br />

(72) FRANZEN, Stefan, 59174 Kamen, DE<br />

GUTSCHE, Bernhard, 40724 Hilden, DE<br />

FABRY, Bernd, 41352 Korschenbroich, DE<br />

MAHNKE, Eike, Ulf, 42553 Velbert, DE<br />

(74) Reinhardt, Jürgen, Cognis IP Management<br />

GmbH Henkelstrasse 67, 40589 Düsseldorf,<br />

DE<br />

C07C 43/11 → (51) C07C 41/03<br />

(51) C07C 67/08 (11) 2 321 251 B1<br />

C07C 67/54 C07C 69/68<br />

(25) Fr (26) Fr<br />

(21) <strong>09</strong>780717.6 (22) 16.07.20<strong>09</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(43) 18.05.2011<br />

(86) EP 20<strong>09</strong>/059162 16.07.20<strong>09</strong><br />

(87) WO 2010/012606 2010/05 04.02.2010<br />

(30) 30.07.2008 BE 200800424<br />

(54) KONTINUIERLICHES VERFAHREN ZUR<br />

GEWINNUNG EINES MILCHSÄUREES-<br />

TERS<br />

CONTINUOUS PROCESS FOR OBTAINING<br />

A LACTIC ESTER<br />

PROCÉDÉ CONTINU D'OBTENTION D'UN<br />

ESTER LACTIQUE<br />

(73) Galactic S.A., Place d'Escanaffles 23, 7760<br />

Escanaffles, BE<br />

(72) HOTTOIS, Delphine, B-7760 Escanaffles, BE<br />

BRUNEAU, Alexandre, B-7760 Escanaffles,<br />

BE<br />

BOGAERT, Jean-Christophe, B-7760 Escanaffles,<br />

BE<br />

COSZACH, Philippe, B-7760 Escanaffles, BE<br />

(74) Vandeberg, Marie-Paule L.G., et al, <strong>Office</strong><br />

Kirkpatrick S.A. Avenue Wolfers 32, 1310 La<br />

Hulpe, BE<br />

C07C 67/14 → (51) A61K 8/37<br />

C07C 67/26 → (51) C07C 41/03<br />

C07C 67/36 → (51) C07B 59/00<br />

C07C 67/54 → (51) C07C 67/08<br />

C07C 69/68 → (51) C07C 67/08<br />

C07C 69/734 → (51) A61K 8/37<br />

C07C 211/44 → (51) A61K 8/41<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(51) C07C 211/48 (11) 2 <strong>09</strong>4 643 B1<br />

C07C 215/20 C07C 233/18<br />

C07C 275/08 C07C 275/18<br />

C07C 275/26 C07D 213/61<br />

C07D 307/32 C07D 3<strong>09</strong>/14<br />

A61K 31/44 A61K 31/165<br />

A61K 31/17 A61K 31/137<br />

A61P 3/06 A61P 3/04<br />

(25) En (26) En<br />

(21) 07864837.5 (22) 28.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL<br />

PT RO SE SI SK TR<br />

HR<br />

(43) 02.<strong>09</strong>.20<strong>09</strong><br />

(86) US 2007/085733 28.11.2007<br />

(87) WO 2008/070496 2008/24 12.06.2008<br />

(30) 01.12.2006 US 868112 P<br />

(54) N-((3-BENZYL)-2,2-(BIS-PHENYL)-PRO-<br />

PAN-1-AMINDERIVATE ALS CETP-HEM-<br />

MER FÜR DIE BEHANDLUNG VON ATHE-<br />

ROSKLEROSE UND HERZ-KREISLAUF-<br />

ERKRANKUNGEN<br />

N-((3-BENZYL)-2,2-(BIS-PHENYL)-<br />

PROPAN-1-AMINE DERIVATIVES AS<br />

CETP INHIBITORS FOR THE TREATMENT<br />

OF ATHEROSCLEROSIS AND CARDIO-<br />

VASCULAR DISEASES<br />

INHIBITEURS D'AMINO CETP ÉTENDUS<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton, NJ<br />

08543-4000, US<br />

(72) SALVATI, Mark E., Pennington, New Jersey<br />

08534, US<br />

JOHNSON, James A., Pennington, New<br />

Jersey 08534, US<br />

XU, Ningning, Pennington, New Jersey<br />

08534, US<br />

(74) Nevant, Marc, et al, Cabinet Beau de<br />

Loménie 158, rue de l'Université, 75340<br />

Paris Cedex 07, FR<br />

C07C 213/04 → (51) C07C 41/03<br />

C07C 215/20 → (51) C07C 211/48<br />

(51) C07C 217/64 (11) 1 622 860 B1<br />

C07C 217/72 C07D 317/64<br />

C07F 9/<strong>09</strong> C07F 9/6574<br />

A61K 31/661 A61K 31/137<br />

A61P 37/02<br />

(25) En (26) En<br />

(21) 04730206.2 (22) 29.04.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI<br />

SK TR<br />

(43) 08.02.2006<br />

(86) EP 2004/004569 29.04.2004<br />

(87) WO 2004/<strong>09</strong>6752 2004/46 11.11.2004<br />

(30) 30.04.2003 GB 03<strong>09</strong>944<br />

19.12.2003 GB 0329505<br />

19.12.2003 GB 0329500<br />

(54) AMINOPROPANOL-DERIVATE ALS MO-<br />

DULATOREN DES SPHINGOSIN-1-PHOS-<br />

PHAT-REZEPTORS<br />

AMINO-PROPANOL DERIVATIVES AS<br />

SPHINGOSINE-1-PHOSPHATE RECEPTOR<br />

MODULATORs<br />

DERIVES D'AMINO-PROPANOL COMME<br />

MODULATEURS DE RECEPTEUR DE<br />

SPHINGOSINE-1-PHOSPHATE<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(84) BE BG CH CY CZ DE DK EE ES FI FR GB GR<br />

HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

(73) Novartis Pharma GmbH, Brunner Strasse 59,<br />

1230 Wien, AT<br />

(84) AT<br />

(72) HINTERDING, Klaus, 79599 Wittlingen, DE<br />

655<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />

SPANKA, Carsten, 79618 Rheinfelden, DE<br />

ZECRI, Frédéric, F-68510 Uffheim, FR<br />

(74) <strong>Patent</strong>- und Rechtsanwaltssozietät Maucher,<br />

Börjes & Kollegen, et al, Urachstrasse 23,<br />

79102 Freiburg i. Br., DE<br />

C07C 217/72 → (51) C07C 217/64<br />

C07C 233/18 → (51) C07C 211/48<br />

C07C 235/06 → (51) C11C 3/00<br />

C07C 249/08 → (51) C01B 21/14<br />

C07C 251/66 → (51) C07C 323/47<br />

C07C 251/68 → (51) C07C 323/47<br />

C07C 275/08 → (51) C07C 211/48<br />

(51) C07C 275/14 (11) 1 904 438 B1<br />

C07C 275/52 C07C 275/62<br />

A61K 31/33<br />

(25) En (26) En<br />

(21) 06777658.3 (22) 07.07.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

(43) 02.04.2008<br />

(86) EP 2006/064028 07.07.2006<br />

(87) WO 2007/006761 2007/03 18.01.2007<br />

(30) 08.07.2005 EP 05106283<br />

(54) DICYCLOALKYLCARBAMOYL-HARN-<br />

STOFFE ALS GLUCOKINASE-AKTIVA-<br />

TOREN<br />

DICYCLOALKYLCARBAMOYL UREAS AS<br />

GLUCOKINASE ACTIVATORS<br />

DICYCLOALKYLCARBAMOYLURÉES EN<br />

TANT QU' ACTIVATEURS DE GLUCOKI-<br />

NASE<br />

(73) Novo Nordisk A/S, Novo Allé, 2880<br />

Bagsværd, DK<br />

(72) MURRAY, Anthony, DK-2900 Hellerup, DK<br />

LAU, Jesper, DK-3520 Farum, DK<br />

VEDSØ, Per, DK-3500 Værløse, DK<br />

JEPPESEN, Lone, DK-2830 Virum, DK<br />

KRISTIANSEN, Marit, DK-2860 Søborg, DK<br />

(74) Nielsen, Lars Balzer, et al, Novo Nordisk A/S<br />

Corporate <strong>Patent</strong>s Novo Allée, 2880<br />

Bagsvaerd, DK<br />

C07C 275/18 → (51) C07C 211/48<br />

C07C 275/26 → (51) C07C 211/48<br />

C07C 275/52 → (51) C07C 275/14<br />

C07C 275/62 → (51) C07C 275/14<br />

(51) C07C 3<strong>09</strong>/24 (11) 1 606 248 B1<br />

C07C 3<strong>09</strong>/29 C07C 311/16<br />

C07C 311/21 C07D 207/263<br />

C07D 207/333 A61K 31/18<br />

A61K 31/10 A61P 29/00<br />

(25) En (26) En<br />

(21) 04719463.4 (22) 11.03.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI<br />

SK TR<br />

AL LT LV MK<br />

(43) 21.12.2005<br />

(86) EP 2004/050293 11.03.2004<br />

(87) WO 2004/08<strong>09</strong>51 2004/39 23.<strong>09</strong>.2004<br />

(30) 14.03.2003 EP 03005783<br />

(54) SULFONSÄUREN, DEREN DERIVATE SO-<br />

WIE SIE ENTHALTENDEN PHARMAZEU-<br />

TISCHEN ZUBEREITUNGEN

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