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European Patent Bulletin 2012/09 - European Patent Office

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(C07D) I.1(2)<br />

HIGASHIMURA, Hideyuki, Tsukuba-shi<br />

Ibaraki 305-0045, JP<br />

(74) Duckworth, Timothy John, et al, J.A. Kemp<br />

& Co. 14 South Square Gray's Inn, London<br />

WC1R 5JJ, GB<br />

(51) C07D 213/53 (11) 2 423 193 A1<br />

C07D 213/61 C07F 15/02<br />

(25) En (26) En<br />

(21) 11178387.4 (22) 12.01.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 13.01.2006 DE 102006001960<br />

<strong>09</strong>.05.2006 US 798866 P<br />

(54) Verfahren zur Herstellung von Iminoverbindungen<br />

Process for preparing imino compounds<br />

Procédé de préparation de composants<br />

imino<br />

(71) Basell Polyolefine GmbH, Brühler Strasse 60,<br />

50389 Wesseling, DE<br />

(72) Kölling, Lars, 68163 Mannheim, DE<br />

(74) Seelert, Stefan, Basell Polyolefine GmbH Intellectual<br />

Property Industriepark Hoechst,<br />

B852, 3rd floor, 65926 Frankfurt am Main,<br />

DE<br />

(62) 07702728.2 / 1 973 879<br />

C07D 213/55 → (51) C07C 303/30<br />

C07D 213/61 → (51) C07D 213/53<br />

C07D 213/64 → (51) A61K 31/192<br />

(51) C07D 213/65 (11) 2 423 194 A1<br />

A61K 31/44 A61K 31/4418<br />

A61K 31/443 A61K 31/4433<br />

A61K 31/4439 A61P 1/16<br />

A61P 3/04 A61P 3/06<br />

A61P 3/10 A61P 5/14<br />

A61P 9/00 A61P 9/04<br />

A61P 9/10<br />

(25) Ja (26) En<br />

(21) 10767037.4 (22) 19.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/056936 19.04.2010<br />

(87) WO 2010/122980 2010/43 28.10.2010<br />

(30) 20.04.20<strong>09</strong> JP 20<strong>09</strong>102259<br />

(54) NEUER SCHILDDRÜSENHORMON-ß-RE-<br />

ZEPTOR-AGONIST<br />

NOVEL THYROID HORMONE beta<br />

RECEPTOR AGONIST<br />

NOUVEL AGONISTE DU RÉCEPTEUR béta<br />

DE L'HORMONE THYROÏDIENNE<br />

(71) Mitsubishi Tanabe Pharma Corporation, 2-6-<br />

18, Kitahama Chuo-ku 3-chome, Osaka-shi<br />

Osaka 541-8505, JP<br />

(72) KAWATA, Shinji, Osaka-shi Osaka 541-8505,<br />

JP<br />

MATSUMOTO, Koji, Osaka-shi Osaka 541-<br />

8505, JP<br />

NIIJIMA, Maki, Osaka-shi Osaka 541-8505,<br />

JP<br />

TAKAHASHI, Taichi, Osaka-shi Osaka 541-<br />

8505, JP<br />

(74) Wiedemann, Peter, Hoffmann · Eitle <strong>Patent</strong>und<br />

Rechtsanwälte Arabellastraße 4, DE-<br />

81925 München, DE<br />

C07D 213/81 → (51) C07C 271/28<br />

(51) C07D 215/14 (11) 2 423 195 A1<br />

C07D 239/46 C07C 49/233<br />

C07C 49/235<br />

(25) En (26) En<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(21) 10170739.6 (22) 26.07.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

BA ME RS<br />

(54) Verfahren zur Herstellung von wesentlichen<br />

Zwischenstufen zur Synthese von<br />

Rosuvastatin oder pharmazeutisch annehmbaren<br />

Salzen davon<br />

Process for the preparation of key intermediates<br />

for the synthesis of statins or<br />

pharmaceutically acceptable salts thereof<br />

Procédé pour la préparation d'intermédiaires<br />

clé pour la synthèse de statines ou<br />

de ses sels pharmaceutiquement acceptables<br />

(71) LEK Pharmaceuticals d.d., Verovskova 57,<br />

1526 Ljubljana, SI<br />

(72) The designation of the inventor has not yet<br />

been filed<br />

(74) Kunic Tesovic, Barbara, Lek Pharmaceuticals<br />

d.d. Sandoz Development Center Slovenia -<br />

<strong>Patent</strong>s Verovskova 57, 1526 Ljubljana, SI<br />

(51) C07D 217/22 (11) 2 423 196 A1<br />

C07D 401/04 C07D 405/04<br />

C07D 4<strong>09</strong>/04 C07D 491/04<br />

A61K 31/472 A61K 31/4725<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 11190786.1 (22) 16.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL<br />

PT RO SE SI SK TR<br />

(30) 17.11.2006 US 866269 P<br />

(54) 5-, 6- oder 7-substituierte 3-Phenylisochinolinaminderivate<br />

und deren therapeutische<br />

Verwendung<br />

5, 6 or 7-substituted-3-phenylisoquinolinamine<br />

derivatives and therapeutic use<br />

thereof<br />

Dérivés de 3-phénylisoquinolinamine à<br />

substitution 5, 6 ou 7 et leur utilisation<br />

thérapeutique<br />

(71) Rexahn Pharmaceuticals, Inc., 15245 Shady<br />

Grove Road, Suite 455, Rockville, MD<br />

20850, US<br />

(72) Lee, Young Bok, Clarksburg, MD Maryland<br />

20871, US<br />

Ahn, Chang-ho, Potomac, MD Maryland<br />

20854, US<br />

Cho, Won-jea, 500-757 KWANGJU, KR<br />

(74) Fagerlin, Heléne, Albihns.Zacco Valhallavägen<br />

117 Box 5581, 114 85 Stockholm, SE<br />

(62) 07840063.7 / 2 <strong>09</strong>9 765<br />

(51) C07D 231/38 (11) 2 423 197 A1<br />

G03G 9/08 C07F 15/02<br />

(25) En (26) En<br />

(21) 110<strong>09</strong>333.3 (22) 20.11.2003<br />

(84) DE FR GB<br />

(30) 31.03.2003 JP 2003<strong>09</strong>6578<br />

24.07.2003 JP 2003<strong>2012</strong>62<br />

11.08.2003 JP 2003207208<br />

16.10.2003 JP 2003356674<br />

(54) Monoazoeisenkomplexverbindung<br />

A monoazo iron complex compound<br />

Composé complexe de monoazo de fer<br />

(71) Hodogaya Chemical Co., Ltd., 66-2,<br />

Horikawa-cho, Saiwai-ku, Kawasaki-shi,<br />

Kanagawa 212-8588, JP<br />

(72) Otsuka, Hideyuki, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Nemoto, Kazuo, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Otani, Shinji, Sunto-gun Shizuoka 411-<strong>09</strong>33,<br />

JP<br />

Suzuki, Noriyuki, Koriyama-shi Fukushima<br />

963-8802, JP<br />

253<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />

Yamada, Eisuke, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Okubo, Masaki, Koriyama-shi Fukushima<br />

963-8802, JP<br />

(74) Blodig, Wolfgang, Wächtershäuser & Hartz<br />

Weinstrasse 8, 80333 München, DE<br />

(62) 03774<strong>09</strong>1.7 / 1 6<strong>09</strong> 782<br />

(51) C07D 231/38 (11) 2 423 198 A1<br />

G03G 9/08 C07F 15/02<br />

(25) En (26) En<br />

(21) 110<strong>09</strong>334.1 (22) 20.11.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

AL LT LV MK<br />

(30) 31.03.2003 JP 2003<strong>09</strong>6578<br />

24.07.2003 JP 2003<strong>2012</strong>62<br />

11.08.2003 JP 2003207208<br />

16.10.2003 JP 2003356674<br />

(54) Ladungskontrollmittel, das eine Monoazoeisenkomplexverbindung<br />

enthält<br />

Charge controlling agaent containing a<br />

monoazo iron complex compound<br />

Agent de contrôle de charge contenant un<br />

composé complexe de monoazo de fer<br />

(71) Hodogaya Chemical Co., Ltd., 66-2,<br />

Horikawa-cho, Saiwai-ku, Kawasaki-shi,<br />

Kanagawa 212-8588, JP<br />

(72) Otsuka, Hideyuki, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Nemoto, Kazuo, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Otani, Shinji, Sunto-gun Shizuoka 411-<strong>09</strong>33,<br />

JP<br />

Suzuki, Noriyuki, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Yamada, Eisuke, Koriyama-shi Fukushima<br />

963-8802, JP<br />

Okubo, Masaki, Koriyama-shi Fukushima<br />

963-8802, JP<br />

(74) Blodig, Wolfgang, Wächtershäuser & Hartz<br />

Weinstrasse 8, 80333 München, DE<br />

(62) 03774<strong>09</strong>1.7 / 1 6<strong>09</strong> 782<br />

C07D 231/56 → (51) A61K 31/335<br />

C07D 231/56 → (51) C07D 2<strong>09</strong>/14<br />

(51) C07D 233/54 (11) 2 423 199 A1<br />

C07D 401/12 C07D 403/12<br />

C07D 405/12 C07D 417/12<br />

C07D 417/04 A01N 43/50<br />

(25) En (26) En<br />

(21) 11161432.7 (22) 08.01.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 19.01.2006 US 760765 P<br />

(54) Substituierte Imidazole und ihre Verwendung<br />

als Pestizide<br />

Substituted imidazoles and their use as<br />

pesticides<br />

Imidazoles substitués et leur utilisation<br />

comme pesticides<br />

(71) Pfizer Limited, Ramsgate Road, Sandwich,<br />

Kent CT13 9NJ, GB<br />

(72) Chubb, Nathan, Anthony, Logan, Sandwich,<br />

Kent CT13 9NJ, GB<br />

Cox, Mark, Roger, Sandwich, Kent CT13<br />

9NJ, GB<br />

Dauvergne, Jérôme, Sébastien, Sandwich,<br />

Kent CT13 9NJ, GB<br />

Ewin, Richard, Andrew, Sandwich, Kent<br />

CT13 9NJ, GB<br />

Lauret, Christelle, Sandwich, Kent CT13 9NJ,<br />

GB

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