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European Patent Bulletin 2012/09 - European Patent Office

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(A61K) I.1(2)<br />

(74) Carpmaels & Ransford, One Southampton<br />

Row, London WC1B 5HA, GB<br />

(62) 05745707.9 / 1 750 696<br />

A61K 31/337 → (51) A61K 9/51<br />

A61K 31/343 → (51) A61K 31/335<br />

A61K 31/343 → (51) C07C 235/46<br />

A61K 31/351 → (51) C07C 235/46<br />

A61K 31/352 → (51) A61P 35/00<br />

A61K 31/353 → (51) A61K 31/335<br />

A61K 31/353 → (51) A61K 31/513<br />

A61K 31/353 → (51) A61K 45/06<br />

A61K 31/353 → (51) A61P 35/00<br />

A61K 31/357 → (51) C07C 235/46<br />

A61K 31/36 → (51) C07C 235/46<br />

A61K 31/381 → (51) C07C 235/46<br />

A61K 31/382 → (51) C07D 495/04<br />

A61K 31/40 → (51) A61K 9/00<br />

A61K 31/40 → (51) C07C 43/225<br />

A61K 31/40 → (51) C07C 235/46<br />

A61K 31/4015 → (51) C07C 43/225<br />

A61K 31/402 → (51) C07C 235/46<br />

A61K 31/4025 → (51) C12P 17/16<br />

A61K 31/403 → (51) C07D 2<strong>09</strong>/14<br />

A61K 31/4035 → (51) C07C 235/46<br />

A61K 31/404 → (51) A61P 35/00<br />

A61K 31/404 → (51) C07C 235/46<br />

A61K 31/405 → (51) C07D 2<strong>09</strong>/14<br />

A61K 31/41 → (51) C07C 235/46<br />

A61K 31/415 → (51) C07C 235/46<br />

A61K 31/416 → (51) A61K 31/335<br />

A61K 31/421 → (51) C07C 235/46<br />

A61K 31/427 → (51) C07D 277/20<br />

A61K 31/4365 → (51) C07D 495/04<br />

A61K 31/437 → (51) A61K 31/192<br />

(51) A61K 31/44 (11) 2 422 782 A1<br />

(25) En (26) En<br />

(21) 11168901.4 (22) 11.04.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR LV MK YU<br />

(30) <strong>09</strong>.04.2004 US 560894<br />

08.04.2005 US 102559<br />

(54) Verfahren zur Verwendung von Aminopyrin-Zusammensetzungen<br />

mit verzögerter<br />

Freisetzung<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

Methods of Using Sustained Release<br />

Aminopyridine Compositions<br />

Utilisation de compositions d'aminopyridine<br />

à libération soutenue<br />

(71) Acorda Therapeutics, Inc., 15 Skyline Drive,<br />

Hawthorne NY 10531, US<br />

(72) Blight, Andrew R., Mahopac, NY 10541, US<br />

Cohen, Ron, Irvington, NY 10533, US<br />

(74) Carpmaels & Ransford, One Southampton<br />

Row, London WC1B 5HA, GB<br />

(62) 05732613.4 / 1 732 548<br />

A61K 31/44 → (51) A61K 31/513<br />

A61K 31/44 → (51) C07D 213/65<br />

A61K 31/4406 → (51) A61K 45/00<br />

A61K 31/4412 → (51) A61K 31/192<br />

A61K 31/4418 → (51) C07D 213/65<br />

A61K 31/443 → (51) C07D 213/65<br />

A61K 31/4433 → (51) C07D 213/65<br />

A61K 31/4439 → (51) C07D 213/65<br />

A61K 31/454 → (51) C07D 2<strong>09</strong>/14<br />

A61K 31/454 → (51) C07D 277/20<br />

A61K 31/47<strong>09</strong> → (51) C07D 277/20<br />

A61K 31/47<strong>09</strong> → (51) C07D 401/12<br />

A61K 31/472 → (51) C07D 217/22<br />

A61K 31/4725 → (51) C07D 217/22<br />

(51) A61K 31/496 (11) 2 422 783 A1<br />

A61K 9/20 A61K 47/10<br />

A61K 47/26 A61K 47/38<br />

C07D 417/12<br />

(25) En (26) En<br />

(21) 11181100.6 (22) 26.05.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

(30) 26.05.2005 JP 2005153508<br />

(54) Pharmazeutische Zusammensetzung<br />

Pharmaceutical Composition<br />

Composition pharmaceutique<br />

(71) Dainippon Sumitomo Pharma Co., Ltd., 6-8,<br />

Dosho-machi 2-chome Chuo-ku Osaka-shi,<br />

Osaka 541-8524, JP<br />

(72) Fujihara, Kazuyuki, Ibaraki-shi, Osaka 567-<br />

0878, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(62) 06746900.7 / 1 884 242<br />

A61K 31/496 → (51) A61K 9/12<br />

A61K 31/496 → (51) C07D 277/20<br />

(51) A61K 31/513 (11) 2 422 784 A1<br />

A61K 31/216 A61P 35/00<br />

A61K 31/353<br />

(25) En (26) En<br />

(21) 10173256.8 (22) 18.08.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

BA ME RS<br />

(54) Zusammensetzung aus TEGAFUR und<br />

Kaffeinsäurephenethyl-Ester (CAPE) und<br />

entweder Catechin, Kaempherol, Myrecetin<br />

oder Luteolin zur Potenzierung der<br />

203<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />

Antitumor-Wirkung und zur Behandlung<br />

von Tumoren<br />

Composition of TEGAFUR, caffeic acid<br />

phenethyl ester (CAPE) and either<br />

catechin, kaempherol, myricetin or luteolin<br />

for potentiating antitumour effect and for<br />

treating tumours<br />

Composition de TEGAFUR et d'ester<br />

phénéthylique de l'acide caféique (CAPE)<br />

en combinaison avec de catéchine, de<br />

caempherol, de myricetine ou de luteoline<br />

pour augmenter l'effet anti-tumeur et pour<br />

traiter des tumeurs<br />

(71) Grindeks, a joint stock company, 53,<br />

Krustpils Street, 1057 Riga, LV<br />

(72) Kalvins, Ivars, 1006 Riga, LV<br />

Stonans, Ilmars, 1057 Riga, LV<br />

Sestakova, Irina, 1006 Riga, LV<br />

Domracova, Ilona, 1006 Riga, LV<br />

Jascenko, Elina, 1006 Riga, LV<br />

Bridane, Veronika, 1006 Riga, LV<br />

Kanepe, Iveta, 1006 Riga, LV<br />

(51) A61K 31/513 (11) 2 422 785 A1<br />

A61K 31/44 A61P 35/00<br />

A61P 43/00 C07D 405/02<br />

(25) Ja (26) En<br />

(21) 10767135.6 (22) 22.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/057176 22.04.2010<br />

(87) WO 2010/123078 2010/43 28.10.2010<br />

(30) 22.04.20<strong>09</strong> JP 20<strong>09</strong>104189<br />

(54) VERFAHREN ZUR VORHERSAGE DER<br />

WIRKSAMKEIT VON CHEMOTHERAPIE<br />

BEI NIERENZELLKARZINOM<br />

METHOD FOR PREDICTING THERA-<br />

PEUTIC EFFECT OF CHEMOTHERAPY ON<br />

RENAL CELL CANCER<br />

PROCÉDÉ DE PRÉDICTION DE L'EFFET<br />

THÉRAPEUTIQUE D'UNE CHIMIOTHÉ-<br />

RAPIE SUR UN CANCER À CELLULES<br />

RÉNALES<br />

(71) Taiho Pharmaceutical Co., Ltd., 1-27,<br />

Kandanishiki-cho, Chiyoda-ku, Tokyo 101-<br />

8444, JP<br />

(72) AKAZA, Hideyuki, Tokyo 160-0023, JP<br />

NAITO, Seiji, Fukuoka-shi Fukuoka 810-<br />

0053, JP<br />

OKA, Toshinori, Tokushima-shi Tokushima<br />

771-0194, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

A61K 31/513 → (51) A61K 45/06<br />

A61K 31/513 → (51) A61P 35/00<br />

A61K 31/513 → (51) C07D 401/04<br />

A61K 31/525 → (51) A61K 9/20<br />

A61K 31/53 → (51) A61K 31/05<br />

A61K 31/536 → (51) C07D 265/26<br />

A61K 31/5377 → (51) C07D 277/20<br />

A61K 31/5377 → (51) C07D 401/04<br />

(51) A61K 31/538 (11) 2 422 786 A1<br />

A61P 11/06<br />

(25) De (26) De<br />

(21) 11187038.2 (22) 18.04.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO<br />

SE SI SK TR<br />

(30) 07.02.2005 EP 05002496<br />

22.04.2004 DE 102004019540

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