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(12) PATENT APPLICATION PUBLICATION (21) Application No.6273/DELNP/2008 A (19) INDIA (22) Date of filing of Application :18/07/2008 (43) Publication Date : 24/10/2008 (54) Title of the invention : THIAZOLES AS 11 BETA-HSD1 INHIBITORS (51) International classification : C07D 277/56 (71)Name of Applicant : (31) Priority Document No :60/759,676 1)F. HOFFMANN-LA ROCHE AG (32) Priority Date :18/01/2006 Address of Applicant :GRENZACHERSTRASSE 124, CH- (33) Name of priority country :U.S.A. 4070 BASEL, SWITZERLAND. (86) International Application No :PCT/EP2007/050141 (72)Name of Inventor : Filing Date :08/01/2007 1)GILLESPIE,PAUL (87) International Publication No :WO 2007/082808 2)GOODNOW JR. ROBERT ALAN (61) Patent of Addition to Application Number Filing Date :NA :NA 3)KOWALCZYK, AGNIESZKA 4)LE, KANG 5)ZHANG, QIANG (62) Divisional to Application Number :NA Filing Date :NA (57) Abstract : Provided herein are compounds of the formula (I): as well as pharmaceutically acceptable salts thereof, wherein the substituents are as those disclosed in the specification. These compounds, and the pharmaceutical compositions containing them, are useful for the treatment of diseases such as, for example, type II diabetes mellitus and metabolic syndrome. No. of Pages : 114 No. of Claims : 24 The Patent Office Journal 24/10/2008 25734
(12) PATENT APPLICATION PUBLICATION (21) Application No.6274/DELNP/2008 A (19) INDIA (22) Date of filing of Application :18/07/2008 (43) Publication Date : 24/10/2008 (54) Title of the invention : CYCLOHEXYL SULFONAMIDE DERIVATIVES HAVING H3 RECEPTOR ACTIVITY (51) International classification :C07D 213/71 (71)Name of Applicant : (31) Priority Document No :06100701.9 1)F.HOFFMANN-LA ROCHE AG (32) Priority Date :23/01/2006 Address of Applicant :GRENZACHERSTRASSE 124, CH- (33) Name of priority country :EPO 4070 BASEL, SWITZERLAND. (86) International Application No :PCT/EP2007/050279 (72)Name of Inventor : Filing Date :12/01/2007 1)NETTEKOVEN MATTHIAS (87) International Publication No :WO 2007/082840 2)ROCHE, OLIVIER (61) Patent of Addition to Application Number Filing Date :NA :NA (62) Divisional to Application Number :NA Filing Date :NA (57) Abstract : The present invention relates to compounds of formula I wherein R1 to R3 are as defined in the description and claims, and pharmaceutically acceptable salts thereof. The compounds are useful for the treatment and/or prevention of diseases which are associated with the modulation of H3 receptors. No. of Pages : 102 No. of Claims : 34 The Patent Office Journal 24/10/2008 25735
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