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CH 3NNClORWhere,R= Aryl(2Z)-3-[2-(4-chlorophenyl)-8-methyl imidazo[1,2-a]pyridine-3-yl]-1-aryl prop-2-en-1-one derivatives prepared by the condensation of 2-(4-chlorophenyl)-6-methylimidazo[1,2-a]pyridine-3-carbaldehyde with various substituted ketone in methanol.PART-II :SYNTHESIS OF 6-(2-(4-CHLOROPHENYL)-8-METHYL-1H-IMIDAZO[1,2-a]PYRIDINE-3-YL)-4-ARYL PYRIMIDINE-2(H)-ONE.Pyrimidine derivatives have been reported to possess variouspharmacological activities like antibacterial, antifungal, insecticide etc. In order toachive better potency, we have synthesized pyrimidine derivatives.CH 3NNClHNXNRWhere,R= ArylX = O,S,NH2Synopsis…..
Pyrimidine derivatives have been prepared by the reaction of (2Z)-3-[2-(4-chlorophenyl)-8-methyl imidazo[1,2-a]pyridine-3-yl]-1-aryl prop-2-en-1-one andUrea/Thiourea/Guanidine in basic media and methanol as a solvents.PART-III :SYNTHESIS OF ETHYL-6-(2-(4-CHLOROPHENYL)-8-METHYL-1H-IMIDAZO[1,2-a]PYRIDINE-3-YL)-4-ARYL-2-OXOCYCLOHEX-3-ENE-CARBOXYLATE.Cyclohexenone derivatives have been reported to possess variousPharmacological activities like antibacterial, antifungal etc. In order to achieve betterpotency, we have synthesized Cyclohexenone derivatives.CH 3ONNClCOOR 1RWhere,R= ArylR 1= Methyl,Ethyl,t-ButylCyclohexenone derivatives have been prepared by the reaction of (2Z)-3-[2-(4-chlorophenyl)-8-methyl imidazo[1,2-a]pyridine-3-yl]-1-aryl prop-2-en-1-one andMethylacetoacetate/Ethylacetoacetate/t-Butylacetoacetate with Na 2 CO 3 in acetoneas solvent.PART-IV :SYNTHESIS OF 2-(4-CHLOROPHENYL)-3-(4,5-DIHYDRO-3-ARYL-1H-PYRAZOL-5-YL)-8-METHYL-1H-IMIDAZO[1,2-a]PYRIDINE.Pyrazoline derivatives are endowed with various antimicrobial activities.3Synopsis…..
Page 3: The Sarvodaya Education Society’s
Page 6 and 7: selfless help, moral support and gu
Page 9 and 10: Introduction and Spectral studies .
Page 11: “STUDIES ON SOME HETEROCYCLICENTI
Page 15 and 16: Isoxazole derivative synthesized by
Page 17 and 18: “STUDIES ON SOMEHETEROCYCLIC ENTI
Page 19 and 20: (b) Pharmacokinetics: It is derived
Page 21 and 22: (C) Drug DevelopmentMany natural pr
Page 23 and 24: The process of drug design is exten
Page 25 and 26: (l) Non steroidal anti-inflammatory
Page 27 and 28: INTRODUCTIONThe aza-indolizine cont
Page 29 and 30: PHARMACEUTICAL IMPORTANTMuch resear
Page 31 and 32: Compd. R 1 R 2 R 3a :- H 7-Me-6,8-B
Page 33 and 34: S. Kristjan, Gudmundsson and A. Bra
Page 35 and 36: STUDIES ON IMIDAZOPYRIDINE DERIVATI
Page 37 and 38: (a) Chalcones with monoethanolamine
Page 39 and 40: Das B.P. et al. 111 have found that
Page 41 and 42: Furthermore, Alcaraz M.J, et al. 13
Page 43 and 44: REACTION SCHEMECl+ClOClOClClCH 3NH
Page 45 and 46: Instrument : SHIMADZU FTIR 8400 Spe
Page 47 and 48: SignalNo.SignalPosition(δppm)Relat
Page 49 and 50: ANTIMICROBIAL ACTIVITYProducts : Ch
Page 51 and 52: The reaction mixture was poured on
Page 53 and 54: TABLE NO.- 1A BIOLOGICAL SCREENING
Page 55 and 56: PART-IISTUDIES ON PYRIMIDINES
Page 57 and 58: The self consistent (pi)electron de
Page 59 and 60: class of dye viz. trichloro pyrimid
Page 61 and 62: ability to cleave nucleic acid targ
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SSNHNHoONOoONOo(11) (12)oOHThe Pyri
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called ABPP or bropirimine(2-amino-
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acid so that it could be utilized f
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have reported the 5-substitutedfuro
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maturation of the viral mRNA molecu
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Nevertheless, these compounds const
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OHHNCH 3Cl(CH 2 )nSNNR 2R 1N H 2NSR
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SECTION-ISTUDIES ONOXOPYRIMIDINES
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PHARMACEUTICAL IMPORTANCEIn recent
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REACTION SCHEMECH 3NNCHOCl10% KOH R
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INSTRUMENT :SHIMADZU FTIR 8400 Spec
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SignalNo.SignalPosition(δppm)Relat
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EXPERIMENTALSynthesis and therapeut
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TABLE NO.- 2(IB)PHYSICAL CONSTANTS
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INTRODUCTIONThiopyrimidine derivati
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H 3 COHNRH 3 CH 3 CNHS( IV ) R = ar
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SYNTHESIS AND THERAPEUTIC EVALUATIO
Page 97 and 98:
IR SPECTRAL STUDIES OF 6-(2-(4-CHLO
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NMR SPECTRAL STUDIES OF 6-(2-(4-CHL
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MASS SPECTRAL STUDIES OF 6-(2-(4-CH
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[F] Antimicrobial activity of 6-(2-
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SECTION-IIISTUDIES ONAMINOPYRIMIDIN
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ArCHO+ArCOCH3NaOHMethanolR R 1ONaOH
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Page 111 and 112:
IR SPECTRAL STUDIES OF 4-(2-(4-CHLO
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NMR SPECTRAL STUDIES OF 4-(2-(4-CHL
Page 115 and 116:
MASS SPECTRAL STUDIES OF 4-(2-(4-CH
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[F] Antimicrobial activity of 4-(2-
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PART-IIISTUDIES ONCYCLOHEXENONES
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2. Michael addition of chalcone wit
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Rheinheimer J. et al. 381have synth
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Page 127 and 128:
IR SPECTRAL STUDIES OF ETHYL-6-(2-(
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NMR SPECTRAL STUDIES OF ETHYL-6-(2-
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MASS SPECTRAL STUDIES OF ETHYL-6-(2
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Antimicrobial testing was carried o
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PART-IVSTUDIES ON PYRAZOLINES
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H 2 C= CHCN + Ar - NHNH 2NArN(3) 2
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PHARMACEUTICAL IMPORTANCE :2- Pyraz
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Kadu et al. 424 and antimicrobial b
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REACTION SCHEMECH 3NNClCHO10% KOHRO
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Instrument : SHIMADZU FTIR 8400 Spe
Page 147 and 148:
SignalNo.SignalPosition(δppm)Relat
Page 149 and 150:
EXPERIMENTALSynthesis and therapeut
Page 151 and 152:
TABLE NO.- 4(B)PHYSICAL CONSTANTS O
Page 153 and 154:
INTRODUCTION:Isoxazole come under t
Page 155 and 156:
PHARMACEUTICAL IMPORTANCE :Isoxazol
Page 157 and 158:
SYNTHESISAND THERAPEUTIC EVALUATION
Page 159 and 160:
IR SPECTRAL STUDIES OF 2-(4-CHLOROP
Page 161 and 162:
NMR SPECTRAL STUDIES OF 2-(4-CHLORO
Page 163 and 164:
MASS SPECTRAL STUDIES OF 2-(4-CHLOR
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[F]Antimicrobial activity of 2-(4-c
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PART-VISTUDIES ON OXIRANES
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( iii ) Epoxidation can also been c
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Moreover, Nomura Yutaka et al. 487
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Page 175 and 176:
IR SPECTRAL STUDIES OF (3-(2-(4-CHL
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NMR SPECTRAL STUDIES OF (3-(2-(4-CH
Page 179 and 180:
MASS SPECTRAL STUDIES OF (3-(2-(4-C
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[F] Antimicrobial activity of (3-(2
Page 184 and 185:
1. J. A. Joule and K. Mills; Hetero
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37. James J. Kaminski, D. G. perkin
Page 188 and 189:
78. Ms. B. S. Hastak and B. J. Ghiy
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116. V. R. Mudalir and V. Joshi ; I
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150. S. Inoue, A. J. Saggimoto and
Page 194 and 195:
197. S. S. Bahekar, D. B. Shinde; A
Page 196 and 197:
238. A. Kreutzberger and M. Sellhei
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280. See, for example, W. H. Prusof
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326. C. W. Whitehead and J. J. Trav
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366. Nagarjan K., Shenoy S. J.; Ind
Page 204 and 205:
396. Ausra Voskiene,Vytautas Mickev
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432. Solankee Sejal; Prajapati Yoge
Page 208 and 209:
463. Mishra Ashutosh ; Jain Sanmati
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496. Kaneko Mashami, Saitoh Yutaka,
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CH 3CH 3NNClNNClORHNONRRRC 6 H 5 -
Page 214 and 215:
CH 3CH 3NNClNNClEtOOCORHNNRRRC 6 H
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