IonWorks Quattro Assay - Molecular Devices
IonWorks Quattro Assay - Molecular Devices
IonWorks Quattro Assay - Molecular Devices
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Comparison of 23 standard Nav blockers<br />
Use-Dependence<br />
Selectivity<br />
100<br />
10<br />
20th IC50<br />
1st IC50<br />
100<br />
10<br />
Nav1.2<br />
Nav1.3<br />
Nav1.7<br />
Nav1.5<br />
Nav1.5 IC50 (µM)<br />
IC 50 (µM)<br />
1<br />
tetracaine<br />
ambroxol<br />
amitriptyline<br />
dibucaine<br />
(+/-)-fluoxetine<br />
mexiletine<br />
(+/-)-reboxetine<br />
riluzole<br />
vinpocetine<br />
lamotrigine<br />
lidocaine<br />
bupivacaine<br />
imipramine<br />
clomipramine<br />
propafenone<br />
haloperidol<br />
cinnarizine<br />
verapamil<br />
amiodarone<br />
S-(+)-fluoxetine<br />
(R,R)-reboxetine<br />
R-(-)-fluoxetine<br />
(S,S)-reboxetine<br />
-140 mV<br />
-20 mV<br />
P1 P20<br />
-70<br />
5-10 Hz<br />
1<br />
tetracaine<br />
ambroxol<br />
amitriptyline<br />
dibucaine<br />
(+/-)-fluoxetine<br />
mexiletine<br />
(+/-)-reboxetine<br />
riluzole<br />
vinpocetine<br />
lamotrigine<br />
lidocaine<br />
bupivacaine<br />
imipramine<br />
clomipramine<br />
propafenone<br />
haloperidol<br />
cinnarizine<br />
verapamil<br />
amiodarone<br />
S-(+)-fluoxetine<br />
(R,R)-reboxetine<br />
R-(-)-fluoxetine<br />
(S,S)-reboxetine