32. V. Nagy, S. Vidal, K. M. Benltifa, E. Berzsényi, C. Teilhet, K. Czifrák, Gy. Batta, T. Docsa, P. Gergely, L. Somsák, J.-P. Praly, Bioorg. Med. Chem., 17 (2009) 5696-5707. 33. Benltifa, M., De Kiss, M., Isabel Garcia-Moreno, M., Ortiz Mellet, C., Gueyrard, D., Wadouachi, A., TETRAHEDRON-ASYMMETRY 20 (2009) 1817-1823. 34. Maza, S., Lopez, O., Martos, S., Maya, I., Fernandez-Bolanos, J. G., EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 30 (2009) 5239-5246. 35. É. Bokor, T. Docsa, P. Gergely, L. Somsák, Bioorg. Med. Chem., 18 (2010) 1171-1180. 36. Somsák L., Bokor É., Czifrák K., Kónya B., Kun S., Tóth, M. Magy. Kém. Folyóirat, 116 (2010) 19-30. 37. T. Docsa, K. Czifrák, Cs. Hüse, L. Somsák, P. Gergely, Mol. Med. Rep., 4 (2011) 477-481. 38. N.G. Oikonomakos, M. N. Kosmopoulou, D. D. Leonidas, E. D. Chrysina, C. Tiraidis, N. Bischler, K. E. Tsitsanou, S. E. Zographos, I. D. Kostas, and G. Eisenbrand (2006). Indirubin and indigo analogues as potential inhibitors of glycogenolysis: structural basis of glycogen phosphorylase inhibition. In Indirubin, the red shade of indigo (Meijer L., Guyard N., Skaltsounis L. & Eisenbrand G., eds) Editions “Life in Progress”, Station Biologique, Roscoff, Chapter 18, pp. 177-189. ISBN: 2-9518029-0-0. http://www.sbroscoff.fr/usr3151-editions/132-indirubin-.html 60. N. G. Oikonomakos, M. Kosmopoulou, S. E. Zographos, D. D. Leonidas, E. D. Chrysina, L. Somsák, V. Nagy, J.-P. Praly, T. Docsa, B. Tóth, P. Gergely: The binding of N-acetyl- and N-benzoyl-N’-D-glucopyranosyl ureas to glycogen phosphorylase b: Kinetic and crystallographic studies Eur. J. Biochem., 269 (2002) 1684-1696. Cover story. IF: 2.999 (2002) Cited by/Idézi: 1. Pinotsis N, Leonidas DD, Chrysina ED, Oikonomakos NG, Mavridis IM, PROTEIN SCIENCE, 12 (2003): 1914-1924. 2. Somsak L, Nagy V, Hadady Z, et al., CURRENT PHARMACEUTICAL DESIGN, 9 (2003): 1177-1189. 3. Oikonomakos NG, Chrysina ED, Kosmopoulou MN, Leonidas DD, BIOCHIMICA ET BIOPHYSICA ACTA-PROTEINS AND PROTEOMICS, 1647 (2003): 325-332. 4. Maya, I.; Lopez, O.; Maza, S.; Fernandez-Bolanos, J. G.; Fuentes, J., Tetrahedron Letters 2003, 44, 8539-8543. 5. E. D. Chrysina, N. G. Oikonomakos, S. E. Zographos, M. N. Kosmopolou, N. Bischler, D. D. Leonidas, L. Kovács, T. Docsa, P. Gergely, L. Somsák, Biocatal. Biotransform., 21 (2003) 233-242. 6. Zea CJ, Pohl NL, ANAL BIOCHEM 327 (2004) 107-113. 7. Kristiansen M, Andersen B, Iversen LF, Westergaard N, JOURNAL OF MEDICINAL CHEMISTRY 47 (2004) 3537-3545. 8. Z. Györgydeák, Zs. Hadady, N. Felföldi, A. Krakomperger, V. Nagy, M. Tóth, A. Brunyánszki, T. Docsa, P. Gergely, L. Somsák, Bioorg. Med. Chem., 12 (2004) 4861-4870. 9. Lopez O, Maza S, Maya I, Fuentes J, Fernandez-Bolanos JG, TETRAHEDRON 61 (2005) 9058-9069. 10. Praly JP, He L, Qin BB, Tanoh M, Chen GR, TETRAHEDRON LETTERS 46 (2005) 7081-7085. 11. Anagnostou, E.; Kosmopoulou, M. N.; Chrysina, E. D.; Leonidas, D. D.; Hadjiloi, T.; Tiraidis, C.; Zographos, S. E.; Györgydeák, Z.; Somsák, L.; Docsa, T.; Gergely, P.; Kolisise, F. N.; Oikonomakos, N. G. Bioorganic and Medicinal Chemistry 2006, 14, 181-189. 12. G. Archontis, K. A. Watson, Q. Xie, G. Andreou, E. D. Chrysina, S. E. Zographos, N. G. Oikonomakos, M. Karplus, PROTEINS: Structure, Function, and Bioinformatics 61 (2005) 984–998. 13. Kimberly A. Watson, Evangelia D. Chrysina, Katerina E. Tsitsanou, Spyros E. Zographos, Georgios Archontis, George W.J. Fleet, Nikos G. Oikonomakos, PROTEINS: Structure, Function, and Bioinformatics 61 (2005) 966–983. 14. Kosmopoulou, M. N.; Leonidas, D. D.; Chrysina, E. D.; Oikonomakos, N. G.; Eisenbrand, G. Letters in Drug Design and Discovery 2005, 2, 377-390. 15. Baker DJ, Greenhaff PL, Timmons JA, EXPERT OPINION ON THERAPEUTIC PATENTS 16 (2006) 459-466. 44
16. K. Czifrák, Zs. Hadady, T. Docsa, P. Gergely, J. Schmidt, L. Wessjohann, L. Somsák, Carbohydr. Res., 341 (2006) 947-956. 17. Hadjiloi, T.; Tiraidis, C.; Chrysina, E. D.; Leonidas, D. D.; Oikonomakos, N. G.; Tsipos, P.; Gimisis, T. Bioorganic & Medicinal Chemistry 2006, 14, 3872-3882. 18. Menuel S, Porwanski S, Marsura A., NEW JOURNAL OF CHEMISTRY 30 (2006) 603-608. 19. Lukacs CM, Oikonomakos NG, Crowther RL, Hong LN, Kammlott RU, Levin W, Li S, Liu CM, Lucas- McGady D, Pietranico S, Reik L, PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS 63 (2006) 1123-1126. 20. Benltifa M, Vidal S, Gueyrard D, Goekjian PG, Msaddek M, Praly JP, Tetrahedron Lett., 47 (2006) 6143- 6147. 21. Benltifa, M.; Vidal, S.; Fenet, B.; Msaddek, M.; Goekjian, P. G.; Praly, J.-P.; Brunyánszki, A.; Docsa, T.; Gergely, P., European Journal of Organic Chemistry 2006, 4242-4256. 22. He, L., Zhang, Y.-Z., Tanoh, M., Chen, G.-R., Praly, J.-P., Chrysina, E. D., Tiraidis, C., Kosmopoulou, M., Leonidas, D. D., Oikonomakos, N. G., EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2007) 596- 606. 23. Chen, L., Li, H., Liu, J., Zhang, L., Liu, H., Jiang, H., BIOORGANIC & MEDICINAL CHEMISTRY 15 (2007) 6763-6774. 24. Aouadi, K., Jeanneau, E., Msaddek, M., Praly, J.-P., SYNTHESIS-STUTTGART (2007) 3399-3405. 25. Chen, G.-R., Praly, J.-P. Comptes Rendus Chimie, 11 (2008) 19-28. 26. Oikonomakos NG, Somsak L, CURRENT OPINION IN INVESTIGATIONAL DRUGS 9 (2008) 379-395. 27. Khan, M. T. H., Top. Heterocycl. Chem., 2007, 9, 33-52. 28. Aouadi, K., Jeanneau, E., Msaddek, M., Praly, J.-P. TETRAHEDRON-ASYMMETRY 19 (2008) 1145- 1152. 29. L. Somsák, N. Felföldi, B. Kónya, Cs. Hüse, K. Telepó, É. Bokor, K. Czifrák, Carbohydr. Res., 343 (2008) 2083-2093. 30. Bertus, P., Szymoniak, J., Jeanneau, E., Docsa, T., Gergely, P., Praly, J.-P., Vidal, S., BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 18 (2008) 4774-4778. 31. Spanu, P., Ulgheri, F., CURRENT ORGANIC CHEMISTRY, 12 (2008) 1071-1092. 32. M. Bols, Ó. López, F. Ortega-Caballero Glycosidase Inhibitors: Stucture, Activity, Synthesis, and Medical Relevance in Comprehensive Glycoscience (Ed. J. P. Kamerling), Elsevier, 2007, Vol. 1. pp. 815-882. 33. L. Somsák, V. Nagy, S. Vidal, K. Czifrák, E. Berzsényi, J.-P. Praly, Bioorg. Med. Chem. Lett., 18 (2008) 5680-5683. 34. Ulgheri F, Giunta D, Spanu P, TETRAHEDRON 64 (2008) 11768-11775. 35. L. Somsák, K. Czifrák, M. Tóth, É. Bokor, E. D. Chrysina, K.-M. Alexacou, J. M. Hayes, C. Tiraidis, E. Lazoura, D. D. Leonidas, S. E. Zographos, N. G. Oikonomakos, Curr. Med. Chem., 15 (2008) 2933-2983. 36. Aouadi, K., Lajoix, A.-D., Gross, R., Praly, J.-P., EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, (2009) 61-71. 37. Cecioni, S., Argintaru, O.-A., Docsa, T., Gergely, P., Praly, J.-P., Vidal, S., New Journal of Chemistry, 33 (2009) 148-156. 38. M. Tóth, S. Kun, É. Bokor, M. Benltifa, G. Tallec, S. Vidal, T. Docsa, P. Gergely, L. Somsák, J.-P. Praly, Bioorg. Med. Chem., 17 (2009) 4773-4785. 39. E. D. Chrysina, É. Bokor, K.-M. Alexacou, M.-D. Charavgi, G. N. Oikonomakos, S. E. Zographos, D. D. Leonidas, N. G. Oikonomakos, L. Somsák, Tetrahedron Asymmetry, 20 (2009) 733-740. 40. V. Nagy, S. Vidal, K. M. Benltifa, E. Berzsényi, C. Teilhet, K. Czifrák, Gy. Batta, T. Docsa, P. Gergely, L. Somsák, J.-P. Praly, Bioorg. Med. Chem., 17 (2009) 5696-5707. 41. Motoshima, K., Ishikawa, M., Sugita, K., Hashimoto, Y., BIOLOGICAL & PHARMACEUTICAL BULLETIN, 32 (2009) 1618-1620. 42. É. Bokor, T. Docsa, P. Gergely, L. Somsák, Bioorg. Med. Chem., 18 (2010) 1171-1180. 43. N. Felföldi, M. Tóth, E. D. Chrysina, M.-D. Charavgi, K.-M. Alexacou, L. Somsák,Carbohydr. Res., 345 (2010) 208-213. 44. Yagodkin, A., Loschcke, K., Weisell, J., Azhayev, A., TETRAHEDRON, 66 (2010) 2210-2221. 45. Somsák L., Bokor É., Czifrák K., Kónya B., Kun S., Tóth, M. Magy. Kém. Folyóirat, 116 (2010) 19-30. 46. Antus, S. Acta Pharm. Hung., (2010) 3-17. 47. Chrysina, E. D., Mini Rev. Med. Chem., 10 (2010) 1093-1101. 48. J.-P. Praly, S. Vidal, Mini Rev. Med. Chem., 10 (2010) 1102-1126. 45
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- Page 19 and 20: 34. Sipos Szabolcs; Jablonkai Istva
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- Page 33 and 34: 16. Marinov M, Minchev S, Stoyanov
- Page 35 and 36: 37. Agnihotri G, Misra AK, CARBOHYD
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- Page 57 and 58: synthesis and enzymatic evaluation
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