Chapter 6 Synthesis of benzodiazepines 26. Sabitha, G.; Reddy, G. S. K. K.; Reddy, K. B.; Reddy, N. M.; Yadav, J. S.; Adv. Synth. Catal., 2004, 346, 921. 27. Yadav, J. S.; Reddy, B. V. S.; Kumar, S. P.; Nagaiah, K. Synthesis., 2005, 480. 28. De, S. K.; Gibbs, R. A.; Tetrahedron Lett., 2005, 46, 1811. 29. Reddy, B. M.; Sreekanth, P. M.; Lakshmanan, P.; J. Mol. Catal. A: Chem., 2005, 237, 93. 30. Yadav, J. S.; Reddy, B.V.S.; Satheesh, G.; Srinivasulu, G.; Kunwar, A. C.; Arkivoc, 2005, iii, 221. 31. Varala, R.; Ramu, E.; Sreelatha, N.; Adapa, S. R.; Synlett, 2006, 1009. 32. Pasha, M. A.; Jayashankara,V. P.; Heterocycles, 2006, 68, 1017. 33. Katrizky, A.R.; Abonia, R.; Yang, B.; Qi, M.; Insuasty, B.; Synthesis.,1998, 1487. 34. Clifford, D. P.; Jackson, D.; Edwards, R. V.; Jefferey, P. Pestic. Sci., 1976, 7,453. 35. Werner,W.; Wohlrabe,K.; Gutsche,W.; Jungstand, W.; Roemer, W. FolidaHaematol,1981, 108, 637. 36. Goff, D.A.; Zuckermann, R. N.; Org. Chem., 1995, 60, 5744. 37. Spencer, J.; Rathnam, R. P.; Harvey, A. L.; Clements, C. J.; Clark, R. L.; Barrett, M. P.;Wong, P. E.; Male,L.; Coles,S. J.; Mackay,S. P.; Bioorganic & Medicinal Chemistry., 2011, 19 1802. 38. Bova, F.; Ettari, R.; Micale N.; Carnovale, C.; Schirmeister,T.; Gelhaus, C.; Leippe M.; Grasso, S.; Zappalà, M.; Bioorganic & Medicinal Chemistry., 2010, 18 4928. 39. Guandalini, L.; Cellai, C.; Laurenzana, A.; Scapecchi, S.; Paoletti, F.; Romanelli, M. N.; Bioorganic & Medicinal Chemistry Letters., 2008, 18, 5071. 40. Bolli, M. H.; Marfurt, J.; Grisostomi, C.; Boss, C.; Binkert, C.; Hess, P.; Treiber, A.; Thorin, E.; Morrison.; Buchmann, K. S.; Bur, D.; Ramuz, H.; Clozel, M.; Fischli, W.;Weller, T.; J. Med. Chem., 2004, 47, 2776. 41. Pavlovsky, V. I.; Bachinskii, S. Yu.; Tkachuk, N. A.; Makan, S. Yu.; Andronati, S. A.;. Simonov, Yu. A.; Filippova, I. G.; Gdaniec, M.; Chemistry of Heterocyclic Compounds., 2007, 8, 43. 42. Buckel, D. R.; Cantello, B. V.; Morgan, N. J.; British Patent, 1460938; Chem. Abstr.,1977,87, 68438a. 43. Andronati, K. S.; Kostenko, E. A.; Karaseva, T. L.; Andronati, S. A.; Pharmaceutical Chemistry Journal., 2002, 7, 36. 44. Hemming, K.; Anwar, B.; Grimsey, P.; Krajniewski, M.; Loukou, C.; Tetrahedron Lett., 2007, 41, 10107. 45. Rubin, M. A.; Albach, C. A.; Berlese, D. B.; Braz. J. Med. Biol. Ros., 2000, 33, 1069. 46. Heitmann, W.; Liepmann, H.; Matzel, U.; Zeugner, H.; Fuchs, A. M.; Krahling, H.; Ruhland, M.; Mol, F.; Tulp, M.; Th. M.; Eur. J. Med. Chem.,1988, 23, 249. 47. Kusanur1, R. A.; Ghate, M.; Kulkarni, M. V.; J. Chem. Sci., 2004, 116, 265. 48. Pitt, G. R. W.; Batt, A. R.; Haigh, R. M.; Penson, A. M.; Robson, P. A.; Rooker, D. P.; Tartar, A. L.; Trim, J. E.; Yeaa, C. M.; Roea, M. B. Bioorg. Med. Chem. Lett., 2004, 14, 4585. Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot-360005 232
Chapter 6 Synthesis of benzodiazepines 49. Ha, S. K.; Shobha, D.; Moon, E.; Chari, M. A.; Mukkanti, K.; Kim, S. -H.; Ahn, K. -H.; Kim, S. Y.; Bioorg. Med. Chem. Lett., 2010, 20, 3969. 50. Tinney, F. J.; Sanchez, J. P.; Nogas, J. A.; J. Med. Chem., 1974, 17, 624. 51. Walser, A.; Flynn, T.; Mason, C.; Crowley, H.; Maresca, C.; Yaremko, B.; O'Donnell, M.; J. Med. Chem.,1991, 34, 1209. 52. Namanishi, M.; Tahara, T.; Araki, K.; Shiroki, M.; US Patent, 3920679, 1975. 53. Carter, M. C.; Alber, D. G.; Baxter, R. C.; Bithell, S. K.; Budworth, J.; Chubb, A. G., Cockerill, S.; Verity C. L.; Dowdell, E. A.; Henderson, S. J.; Keegan, R. D.; Kelsey, M. J.; Lockyer, J. N.; Stables, L. J.; Wilson, K. L., Powell, J. Med. Chem., 2006, 49, 2311. 54. Sternbach, L. H., Fryer, R. I., Metlesics, W., Reeder, E., Sach, G., Saucy, G., Stemple, A.; J. Org. Chem., 1962, 27, 3788. 55. Lednicer, D.; The Organic Chemistry of Drug Synthesis; Wiley-Interscience: New-York, 1998. 56. Lednicer, D.; Mitschev, L. A.; The Organic Chemistry of Drug Synthesis; Wiley-Interscience: New York, 1977. 57. Wang, J.Y.; FeiGuo, X.; Wang, D. X.; Huang, Z. T.; Wang, M.X.; J. Org. Chem., 2008, 73, 1979. 58. Joshua, D.; Neukom, A. S.; Aquino, J. P.; Wolfe.; Org. Lett., 2011, 13, 9. 59. Yadav, V.; Yadav, N.; Arch. Appl. Sci. Res., 2011, 3 (1), 139. 60. Laustsen, L S.; Sams,C. K.; J. Comb. Chem., 2007, 9, 1094. 61. Bhatia, M. S.; Choudhari, P. B.; Ingale, K. B.; Oriental J. Chem., 2008, 24, 147. 62. Alizadeh, A.; Zohreh, N.; Helv.Chim.Acta., 2010, 93, 1221. 63. Goswami, P.; Das, B.; Synth. Commu., 2010, 40, 1685. Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot-360005 233
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